Substituted aminomethylphenylsulfonylureas their preparation and their use as herbicides and plant growth regulators

ABSTRACT

Substituted aminomethylphenylsulfonylureas, their preparation, and their use as herbicides and plant growth regulators 
     Compounds of the formula (I) and salts thereof ##STR1## where R 1  to R 7  and A are as defined in claim 1 and, inter alia, F 5  is an acyl radical or NR 4  R 5  together are a heterocyclic radical, are useful as herbicides and plant growth regulators. They can be prepared by the methods of known processes, using novel intermediates of the formula (II), (IV), (VI) or (VII) (cf. claim 5).

DESCRIPTION

Substituted aminomethylphenylsulfonylureas, their preparation, and their use as herbicides and plant growth regulators

Some phenylsulfonylureas are known to have herbicidal and plant growth regulating properties; cf. U.S. Pat. Nos. 4,786,314, 4,927,453, WO 89/10921 and WO 951/10507 (=ZA 94/8063). However, some of these compounds have practical disadvantages, for example a high persistency or insufficient selectivity in important crop plants or a very limited spectrum of harmful plants which can be controlled.

There have now been found novel phenylsulfonylureas having specific radicals at the phenyl ring which can advantageously be employed as herbicides and plant growth regulators.

The present invention relates to a compound of the formula (I) or a salt thereof ##STR2## where R¹ is NR⁸ R⁹ or an unsubstituted or substituted hydrocarbon radical preferably containing inclusive of substituents 1 to 20 carbon atoms,

n is 0, 1 or 2, excluding n=0 or 1 if R¹ =NR⁸ R⁹,

R² and R³ are each independently of the other H or (1-4)alkyl,

R⁴ is H, OH, formyl, or a radical of the formula R, R--O--, R--CO-- or R--SO₂ --, R being an unsubstituted or substituted hydrocarbon radical preferably having inclusive of substituents 1 to 20 carbon atoms,

R⁵ is an acyl radical or

NR⁴ R⁵ together are an unsubstituted or substituted heterocyclic radical preferably containing inclusive of substituents 2 to 12 carbon atoms and in particular an electron-withdrawing radical owing to substituents of the heterocycle at the nitrogen atom of the group NR⁴ R⁵,

W is an oxygen or sulfur atom, R⁶ is H, (1-4)alkyl, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkyl!-carbonyl or (1-4)alkoxy!carbonyl, each of the last radicals being unsubstituted or substituted by one or more halogen atoms, or halogen, NO₂, CN or mono- or disubstituted amino,

R⁷ is H or (1-4)alkyl,

R⁸ and R⁹ are each independently of the other H, (1-4)alkyl,, (1-4)alkoxy, (1-4)alkyl!carbonyl or (1-4)alkylsulfonyl,

A is a radical of the formula ##STR3## one of the radicals X and Y being hydrogen, (1-3)alkyl or (1-3)alkoxy, the last two radicals being unsubstituted or mono- or polysubstituted by halogen or monosubstituted by (1-3)alkoxy, and the other of the radicals X and Y being hydrogen, halogen, (1-3)alkyl,

(1-3)alkoxy or (1-3)alkylthio, the last three alkyl-containing radicals being unsubstituted or mono- or polysubstituted by halogen or mono- or disubstituted by (1-3)alkoxy or (1-3)alkylthio, or a radical of the formula NR^(a) R^(b), where R^(a) and R^(b), independently of each other, are H, (1-3)alkyl or (1-3)alkenyl, or (3-6)cycloalkyl, (2-4)alkenyl, (2-4)alkynyl, (3-4)-alkenyloxy or (3-4)alkynyloxy,

Z isCH or N,

X¹ is CH₃, OCH₃, OC₂ H₅ or OCHF₂, Y¹ is --O-- or --CH₂ --,

X² is CH₃, C₂ H₅ or CH₂ CF₃,

Y² is OCH₃, OC₂ H₅, SCH₂ CH₃, CH₃ or C₂ H₅,

X³ is CH₃ or OCH₃,

Y³ is H or CH₃,

X⁴ is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃ or Cl,

Y⁴ is CH₃, OCH₃, OC₂ H₅ or Cl and

Y⁵ is CH₃, C₂ H₅, OCH₃ or Cl.

The definitions of general radicals having carbon atoms in formula (I) often contain ranges or specific numbers for the number of possible carbon atoms. The range or number of carbon atoms is stated as a prefix in brackets prior to the term of the general chemical group; thus, for example, (1-4)alkyl is an alkyl radical having 1 to 4 carbon atoms; or (1-4)haloalkyl is a haloalkyl having 1 to 4 carbon atoms in the alkyl moiety or alkyl skeleton; (1)alkyl is synonomous to methyl; and the general definition unsubstituted (3) alkyl thus includes n-propyl and i-propyl.

The compounds of the formula (I) can form salts where the hydrogen of the --SO₂ --NH-- group is replaced by an agriculturally useful cation. These salts are, for example, metal salts, in particular alkali metal salts or alkaline earth metal salts, in particular sodium salts and potassium salts, or else ammonium salts or salts with organic amines. Salt formation can also be carried out by addition of an acid to basic groups, such as amino and alkyamino. Suitable acids in this context are strong inorganic and organic acids, for example HCl, HBr, H₂ SO₄ or HNO₃.

In formula (I) and all subsequent formulae, the radicals alkyl, alkoxy, haloalkyl, haloalkoxy, alkylamino and alkylthio and the corresponding unsaturated and/or substituted radicals can be in each case straight-chain or branched in the carbon skeleton. Unless specifically indicated, the lower carbon skeletons, for example those having 1 to 6 carbon atoms or, in the case of unsaturated groups, 2 to 6 carbon atoms, are preferred for these radicals. Alkyl radicals, also in the composite meanings such as alkoxy, haloalkyl and the like, are, for example, methyl, ethyl, n- or i-propyl, n-, i-, t- or 2-butyl, pentyls, hexyls, such as n-hexyl, i-hexyl and 1,3-dimethylbutyl, heptyls, such as n-heptyl, i -methylhexyl and 1,4-dimethylpentyl; alkenyl and alkynyl radicals have the meanings of the unsaturated radicals which are possible and which correspond to the alkyl radicals; alkeanyl is, for example, allyl, 1-methylprop-2-en-1-yl, 2-methylprop-2-en-1-yl, but-2-en-1-yl, but-3-en-1-yl, 1-methylbut-3-en-1-yl and 1-methylbut-2-en-1-yl; alkynyl is, for example, propargyl, but-2-yn-1-yl, but-3-yn-1-yl, 1-methylbut-3-yn-1-yl.

Cycloalkyl is a carbocyclic saturated ring system having for example 3-8 carbon atoms, for example cycopropyl, cyclopantyl or cyclohexyl.

Alkenyl in the form of "(3-4)alkenyl" or "(3-6)alkenyl" is preferably an alkenyl radical having 3 to 4 or 3 to 6 carbon atoms in which the double bond is not positioned at the carbon atom attached to the remainder of the molecule of the compound (I) ("yl" position). The same applies analogously to (3-4)-alkynyl, etc.

Halogen is, for example, fluorine, chlorine, bromine or iodine. Haloalkyl, -alkenyl and -alkynyl are alkyl, alkenyl and alkynyl, respectively, which are partially or fully substituted by halogen, preferably by fluorine, chlorine and/or bromine, in particular by fluorine or chlorine, for example CF₃, CHF₂, CH₂ F, CF₃ CF₂, CH₂ FCHCl, CCl₃, CHCl₂, CH₂ CH₂ Cl; haloalkoxy is, for example, OCF3, OCHF₂, OCH₂ F, CF₃ CF₂ O, OCH₂ CF₃ and OCH₂ CH₂ Cl; the same applies analogously to haloalkenyl and other halogen-substituted radicals.

A hydrocarbon radical is a straight-chain, branched or cyclic saturated or unsaturated aliphatic or aromatic hydrocarbon radical, for example alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or aryl; aryl is, in this context, a mono-, bi- or polycyclic aromatic system, for example phenyl, naphthyl, tetrahydronaphthyl, indenyl, indanyl, pentalenyl, fluorenyl and the like, preferably phenyl; a hydrocarbon radical is preferably alkyl, alkenyl or alkynyl having up to 12 carbon atoms or cycloalkyl having 3, 4, 5, 6 or 7 ring atoms, or phenyl; the same applies analogously to a hydrocarbon radical in a hydrocarbon-oxy radical.

A heterocyclic radical or ring (heterocyclyl) may be saturated, unsaturated or heteroaromatic; it preferably contains one or more hetero units in the ring, preferably selected from the group consisting of N, O, S, SO, SO₂ ; it is preferably an aliphatic heterocyclyl radical having 3 to 7 ring atoms or a heteroaromatic radical having 5 or 6 ring atoms and contains 1, 2 or 3 hetero units. For example, the heterocyclic radical may be a heteroaromatic radical or ring (heteroaryl), for example a mono-, bi- or polycyclic aromatic system in which at least 1 ring contains one or more hetero atoms, for example pyridyl, pyrimidinyl, pyridazinyl, pyrazinyl, thienyl, thiazolyl, oxazolyl, furyl, pyrrolyl, pyrazolyl and imidazolyl, or it is a partially or fully hydrogenated radical such as oxiranyl, pyrrolidyl, piperidyl, piperazinyl, dioxolanyl, morpholinyl, tetrahydrofuryl. Suitable substituents for a substituted heterocyclic radical are the substituents mentioned further below, and additionally also oxo. The oxo group may also be located on the hetero ring atoms which can exist at various oxidation levels, for example in the case of N and S.

Substituted radicals, such as substituted hydrocarbon radicals, for example substituted alkyl, alkenyl, alkynyl, aryl, phenyl and benzyl, or substituted heterocyclyl or heteroaryl, are, for example, a substituted radical which is derived from the unsubstituted skeleton, the substituents being, for example, one or more, preferably 1, 2 or 3, radicals selected from the group consisting of halogen, alkoxy, haloalkoxy, alkylthio, hydroxyl, amino, nitro, carboxyl, cyano, azido, alkoxycarbonyl, alkylcarbonyl, formyl, carbamoyl, mono- and dialkylaminocarbonyl, substituted amino, such as acylamino, mono- and dialkylamino, and alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl and, in the case of cyclic radicals, also alkyl and haloalkyl; and unsaturated aliphatic radicals, such as alkenyl, alkynyl, alkenyloxy, alkynyloxy and the like, corresponding to the abovementioned saturated hydrocarbon-containing radicals. Amongst radicals having carbon atoms, those having 1 to 4 carbon atoms, in particular 1 or 2 carbon atoms are preferred. Preferred are, as a rule, substituents selected from the group consisting of halogen, for example fluorine and chlorine, (1-4)alkyl, preferably methyl or ethyl, (1-4)haloalkyl, preferably trifluoromethyl, (1-4)alkoxy, preferably methoxy or ethoxy, (1-4)haloalkoxy, nitro and cyano. Especially preferred in this context are the substituents methyl, methoxy and chlorine.

Mono- or disubstituted amino is a chemically stable radical selected from the group consisting of the substituted amino radicals which are H-substituted, for example, by one or two identical or different radicals selected from the group consisting of alkyl, alkoxy, acyl and aryl; preferably monoalkylamino, dialkylamino, acylamino, arylamino, N-alkyl-N-arylamino and N-heterocycles; preferred in this context are alkyl radicals having 1 to 4 carbon atoms; aryl is, in this context, preferably phenyl or substituted phenyl; acyl is as defined further below, preferably (1-4)alkanoyl. The same applies analogously to substituted hydroxylamino or hydrazino.

Optionally substituted phenyl is preferably phenyl which is unsubstituted or mono- or polysubstituted, preferably up to trisubstituted, by identical or different radicals selected from the group consisting of halogen, (1-4)alkyl, (1-4)alkoxy, (1-4)haloalkyl, (1-4)haloalkoxy and nitro, for example o-, m- and p-tolyl, dimethylphenyls, 2-, 3- and 4-chlorophenyl, 2-, 3- and 4-trifluoro- and -trichlorophenyl, 2,4-, 3,5-, 2,5- and 2,3-dichlorophenyl, o-, m- and p-methoxyphenyl.

An acyl radical is the radical of an organic acid, for example the radical of a carbonylic acid and radicals of acids derived therefrom, such as thiocarboxylic acid, optionally N-substituted iminocarboxylic acids or the radical of carboxylic monoesters, or of optionally N-substituted carbamic acid, of sulfonic acids, sulfinic acids, phosphonic acids and phosphinic acids. Acyl is, for example, formyl, alkylcarbonyl such as (1-4)alkyl!-carbonyl, phenylcarbonyl, it being possible for the phenyl ring to be substituted as demonstrated above for example for phenyl, or alkyloxycarbonyl, phenyloxycarbonyl, benzyloxycarbonyl, alkylsulfonyl, alkylsulfinyl, N-alkyl-1-iminoalkyl and other radicals of organic acids.

The invention also relates to all stereoisomers which are embraced by formula (I) and to their mixtures. Such compounds of the formula (I) contain one or more asymmetric carbon atoms or else double bonds which are not separately indicated in formula (I). The sterecisomers which are possible and which are defined by their specific spatial form, such as enantiomers, diastereomers and Z and E isomers, are all embraced by formula (I) and can be obtained from mixtures of the sterecisomers by customary methods, or else prepared by stereoselective reactions in combination with the use of stereochemically pure starting materials.

The abovementioned examples of radicals or ranges of radicals included in general terms such as "alkyl", "acy", "substituted radicals", etc. are not a complete enumeration. The general terms include in particular also the definitions of ranges of radicals in groups of preferred compounds listed further below, in particular ranges of radicals including specific radicals from the examples in the tables.

Compounds of the formula (I) or salts thereof according to the invention which are of particular interest, mainly because of more potent herbicidal activity, better selectivity and/or because they can be prepared more easily, are those in which

R¹ is NR⁸ R⁹, (1-6)alkyl, (2-6)alkenyl, (2-6)alkynyl, (3-6)cycloalkyl, (3-6)cycloalkenyl or phenyl, each of the last 6 radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, CN, (1-4)alkoxy, (1-4)haloalkoxy, (1-4)alkoxy(1-4)alkoxy, (1-4)alkylthio, (1-4)alkylsulfinyl, (1-4)-alkylsulfonyl, formyl, (1-4)alkyl!-carbonyl, (1-4)alkoxy!carbonyl, (1-4)alkyl!carbonyloxy and in the case of cyclic radicals also (1-4)alkyl, (1-4)haloalkyl and (1-4)alkoxy-(1-4)alkyl,

n is 0, 1 or 2, excluding n=0 or 1 if R¹ =NR⁸ R⁹,

R² and R³ are each independently of the other H or (1-4)alkyl,

R⁴ is H, OH, formyl, (1-6)alkyl, (2-6)alkenyl, (2-6)alkynyl, (1-6)alkoxy, (2-5)alkenyloxy, (2-5)alkynyloxy, (1-6)alkyl!-carbonyl, (1-6)alkylsulfonyl, (2-6)alkenyl!carbonyl, (2-6)alkenylsulfonyl, (2-6)alkynyl!carbonyl, (2-6)alkynylsulfonyl, (3-6)cycloalkyl, (3-6)cycloalkenyl, (3-6)cycloalkyl!carbonyl, (3-6)cycloalkylsulfonyl, (3-6)cycloalkenyl!carbonyl or (3-6)cycloalkenylsulfonyl, each of the last 18 radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkylsulfinyl, (1-4)alkylsulfonyl, (1-4)alkoxyl!carbonyl, (1-4)alkyl!carbonyl, (1-4)alkylicarbonyloxy and CN and in the case of cyclic radicals also (1-4)alkyl and (1-4)haloalkyl, or phenylcarbonyl or phenylsulfonyl, the phenyl ring in the two last radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, CN, NO₂, (1-4)alkyl, (1-4)haloalkyl, (1-4)alkoxy and (1-4)haloalkoxy, and

R⁵ is CHO, (1-6)alkyl!carbonyl, (2-6)alkenyl!carbonyl, (2-6)alkynyl!carbonyl, (1-6)alkylsulfonyl, (2-6)alkenylsulfonyl, (2-6)alkynysulfonyl, (3-6)cycloalkyl!carbonyl, (3-6)cycloalkenyl!carbonyl, (3-6)cycloalkylsulfonyl or (3-6)cycloalkenylsulfonyl, each of the last 10 radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkylsulfinyl (1-4)alkylsulfonyl, (1-4)alkyl!-carbonyl, (1-4)alkoxy!carbonyl, (1-4)alkyl!carbonyloxy and CN and in the case of cyclic radicals also (1-4)alkyl and (1-4)haloalkyl, or phenylcarbonyl or phenylsulfonyl, each of the last two radicals being unsubstituted in the phenyl ring or substituted by one or more radicals from the group consisting of halogen, CN, NO₂, (1-4)alkyl, (1-4)haloalkyl, (1-4)alkoxy and (1-4)haloalkoxy, or mono- or di- (1-4)alkyl!aminosulfonyl which is unsubstituted in the alkyl moiety or substituted by one or more radicals from the group consisting of halogen, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkylsulfinyl, (1-4)alkyl!-carbonyl, (1-4)alkyl!carbonyloxy, (1-4)alkoxylcarbonyl and CN or a group of the formula COCOR' where R'=H, OH, (1-4)alkoxy or (1-4)alkyl, or a group of the formula ##STR4## R⁴ and R⁵ together are a chain of the formula (--CH₂)_(m1) B¹ -- or --B¹ --(CH₂)_(m2) B² where individual groups CH₂ may be replaced by oxygen atoms and where the chain is unsubstituted or substituted by one or more (1-3)alkyl radicals or halogen and m1=3, 4 or 5 or m2=2, 3 or 4, and

W is O or S,

B¹ and B² are each independently of the other SO₂ or CO,

T is O or S,

R⁶ is H, (1-4)alkyl, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkyl!-carbonyl or (1-4)alkoxy!carbonyl, each of the last 5 radicals being unsubstituted or substituted in the alkyl moiety by one or more halogen atoms, or halogen, NO₂, CN or mono- or di- (1-4)alkyl!amino,

R⁷ H or (1-4)alkyl, preferably H or CH₃,

R⁸ is (1-4)alkyl, (1-4)alkoxy, (3-6)cycloalkyl or (3-6)cycloalkenyl,

R⁹ is H or (1-4)alkyl,

R¹⁰ is (1-4)alkyl, (3-4)alkenyl or (3-4)alkynyl, each of the last three radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkyl!carbonyl and (1-4)alkoxyl!carbonyl,

R¹¹ and R¹² are each independently of the other H, (1-4)alkyl, (3-4)alkenyl or (3-4)alkynyl, each of the last three radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkyl!carbonyl and (1-4)alkoxy!carbonyl,

the radicals R¹³ together with the nitrogen atom are a 5- to 6-membered heterocyclic ring which may contain further hetero atoms from the group consisting of N, O and S in the possible oxidation states and is unsubstituted or substituted by (1-4)alkyl or the oxo group or is benzo-fused.

Further of interest are compounds of the formula (I) and salts thereof according to the invention in which

R¹ is NR⁸ R⁹, (1-4)alkyl, (3-6)cycloalkyl or phenyl, each of the last 3 radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, CN, (1-4)alkoxy, (1-4)haloalkoxy, (1-4)alkylthio, (1-4)-alkylsulfonyl, formyl, (1-4)alkoxy!carbonyl, (1-4)alkyl!carbonyloxy and In the case of cyclic radicals also (1-4)alkyl, (1-4)haloalkyl and (1-4)alkoxy-(1-4)alkyl, or (2-4)alkenyl or (2-4)alkynyl,

n is 0, 1 or 2, excluding n=0 or 1 if R¹ =NR⁸ R⁹,

R² and R³ are each independently of the other H or (1-4)alkyl,

R⁴ H, OH, formyl, (1-4)alkyl, (2-4)alkenyl, (2-4)alkynyl, (1-4)alkoxy, (1-4)alkyl!carbonyl, (1-4)alkylsulfonyl, each of the last 6 radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen and (1-4)alkoxy, or phenylcarbonyl or phenylsulfonyl, the phenyl ring of the last two radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (1-4)alkyl, (1-4)haloalkyl, (1-4)alkoxy and (1-4)haloalkoxy, and

R⁵ is CHO, (1-4)alkyl!carbonyl, (2-4)alkenyl!carbonyl, (2-4)alkynyl!carbonyl, (1-4)alkylsulfonyl, (2-4)alkenylsulfonyl, (2-4)alkynylsulfonyl, (3-6)cycloalkyl!carbonyl, each of the last 7 radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkoxy!carbonyl, (1-4)alkyl!-carbonyloxy and CN and in the case of cyclic radicals also (1-4)alkyl and (1-4)haloalkyl, or phenylcarbonyl or phenylsulfonyl, each of the last two radicals being unsubstituted in the phenyl ring or substituted by one or more radicals from the group consisting of halogen, CN, NO₂, (1-4)alkyl, (1-4)haloalkyl, (1-4)alkoxy and (1-4)haloalkoxy, or mono- or di- (-4)alkyl!aminosulfonyl which is unsubstituted in the alkyl moiety or substituted by one or more halogen atoms, or a group of the formula COCOR'

where R'=H, OH, (1-4)alkoxy or (1-4)alkyl, or a group of the formula ##STR5## or R⁴ and R⁵ together are a chain of the formula (--CH₂)_(m1) B¹ -- or --B¹ --(CH₂)_(m2) B² --, where the chain is unsubstituted or substituted by one or more (1-3)alkyl radicals or halogen and m1=3, 4 or 5 or m2=2, 3 or 4, and

W is O or S, B¹ and B² are each independently of the other SO₂ or CO,

T O is or S, R⁶ is H, (1-4)alkyl, (1-4)alkoxy or halogen,

R⁷ is H or CH₃,

R⁸ is (1-4)alkyl,

R⁹ is H or (1-4)alkyl,

R¹⁰ is (1-4)alkyl, (1-4)haloalkyl, (3-4)alkenyl or (3-4)alkynyl,

R¹¹ and R¹² are each independently of the other H or (1-4)alkyl or an alkylene chain having 4 or 5 carbon atoms,

the radicals R¹³ together are an alkeanylene chain having 4 or 5 carbon atoms,

A is a radical of the formula ##STR6## one of the radicals X and Y being halogen, (1-3)alkyl, halo(1-3)alkyl, (1-3)alkoxy or halo(1-3)alkoxy and the other of the radicals X and Y being (1-3)alkyl, halo(1-3)alkyl, (1-3)alkoxy, halo(1-3)alkoxy, halogen, mono- or di- (1-3)alkyl!amino and

Z is CH or N.

Preferred compounds of the formula (I) and salts thereof according to the invention are those in which

R¹ is mono- or di- (1-4)alkyl!amino or (1-4)alkyl, preferably CH₃, C₂ H₅, n--C₃ H₇, i--C₃ H₇ or N(CH₃)₂,

n is 2,

R² and R³ are each hydrogen,

R⁴ is H or (1-4)alkyl,

R⁵ is CHO, (1-4)alkyl!carbonyl, (1-4)haloalkyl!carbonyl, (1-4)alkylsulfonyl, (1-4)haloalkylsulfonyl, (1-4)alkoxy!-carbonyl, mono- or di- (1-4)alkyl!aminocarbonyl, mono- or di- (1-4)alkyl!aminosulfonyl or

R⁴ and R⁵ together are a chain of the formula (--CH₂)_(m1) B¹ -- or --B¹ --(CH₂)_(m2) B² -- where B¹ and B² independently of each other are SO₂ or CO,

W and T are each O,

R⁶ is H and

R⁷ is H or CH₃.

The present invention also relates to a process for preparing the compounds of the formula (I) or salts thereof, which comprises

a) reacting a compound of the formula (II) ##STR7## with a heterocyclic carbamate of the formula (III),

    R*--O--CO--NR.sup.7 --A                                    (III)

where R* is unsubstituted or substituted phenyl or (1-4)alkyl, or

b) reacting an arylsulfonylcarbamate of the formula (IV) ##STR8## where Ar is an aryl radical, preferably unsubstituted or substituted phenyl, with an amino heterocycle of the formula (V)

    H--NR.sup.7 --A                                            (V)

or

c) reacting a sulfonyl isocyanate of the formula (VI) ##STR9## with an amino heterocycle of the formula H--NR⁷ --A (V), or d) reacting in a one-pot reaction first an amino heterocycle of the formula H-NR⁷ --A (V) in the presence of a base with phosgene and then the intermediate formed with a phenylsulfonamide of the formula (II), or

e) reacting a sulfonyl chloride of the formula (VII) ##STR10## with a cyanate M--OCN where M=a cation, for example NH₄, Na or K, and with an amino heterocycle of the formula H--NR⁷ --A (V) in the presence of a base, or

f) reacting a sulfonamide of the formula (II) mentioned with a (thio)isocyanate of the formula (V')

    W=C=N--A                                                   (V')

in the presence of a base where the radicals or symbols R¹ to R⁷, A, W and n in the formulae (II)-(VII) and (V') are as defined in formula (I) and where the compounds initially obtained in variants a) and c)-e) are compounds of the formula (I) where W=O.

The reaction of the compounds of the formulae (II) and (III) is preferably carried out under base catalysis in an inert organic solvent, for example dichloromethane, acetonitrile, dioxane or THF, at temperatures between 0° C. and the boiling point of the solvent. Suitable bases in this context are, for example, organic amine bases, such as 1,8-diazabicyclo 5.4.0!undec-7-ene (DBU), in particular if R*=(substituted) phenyl (cf. EP-A44807), or trimethylaluminum or triethylaluminum, the latter in particular if R*=alkyl (cf. EP-A-166516).

The sulfonamides (I) are novel compounds. They and their preparation are also part of the subject matter of this invention.

The preparation of the sulfonamides (II) can as a rule be carried out in the following manner:

Starting from unsubstituted or substituted 4-chloro-3-nitrotoluenes (VIII), the chlorine is, in the cases where R¹ is not NR⁸ R⁹, initially substituted by reaction with a mercaptan of the formula R¹ --SH. Reduction of the nitro group in (IX) to give the aniline derivative (X) and subsequent diazotization and coupling with SO₂ /CuCl (cf. H. Meerwein at al., Chem. Ber. 90, 841-1178 (1957)) and aminolysis with tert-butylamine affords sulfonamide (XI) (see Scheme 1). ##STR11##

To prepare the sulfonamides (II), the compounds of the formula (XI) are then, if appropriate after prior oxidation to (XII), converted into the sulfonamides (II) via side chain halogenation to (XIII), subsequent substitution of the halogen atom in (XIII) by amines, or by azide with successive reduction to the benzylamines (XIV), and further functionalization of the amino group and cleavage of the tert-butyl protecting group by known procedures (for example with CF₃ COOH) (see Scheme 2). ##STR12##

In compounds of the formula (II) wherein R¹ =NR⁸ R⁹ (see Scheme 3), for example, the chlorine in unsubstituted or substituted 4-chloro-3-nitrotoluenes (VIII) is initially exchanged with alkyl mercaptans or preferably with benzyl mercaptans to give (IX'). After oxidation and aminolysis of the sulfochloride intermediates with HNR⁸ R⁹, sulfonamides (XV) are obtained which, after reduction to (XVI), are converted into the corresponding sulfonamides (II) where R¹ =NR⁸ R⁹ as described in Schemes 1 and 2 for (X). ##STR13##

The carbamates of the formula (III) can be prepared by methods described in the South African Patent applications 8215671 and 8215045 or EP-A-70804 (U.S. Pat. No. 4,480,101) or RD 275056.

The reaction of the compounds (IV) with the amino heterocycles (V) is preferably carried out in inert aprotic solvents, such as dioxane, acetonitrile or tetrahydrofuran, at temperatures between 0° C. and the boiling temperature of the solvent. The starting materials (V) required are known from the literature or can be prepared by processes known from the literature. The arylsulfonylcarbamates of the formula (IV) can be obtained by the methods of U.S. Pat. No. 4,684,393 or U.S. Pat. No. 4,743,290.

The phenylsulfonyl isocyanates of the formula (VI) can be prepared by the method of U.S. Pat. No. 4,481,029 and reacted with the amino heterocycles (V).

The phosgenation of the compounds of the formula (V) according to variant d) car preferably be carried out in the presence of bases, such as sterically hindered organic amine bases, for example triethylamine. The subsequent reaction with compounds of the formula (II) according to variant d) can be carried out by known procedures (cf. EP-A-232 067).

The sulfochlorides (VII) can be obtained from the corresponding sulfonic acids, for example by standard methods such as the reaction of the potassium salt with phosphorus oxychloride or thionyl chloride in inert solvents such as acetonitrile and/or sulfolane or without a solvent by heating under reflux (cf. Houben-Weyl-Klamann, "Methoden der organischen Chemie", 4th edition Vol. 3 XI/2, pp. 1067-1073, Thieme Verlag Stuttgart, 1985).

The corresponding sulfonic acids can be obtained from the corresponding nitro compounds similarly to the reaction of compounds (IX).

Alternatively, in some cases the sulfochlorides (VII) can be prepared by sulfonation (+chlorination) or sulfochlorination of suitable substituted benzoic esters; sulfochlorination according to Houben-Weyl-Klamann, "Methoden der organischen Chemie", 4th edition Vol. E XI/2, p. 1067 ff., Thieme Verlag Stuttgart, 1985; Houben-Weyl-Muller, "Methoden der organischen Chemie", 4th edition Vol. IX, p. 563ff., Thieme Verlag Stuttgart, 1955; sulfonation according to Houbean-Weyl-Klamann, "Methoden der organischean Chemie, 4th edition Vol. E XI/2, p. 1055ff., Thieme Verlag Stuttgart, 1985; Houben-Weyl-Muller, "Methoden der organischen Chemie", 4th edition Vol. IX, p. 435 ff., Thieme Verlag Stuttgart, 1955.

The (thio)isocyanates of the formula (V') can be obtained by literature methods (EP-A-232067, EP-A-166516). The reaction of the (thio)isocyanates (V') with the compounds (II) is carried out at -10° C. to 100° C., preferably 20 to 100° C., in an inert aprotic solvent, such as acetone or acetonitrile, in the presence of a suitable base, for example N(C₂ H₅)₃ or K₂ CO₃.

The salts of the compounds of the formula (I) are preferably prepared in inert polar solvents such as water, methanol or acetone at temperatures of 0-100° C. Suitable bases for preparing the salts according to the invention are, for example, alkali metal carbonates, such as potassium carbonate, alkali metal hydroxides and alkaine earth metal hydroxides, for example NaOH or KOH, or ammonia or ethanolamine.

Solvents which have been termed "inert solvents" in the above process variants are to be understood as meaning in each case solvents which are inert under the prevailing reaction conditions, but which do not have to be inert under any selected reaction conditions.

The compounds of the formula (I) according to the invention have an outstanding herbicidal activity against a broad spectrum of economically important monocotyledonous and dicotyledonous harmful plants. The active substances also act efficiently on perennial broad-leaved weeds which produce shoots from rhizomes, rootstocks or other perennial organs and which are difficult to control. In this context, it does not matter whether the substances are applied before sowing, pre-emergence or post-emergence.

Specifically, examples may be mentioned of some representatives of the monocotyledonous and dicotyledonous weed flora which can be controlled by the compounds according to the invention, without the enumeration being a restriction to certain species.

Examples of weed species on which the active substance acts efficiently are, from amongst the monocotyledons, Avena, Lolium, Alopecurus, Phalaris, Echinochloa, Digitaria, Setaria and also Cyperus species from the annual sector and from amongst the perennial species Agropyron, Cynodon, Imperata and Sorghum, and also perennial Cyperus species.

In the case of the dicotyledonous weed species, the range of action extends to species such as, for example, Galium, Viola, Veronica, Lamium, Stellaria, Amaranthus, Sinapis, Ipomosa, Matricaria, Abutilon and Sida from amongst the annuals, and Convolvuius, Cirsium, Rumex and Artemisia in the case of the perennial weeds.

The active substances according to the invention also effect outstanding control of weeds which occur under the specific conditions of rice growing, such as, for example, Sagittaria, Alisma, Eleocharis, Scirpus and Cyperus.

If the compounds according to the invention are applied to the soil surface before germination, then the weed seedlings are either prevented completely from emerging, or the weeds grow until they have reached the cotyledon stage but then their growth stops, and, eventually, after three to four weeks have elapsed, they die completely.

Of the active substances are applied post-emergence to the green parts of the plants, growth likewise stops drastically a very short time after the treatment and the weed plants remain at the growth stage of the point of time of application, or they die completely after a certain time, so that in this manner competition by the weeds, which is harmful to the crop plants, is eliminated at a very early point in time and in a sustained manner.

Even though the compounds according to the invention have an excellent herbicidal activity against monocotyledonous and dicotyledonous weeds, crop plants of economically important crops, such as, for example, wheat, barley, rye, rice, maize, sugar beet, cotton and soya, are damaged not at all, or only to a negligible extent. For these reasons, the present compounds are highly suitable for selectively controlling undesired plant growth in areas under agricultural crops.

In addition, the substances according to the invention have outstanding growth-regulatory properties in crop plants. They engage in the plant metabolism in a regulating manner and can thus be employed for the targeted control of plant constituents and for facilitating harvesting, for example by triggering desiccation and stunted growth. Moreover, they are also suitable for the general control and inhibition of undesirable vegetative growth without destroying the plants in the process. The inhibition of vegetative growth is very important in a large number of monocotyledonous and dicotyledonous crops since it can reduce, or completely prevent, lodging.

The compounds according to the invention can be applied in the form of wettable powders, emulsifiable concentrates, sprayable solutions, dusts or granules in the customary preparations. The invention therefore also relates to herbicidal and plant-growth-regulating compositions which comprise the compounds of the formula (I).

The compounds of the formula (I) can be formulated in various ways, depending on the prevailing biological and/or chemico-physical parameters. The following possibilities are suitable formulations: wettable powders (WP), water-soluble powders (SP), water-soluble concentrates, emulsifiable concentrates (EC), emulsions (EW), such as oil-in-water and water-in-oil emulsions, sprayable solutions, suspension concentrates (SC), oil- or water-based dispersions, solutions which are miscible with oils, capsule suspensions (CS), dusts (DP), seed-dressing products, granules for broadcasting and soil application, granules (GR) in the form of microgranules, spray granules, coated granules and adsorption granules, water-dispersible granules (WG), water-soluble granules (SG), ULV formulations, microcapsules and waxes.

These individual types of formulation are known in principle and are described, for example, in: Winnacker-Kuchler, "Chemische Technologie" Chemical Technology!, Volume 7, C. Heuser Verlag Munich, 4th Ed. 19856, Wade van Valkenburg, "Pesticide Formulations", Marcel Dekker, N.Y., 1973; K. Martens, "Spray Drying" Handbook, 3rd Ed. 1979, G. Goodwin Ltd. London.

The formulation auxiliaries required, such as inert materials, surfactants, solvents and other additives are also known and are described, for example, in: Watkins, "Handbook of Insecticide Dust Diluents and Carriers", 2nd Ed., Darland Books, Caldwell N.J., H. v. Olphen, "Introduction to Clay Colloid Chemistry"; 2nd Ed., J. Wiley & Sons, N.Y.; C. Marsden, "Solvents Guide"; 2nd Ed., Interscience, N.Y. 1963; McCutcheon's "Detergents and Emulsifiers Annual", MC Publ. Corp., Ridgewood N.J.; Sisley and Wood, "Encyclopedia of Surface Active Agents", Chem. Publ. Co. Inc., N.Y. 1964; Schonfeldt, "Grenzflachenaktive Athylenoxidaddukte" Surface-active ethylene oxide adducts!, Wiss. Verlagsgesell., Stuttgart 1976; Winnacker-Kuchler, "Chemische Technologie" Chemical Technology!, Volume 7, C. Hauser Verlag Munich, 4th Ed. 1986.

Based on these formulations, it is also possible to prepare combinations with other pesticidally active substances, such as, for example, insecticides, acaricides, herbicides, fungicides, and also with safeners, fertilizers and/or growth regulators, for example in the form of a ready mix or a tank mix.

Wettable powders are preparations which are uniformly dispersible in water and which, besides the active substance, also comprise ionic and/or non-ionic surfactants (wetting agents, dispersants), for example polyoxethylated alkylphenols, polyoxethylated fatty alcohols, polyoxethylated fatty amines, fatty alcohol polyglycol ether sulfates, alkanesulfonates, alkylbenzeanesufonates, sodium lignosulfonate, sodium 2,2'-dinaphthylmethane6,6'-sulfonate, sodium dibutylnaphthalenesulfonate or else sodium oleoylmethyltaurinate, in addition to a diluent or inert substance. To prepare the wettable powders, the herbicidally active substances are ground finely, for example in customary equipment such as hammer mills, blower mills and air-jet mills, and simultaneously or subsequently mixed with the formulation auxiliaries.

Emulsifiable concentrates are prepared, for example, by dissolving the active substance in an organic solvent, for example butanol, cyclohexanone, dimethylformamide, xylene, or else higher-boiling aromatics or hydrocarbons or mixtures of the organic solvents with the addition of one or more ionic and/or non-ionic surfactants (emulsifiers). Examples of emulsifiers which can be used are: calcium salts of alkylarysulfonic acids such as calcium dodecylbenzenesulfonate, or non-ionic emulsifiers such as fatty acid polyglycol esters, alkylaryl polyglycol ethers, fatty alcohol polyglycol ethers, propylene oxide/ethylene oxide condensates, alkyl polyethers, sorbitan esters, for example sorbitan fatty acid esters or polyoxyethylene sorbitan esters, for example polyoxyethylene sorbitan fatty acid esters.

Dusts are obtained by grinding the active substance with finely divided solid substances, for example talc, natural clays such as kaolin, bentonite and pyrophyllite, or diatomaceous earth.

Suspension concentrates can be water- or oil-based. They can be prepared, for example, by wet grinding using commercially available bead mills with an optional addition of surfactants as they have already been mentioned above for example in the case of the other types of formulation.

Emulsions, for example oil-in-water emulsions (EW), can be prepared for example by means of stirrers, colloid mills and/or static mixers using aqueous organic solvents and, if appropriate, surfactants as they have already been mentioned above for example in the case of the other types of formulation.

Granules can be prepared either by spraying the active substance onto adsorptive granulated inert material or by applying active substance concentrates to the surface of carriers such as sand, kaolinites or of granulated inert material by means of binders, for example polyvinyl alcohol, sodium polyacrylate or else mineral oils. Suitable active substances can also be granulated in the manner which is conventional for the production of fertilizer granules, if desired as a mixture with fertilizers.

Water-dispersible granules are generally prepared by the customary processes such as spray drying, fluidized-bed granulation, disk granulation, mixing with high-speed mixers and extrusion without solid inert material.

For the preparation of disk, fluidized-bed, extruder and spray granules, see, for example, the processes in "Spray-Drying Handbook" 3rd ed. 1979, G. Goodwin Ltd., London; J. E. Browning, "Agglomeration", Chemical and Engineering 1967, pages 147 et seq.; "Perry's Chemical Engineer's Handbook", 5th Ed., McGraw-Hill, N.Y. 1973, pp. 8-57.

For further details on the formulation of crop protection products see, for example, G. C. Klingman, "Weed Control as a Science", John Wiley and Sons, Inc., N.Y., 1961, pages 81-96 and J. D. Freyer, S. A. Evans, "Weed Control Handbook", 5th Ed., Blackwell Scientific Publications, Oxford, 1968, pages 101-103.

As a rule, the agrochemical preparations comprise 0.1 to 99% by weight, in particular 0.1 to 95% by weight, of active substance of the formula (I). The active substance concentration in wettable powders is, for example, approximately 10 to 90% by weight, the remainder to 100% by weight being composed of customary formulation components. In the case of emulsifiable concentrates, the active substance concentration may amount to approximately 1 to 90, preferably 5 to 80%, by weight. Formulations in the form of dusts comprise 1 to 30% by weight of active substance, in most cases preferably 5 to 20% by weight of active substance, and sprayable solutions comprise approximately 0.05 to 80, preferably 2 to 50%, by weight of active substance. The active substance content of water-dispersible granules depends partly on whether the active compound is in liquid or solid form and on which granulation auxiliaries, fillers and the like are being used. The active substance content of the water-dispersible granules amounts to, for example, between 1 and 95% by weight, preferably between 10 and 80% by weight.

In addition, the abovementioned formulations of active substances comprise, if appropriate, the adhesives, wetting agents, dispersants, emulsifiers, penetrants, preservatives, antifreeze agents, solvents, fillers, carriers, colorants, antifoams, evaporation inhibitors and pH and viscosity regulators which are customary in each case.

Components which can be used in combination with the active substances according to the invention in mixed formulations or in the tank mix are, for example, known active substances as they are described, for example, in Weed Research 26, 441-445 (1986), or "The Pesticide Manual", 10th edition, The British Crop Protection Council and the Royal Soc. of Chemistry, 1994, and the literature cited therein. Examples of active substances which may be mentioned as herbicides which are known from the literature and which can be combined with the compounds of the formula (I) are the following (note: either the common names in accordance with the International Organization for Standardization (ISO) or the chemical names, if appropriate together with a customary code number, of the compounds are given): acetochlor; acifluorfen; aclonifen; AKH 7088, ie. 1- 5- 2-chloro-4-(trifluoromethyl)phenoxyl!-2-nitrophenyl !-2-methoxyethylidene!amino!oxy!acetic acid and its methyl ester; alachlor; alloxydim; ametryn; amidosulfuron; amitrol; AMS, ie. ammonium sulfamate; anilofos; asulam; atrazine; azimsulfurone (DPX-A8947); aziprotryn; barban; BAS 516 H, ie. 5-fluoro-2-phenyl-4H-3,1-benzoxazin-4-one; benazolin; benfluralin; benfuresate; bensulfuron-methyl; bensulide; bentazone; benzofenap; benzofluor; benzoyloprop-ethyl; benzthiazuron, bialaphos; bifenox; bromacil; bromobutide; bromofenoxim; bromoxynil; bromuron; burinafos; busoxinone; butachlor; butamifos; butenachlor; buthidazole; butralin; butylate; cafenstrole (CH-900); carbetamide; cafentrazone (ICI-A0051); CDAA, ie. 2-chloro-N,N-di-2-propenylacetamide; CDEC, ie. 2-chloroallyl diethyldithiocarbamate; chlormethoxyfen; chloramben; chlorazifop-butyl, chlormesulon (ICI-A0051); chlorbromuron; chlorbufam; chlorfenac; chlorflurecol-methyl; chloridazon; chlorimuron-ethyl; chlornitrofen; chlorotoluron; chloroxuron; chlorpropham; chlorsulfuron; chlorthal-dimethyl; chlorthiamid; cinmethylin; cinosulfuron; clethodim; clodinafop and its ester derivatives (for example clodinafop-propargyl); clomazone; clomeprop; cloproxydim; clopyralid; cumyluron, (JC 940); cyanazine; cycloate; cyclosulfamuron (AC 104); cycloxydim; cycluron; cyhalofop and its ester derivatives (for example butyl ester, DEH-112); cyperquat; cyprazine; cyprazole; daimuron; 2,4-DB; dalapon; desmedipham; desmetryn; di-allate; dicamba; dichlobenil; dichlorprop; diclofop and its esters, such as diclofop-methyl; diethatyl; difenoxuron; difenzoquat; diflufenican; dimefuron; dimethachlor; dimethametryn; dimethenamid (SAN-582H); dimethazone, clomazon; dimethipin; dimetrasulfuron, dinitramine; dinoseb; dinoterb; diphenamid; dipropetryn; diquat; dithiopyr; diuron; DNOC; eglinazine-ethyl; EL 77, ie. 5-cyano-1-(1,1-dimethylethyl)-N-methyl-1H-pyrazole-4-carboxamide; endothal; EPTC; esprocarb; ethalfluralin; ethametsulfuron-methyl; ethidimuron; ethiozin; ethofumesate; F5231, ie. N- 2-chloro-4-fluoro-5- 4-(3-fluoropropyl)-4,5-dihydro-5-oxo-1H-tetrazol-1-yl!phenyl !ethanesulfonamide; ethoxyfen and its esters (for example ethyl ester, HN-252); etobenzanid (HW 52); fenoprop; fenoxan, fenoxaprop and fenoxaprop-P and their esters, for example fenoxaprop-P-ethyl and fenoxaprop-ethyl; fenoxydim; fenuron; flamprop-methyl; flazasulfuron; fluazifop and fluazifop-P and their esters, for example fluazifop-butyl and fluazifop-P-butyl; fluchloralin; flumetsulam; flumeturon; flumiclorac and its esters (for example pentyl ester, S-23031); flumioxazin (S-482); flumipropyn; flupoxam (KNW-739); fluorodifen; fluoroglycofen-ethyl; flupropacil (UBIC-4243); fluridone; flurochloridone; fluroxypyr; flurtamone; fomesafen; fosamine; furyloxyfen; glufosinate; glyphosate; halosafen; halosulfuron and its esters (for example methyl ester, NC-319); haloxyfop and its esters; haloxyfop-P (=R-haloxyfop) and its esters; hexazinone; imazamethabenz-methyl; imazapyr; imazaquin and salts, such as the ammonium salt; imazethamethapyr; imazethapyr; imazosulfuron; ioxynil; isocarbamid; isopropalin; isoproturon; isouron; isoxaben; isoxapyrifop, karbutilate; lactofen; lenacil; linuron; MCPA; MCPB; mecoprop; mefenacet; mefluidid; metamitron; metazachlor; methabenzthiazuron; metham; methazole; methoxyphenone; methyldymron; metabenzuron, methobenzuron; metobromuron; metolachlor; metosulam (XRD 511); metoxuron; metribuzin; metsulfuron-methyl; MH; molinate; monalide; monocarbamide dihydrogensulfate; monolinuron; monuron; MT 128, ie. 6-chloro-N-(3-chloro-2-propenyl)-5-methyl-N-phenyl-3-pyridazinamine; MT 5950, ie. N- 3-chloro-4-(1-methylethyl)phenyl!-2-methylpentanamide; naproanilide; napropamide; naptalam; NC 310 ie. 4-(2,4-dichlorobenzoyl)-1-methyl-5-benzyloxypyrazole; neburon; nicosulfuron; nipyraclophen; nitralin; nitrofen; nitrofluorfen; norflurazon; orbencarb; oryzalin; oxadiargyl (RP-020630); oxadiazon; oxyfluorfen; paraquat; pebulate; pendimethalin; perfluidone; phenisopham; phenmedipham; picloram; piperophos; piributicarb; pirifenop-butyl; pretilachlor; primsulfuron-methyl; procyazine; prodiamine; profluralin; proglinazine-ethyl; prometon; prometryn; propachlor; propanil; propaquizafop and its esters; propazine; propham; propisochlor; propyzamide; prosulfalin; prosulfocarb; prosulfuron (CGA-152005); prynachlor; pyrazolinate; pyrazon; pyrazosulfuron-ethyl; pyrazoxyfen; pyridate; pyrithiobac (KIH-2031); pyroxofop and its esters (for example propargyl ester); quinclorac; quinmerac; quinofop and its ester derivatives, quizalofop and quizalofop-P and their ester derivates, for example quizalofop-ethyl; quizalofop-P-tefuryl and -ethyl; renriduron; rimsulfuron (DPX-E 9636); S 275, ie. 2- 4-chloro-2-fluoro-5-(2-propynyloxy)phenyl!-4,5,6,7-tetrahydro-2H-indazole; secbumeton; sethoxydim; siduron; simazine; simetryn; SN 106279, ie. 2- 7- 2-chloro-4-(trifluoromethyl)phenoxyl!-2-naphthalenyl!oxy!propanoic acid and its methyl ester; sulfentrazone (FMC-97285, F-6285); sulfazuron; sulfometuron-methyl; sulfosate (ICI-A0224); TCA; tebutam (GCP-5544); tebuthiuron; terbacil; terbucarb; terbuchlor; terbumeton; terbuthylazine; terbutryn; TFH 450, ie. N,N-diethyl-3- (2-ethyl-6-methylphenyl)sulfonyl!-1H-1,2,4-triazole-1-carboxamide; thenylchlor (NSK-850); thiazafluron, thiazopyr (Mon-13200); thidiazimine (SN-24085); thifensulfuron-methyl; thiobencarb; tiocarbazil; tralkoxydim; tri-allate; triasulfuron; triazofenamide; tribenuron-methyl; triclopyr; tridiphane; trietazine; trifluralin; triflusulfuron and esters (for example methyl ester, DPX-66037); trimeturon; tsitodef; vernolate; WL 110547, ie. 5-phenoxy-1- 3-(trifluoromethyl)phenyl!-1H-tetrazole; UBH-509; D-489; LS 82-556; KPP-300; NC-324; NC-330; KH-218; DPX-N8189; SC-0774; DOWCO-535; DK-8910; V-53482; PP-600; MBH-001; KIH-9201; ET-751; KIH-6127 and KIH-2023.

For use, the formulations, which are in commercially available form, are, if appropriate, diluted in the customary manner, for example using water in the case of wettable powders, emulsifiable concentrates, dispersions and water-dispersible granules. Preparations in the form of dusts, granules for soil application or for broadcasting and sprayable solutions are conventionally not diluted any further with inert substances prior to use.

The application rate required, of the compounds of the formula (I), varies with the external factors such as, inter alia, temperature, humidity and nature of the herbicide used. It can vary within wide limits, for example between 0.001 and 10.0 kg/ha or more of active substance, but it is preferably between 0.005 and 5 kg/ha.

A. CHEMICAL EXAMPLES

Abbreviations:

If not further specified, the % details and molar ratios are based on weight.

in vacuo=under reduced pressure

h=hour(s)

DMF=dimethylformamide

EtOH=C₂ H₅ OH

Example A1

4-Methylthio-3-nitrotoluene

138 g (1 mol) of K₂ CO₃ are added to a solution of 171.6 g (1 mol) of 4-chloro-3-nitrotoluene in 500 ml of DMF. 1 molar equivalent of methyl mercaptan is passed through, and stirring is continued at 50° C. for 3 h. The reaction mixture is poured on a large amount of ice-water and the precipitate is filtered off under suction, washed with water and dried; 146.3 g (80%) of 4-methylthio-3-nitrotoluene of melting point 71-73° C. are obtained.

Example A2

3-Amino-4-methylthiotoluene

A solution of 146 g (0.8 mol) of 4-methylthio-3-nitrotoluene in a mixture of 1000 ml of EtOH and 700 ml of glacial acetic acid is heated to 65-80° C. and, over a period of about 8 h, admixed with a total of 122.9 g (2.2 mol) of powdered iron, a little at a time. After the reaction has ended, the mixture is filtered off under suction through Na₂ SO₄, washed thoroughly with EtOH and concentrated in vacuo. 122 g (99%) of 3-amino4-methylthiotoluens are obtained as a dark brown oil.

¹ H--NMR (300 MHz, CDCl₃):

δ=2.24 (s, 3H, SCH₃)

2.30 (s, 3H, Ar--CH₃)

4.25 (bs, 2H, NH₂)

6.52 (m, 2H, Ar--H)

7.25 (d, 1H, Ar--H)

Example A3

N-tert-Butyl-2-methylthio-5-methylbenzenesulfonamide

At 0-10° C., 24.3 g (0.352 mol) of NaNO₂ dissolved in 50 ml of H₂ O are added dropwise to a suspension of 49 g (0.32 mol) of 3-amino-4-methylthiotoluene in 180 ml of conc. HCl, and stirring is continued for half an hour. The diazonium salt suspension obtained is added a little at a time to a mixture of SO₂ -saturated glacial acetic acid (450 ml), 9.5 g (0.096 mol) of CuCl and CH₂ Cl₂ (450 ml) which has been warmed to 30° C. After the addition, stirring is continued at 30° C. for 1-2 h and the mixture is poured into ice-water. The phases are separated and the aqueous phase is extracted two more times with CH₂ Cl₂. The combined organic extracts are washed, dried over Na₂ SO₄ and completely evaporated in vacuo.

The crude product obtained (66.5 g, 0.28 mol) is dissolved in 650 ml of CH₂ Cl₂ and treated with 73 ml (0.7 mol, 2.5 equivalents) of tert-butylamine at 0° C.

For work-up, the mixture is poured into ice-water after about 1 h, the phases are separated and the aqueous phase is extracted two more times with CH₂ Cl₂. The combined organic extracts are washed, dried over Na₂ SO₄ and concentrated in vacuo. The solid obtained on digesting the residue with a mixture of diisopropyl etherlethyl acetate is filtered off and dried. 41.5 g (47.4%) of N-tert-butyl-2-methylthio-5-methylbenzenesulfonamide of melting point 119-121° C. are obtained.

Example A4

N-tert-Butyl-2-methanesulfonyl-5-methylbenzenesulfonamide

A solution of 41.5 g (0.152 mol) of N-tert-butyl-2-methylthio-5-methylbenzenesulfonamide in 470 ml of MeOH and 190 ml of H₂ O is heated to 50° C. and, over a period of 7 h, admixed with 140.2 g (0.228 mol) of sodium peroxomonosulfate (®Oxone), a little at a time. After the reaction has ended, the mixture is poured into a large volume of ice-water and the precipitated product is filtered off. After drying, 46.0 g (99%) of N-tert-butyl-2-methanesulfonyl-5-methylbenzenesulfonamide of melting point 129-133° C. are obtained.

Example A5

N-tert-Butyl-5-bromomethyl-2-methanesulfonylbenzenesulfonamide

A solution of 46 g (0.152 mol) of N-tert-butyl-2-methanesulfonyl-5-methyl-benzenesulfonamide in 450 ml of CCl₄ is, after the addition of 27.0 g (0.152 mol) of NBS (N-bromosuccinimide) and 1 g of AIBN (azobisisobutyronitrile), heated under reflux for 7 h using a daylight lamp. The reaction mixture is then filtered and washed successively with NaHSO₃ solution, NaHCO₃ solution and water, dried over MgSO₄ and completely concentrated in vacuo. 51.2 g of a crude mixture containing 55% by weight of N-tert-butyl-5-bromomethyl-2-methanesulfonylbenzenesulfonamide are obtained.

¹ H-NMR (300 MHz, CDCl₃):

δ=1.25 (s, 9H, tert-butyl)

3.40 (s, 3H, SO₂ CH₃)

4.52 (s, 2H, ArCH₂)

6.26 (s, 1H, NH)

7.75 (dd, 1H, Ar--H, J=2 Hz, 8 Hz)

8.25 (d, 1H, Ar--H, J=8 Hz)

8.31 (d, 1H, Ar--H, J=2 Hz)

Example A6

At 0° C., 51 g of N-tert-butyl-5-bromomethyl-2-methanesulfonylbenzenesulfonamide (55% by weight ^(A) 28.05 g=0.669 mol) dissolved in 250 ml of THF are added to a solution of 59.5 ml (0.69 mol) of a 40% strength aqueous methylamine solution in 150 ml of THF. Stirring is continued at 0-5° C. for 2-3 h. For work-up, the solution is completely concentrated, the residue is taken up in plenty of 2N HCl and extracted with diethyl ether (2×200 ml). The acidic aqueous phase is adjusted to pH 9 with 4N NaOH and extracted with ethyl acetate (3×200 ml). The combined ethyl acetate extracts are washed with water, dried over Na₂ SO₄ and evaporated in vacuo. 17 g (73.7%) of N-tert-butyl-5-methylaminomethyl-2-methanesulfonylbenzenesulfonamide of melting point 76-78° C. are obtained as residue.

Example A7

N-tert-Butyl-5-(N-methyl-N-methanesulfonylaminomethyl)-2-methanesulfonylbenzenesulfonamide

0.39 ml (5 mmol) of methenesulfonyl chloride dissolved in 5 ml of dichloromethane are added dropwise to a solution of 1.67 g (5 mmol) of N-tert-butyl-5-methylaminomethyl-2-methanesulfonylbenzenesulfonamide and 0.73 ml (5.3 mmol) of triethylamine in 20 ml of dichloromethane which had been cooled to 0° C. After 30 min at room temperature, the reaction solution is washed with water, dried and completely evaporated in vacuo. 1.85 g (89.7%) of N-tert-butyl-5-(N-methyl-N-methanesulfonylaminomethyl)-2-methanesulfonylbenzenesulfonamide are obtained as a viscous oil.

¹ H--NMR (300 MHz, CDCl₃):

δ=1.23 (s, 9H, tert-butyl)

2.82 (s, 3H, N--CH₃)

2.94 (s, 3H, N--SO₂ CH₃)

3.40 (s, 3H, Ar--SC₂ CH₃)

4.46 (s, 2H, Ar--CH₂)

6.30 (s, 1H, NH)

7.83 (dd, 1H, Ar--H, J=2 Hz, 8 Hz)

8.20 (d, 1H, Ar--H, J=2 Hz)

8.30 (d, 1H, Ar--H, J=8 Hz)

Example A8

5-(N-Methyl-N-methanesulfonylaminomethyl)-2-methanesulfonylbenzenesulfonamide

A solution of 1.85 g (4.5 mmol) of N-tert-butyl-5-(N-methyl-N-methanesulfonylaminomethyl)-2-methanesulfonylbenzenesulfonamide in 20 ml of trifluoroacetic acid is stirred at room temperature for 8 h. The mixture is evaporated to dryness and then coevaporated with toluene, and the residue obtained is crystallized from ethyl acetate/diisopropyl ether. 1.32 g (83%) of 5-(N-methyl-N-methanesulfonylaminomethyl)-2-methanesulfonylbenzenesulfonamide of melting point 165-169° C. are obtained.

Example A9

N-(4,6-Dimethoxypyrimidin-2-ylaminocarbonyl)-5-(N-methyl-N-methanesulfonylaminomethyl)-2-methanesulfonylbenzenesulfonamide

0.56 ml (3.7 mmol) of DBU is added dropwise to a suspension of 1.33 g (3.7 mmol) of 5-(N-methyl-N-methanesulfonylaminomethyl)-2-methanesulfonylbenzenesulfonamide and 1.03 g (3.7 mmol) of phenyl N-(4,6-dimethoxypyrimidin-2-yl)carbamate in 20 ml of acetonitrile. After 2 h, the mixture is diluted with water and diethyl ether and acidified to pH 1-2 with HCl and the precipitated product is filtered off, washed with water and diethyl ether and dried; yield: 1.78 g (89.5%) of N-(4,6-dimethoxypyrimidin-2-ylaminocarbonyl)-5-(N-methyl-N-methanesulfonylamiinomethyl)-2-methanesulfonylbenzenesulfonamide of melting point 205-210° C. (decomposition).

The compounds according to the invention listed in the tables below are obtained by or analogously to Examples A1 to A8 or by the processes mentioned in the general part.

Abbreviations in the Tables:

No.=Example number, Example compound number

mp.=melting point

n-, i-, s-, t-C₄ H₉ =n-, iso-, secondary-, tertiary-butyl

n-C₃ H₇ =n-propyl

i-C₃ H₇ =isopropyl

                                      TABLE 1     __________________________________________________________________________     Compound of the formula (1a)     1 #STR14##     No.        R.sup.1             R.sup.4                R.sup.5  R.sup.7                             X    Y     Z  mp.(°C.)     __________________________________________________________________________     1  CH.sub.3             H  CHO      H   OCH.sub.3                                  OCH.sub.3                                        CH 142-148     2  CH.sub.3             H  CHO      H   OCH.sub.3                                  CH.sub.3                                        CH     3  CH.sub.3             H  CHO      H   CH.sub.3                                  CH.sub.3                                        CH     4  CH.sub.3             H  CHO      H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     5  CH.sub.3             H  CHO      H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     6  CH.sub.3             H  CHO      H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     7  CH.sub.3             H  CHO      H   OCHF.sub.2                                  OCHF.sub.2                                        CH     8  CH.sub.3             H  CHO      H   CH.sub.3                                  OCHF.sub.2                                        CH     9  CH.sub.3             H  CHO      H   Cl   OCH.sub.3                                        CH     10 CH.sub.3             H  CHO      H   OCH.sub.3                                  OCH.sub.3                                        N     11 CH.sub.3             H  CHO      H   OCH.sub.3                                  CH.sub.3                                        N     12 CH.sub.3             H  CHO      H   CH.sub.3                                  CH.sub.3                                        N     13 CH.sub.3             H  CHO      H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     14 CH.sub.3             H  CHO      H   OCH.sub.3                                  CF.sub.3                                        N     15 CH.sub.3             H  CHO      H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     16 CH.sub.3             H  CHO      CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     17 CH.sub.3             H  CHO      CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     18 CH.sub.3             H  COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 195-200     19 CH.sub.3             H  COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     20 CH.sub.3             H  COCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     21 CH.sub.3             H  COCH.sub.3                         H   CH.sub.3                                  OC.sub.2 C.sub.5                                        CH     22 CH.sub.3             H  COCH.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     23 CH.sub.3             H  COCH.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     24 CH.sub.3             H  COCH.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     25 CH.sub.3             H  COCH.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     26 CH.sub.3             H  COCH.sub.3                         H   Cl   OCH.sub.3                                        CH     27 CH.sub.3             H  COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     28 CH.sub.3             H  COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     29 CH.sub.3             H  COCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     30 CH.sub.3             H  COCH.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     31 CH.sub.3             H  COCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     32 CH.sub.3             H  COCH.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     33 CH.sub.3             H  COCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     34 CH.sub.3             H  COCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     35 CH.sub.3             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH 196-200     36 CH.sub.3             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     37 CH.sub.3             H  COC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     38 CH.sub.3             H  COC.sub.2 H.sub.5                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     39 CH.sub.3             H  COC.sub.2 H.sub.5                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     40 CH.sub.3             H  COC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     41 CH.sub.3             H  COC.sub.2 H.sub.5                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     42 CH.sub.3             H  COC.sub.2 H.sub.5                         H   CH.sub.3                                  OCHF.sub.2                                        CH     43 CH.sub.3             H  COC.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     44 CH.sub.3             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     45 CH.sub.3             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     46 CH.sub.3             H  COC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        N     47 CH.sub.3             H  COC.sub.2 H.sub.5                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     48 CH.sub.3             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     49 CH.sub.3             H  COC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     50 CH.sub.3             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     51 CH.sub.3             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     52 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH     53 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     54 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     55 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     56 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     57 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     58 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     59 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     60 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     61 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     62 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     63 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     64 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     65 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     66 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     67 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     68 CH.sub.3             H  CO-n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     69 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH 80-89     70 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     71 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     72 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     73 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     74 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     75 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     76 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     77 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     78 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     79 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     80 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     81 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     82 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     83 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     84 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     85 CH.sub.3             H  CO-i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     86 CH.sub.3             H  COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 138-141     87 CH.sub.3             H  COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     88 CH.sub.3             H  COCF.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     89 CH.sub.3             H  COCF.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     90 CH.sub.3             H  COCF.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     91 CH.sub.3             H  COCF.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     92 CH.sub.3             H  COCF.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     93 CH.sub.3             H  COCF.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     94 CH.sub.3             H  COCF.sub.3                         H   Cl   OCH.sub.3                                        CH     95 CH.sub.3             H  COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     96 CH.sub.3             H  COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     97 CH.sub.3             H  COCF.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     98 CH.sub.3             H  COCF.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     99 CH.sub.3             H  COCF.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     100        CH.sub.3             H  COCF.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     101        CH.sub.3             H  COCF.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     102        CH.sub.3             H  COCF.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     103        CH.sub.3             H  COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 150-154     104        CH.sub.3             H  COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     105        CH.sub.3             H  COOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     106        CH.sub.3             H  COOCH.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     107        CH.sub.3             H  COOCH.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     108        CH.sub.3             H  COOCH.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     109        CH.sub.3             H  COOCH.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     110        CH.sub.3             H  COOCH.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     111        CH.sub.3             H  COOCH.sub.3                         H   Cl   OCH.sub.3                                        CH     112        CH.sub.3             H  COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     113        CH.sub.3             H  COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     114        CH.sub.3             H  COOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     115        CH.sub.3             H  COOCH.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     116        CH.sub.3             H  COOCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     117        CH.sub.3             H  COOCH.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     118        CH.sub.3             H  COOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     119        CH.sub.3             H  COOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     120        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH 151-156     121        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     122        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     123        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     124        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     125        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     126        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     127        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   CH.sub.3                                  OCHF.sub.2                                        CH     128        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     129        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     130        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     131        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        N     132        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     133        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     134        CH.sub.3             H  COOC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     135        CH.sub.3             H  COOC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     136        CH.sub.3             H  COOC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        CH     137        CH.sub.3             H  COOC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     138        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 208-210     139        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     140        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     141        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     142        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     143        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     144        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     145        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     146        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   Cl   OCH.sub.3                                        CH     147        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     148        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     149        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     150        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     151        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     152        CH.sub.3             H  SO.sub.2 CH.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     153        CH.sub.3             H  SO.sub.2 CH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     154        CH.sub.3             H  SO.sub.2 CH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     155        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH 157-160     156        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     157        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     158        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     159        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     160        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     161        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     162        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   CH.sub.3                                  OCHF.sub.2                                        CH     163        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     164        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     165        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     166        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        N     167        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     168        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     169        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     170        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     171        CH.sub.3             H  C.sub.2 H.sub.5 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     172        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     173        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   OC.sub.2 H.sub.5                                  OCH.sub.3                                        CH     174        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     175        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     176        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     177        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     178        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     179        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     180        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   CH.sub.3                                  OCHF.sub.2                                        CH     181        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     182        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     183        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     184        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        N     185        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     186        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     187        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     188        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     189        CH.sub.3             H  n-C.sub.3 H.sub.7 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     190        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     191        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     192        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     193        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     194        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     195        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     196        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     197        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   CH.sub.3                                  OCHF.sub.2                                        CH     198        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     199        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     200        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     201        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        N     202        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     203        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     204        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     205        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     206        CH.sub.3             H  i-C.sub.3 H.sub.7 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     207        CH.sub.3             H  ClCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     208        CH.sub.3             H  ClCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        CH     209        CH.sub.3             H  ClCH.sub.2 CO                         H   CH.sub.3                                  CH.sub.3                                        CH     210        CH.sub.3             H  ClCH.sub.2 CO                         H   Cl   OCH.sub.3                                        CH     211        CH.sub.3             H  ClCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        N     212        CH.sub.3             H  ClCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        N     213        CH.sub.3             H  ClCH.sub.2 CO                         H   OCH.sub.3                                  CF.sub.3                                        N     214        CH.sub.3             H  ClCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     215        CH.sub.3             H  ClCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     216        CH.sub.3             H  Cl.sub.2 CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     217        CH.sub.3             H  Cl.sub.2 CHCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     218        CH.sub.3             H  Cl.sub.2 CHCO                         H   CH.sub.3                                  CH.sub.3                                        CH     219        CH.sub.3             H  Cl.sub.2 CHCO                         H   Cl   OCH.sub.3                                        CH     220        CH.sub.3             H  Cl.sub.2 CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     221        CH.sub.3             H  Cl.sub.2 CHCO                         H   OCH.sub.3                                  CH.sub.3                                        N     222        CH.sub.3             H  Cl.sub.2 CHCO                         H   OCH.sub.3                                  CF.sub.3                                        N     223        CH.sub.3             H  Cl.sub.2 CHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     224        CH.sub.3             H  Cl.sub.2 CHCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     225        CH.sub.3             H  Cl.sub.3 CCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH 125-130     226        CH.sub.3             H  Cl.sub.3 CCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     227        CH.sub.3             H  Cl.sub.3 CCO                         H   CH.sub.3                                  CH.sub.3                                        CH     228        CH.sub.3             H  Cl.sub.3 CCO                         H   Cl   OCH.sub.3                                        CH     229        CH.sub.3             H  Cl.sub.3 CCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     230        CH.sub.3             H  Cl.sub.3 CCO                         H   OCH.sub.3                                  CH.sub.3                                        N     231        CH.sub.3             H  Cl.sub.3 CCO                         H   OCH.sub.3                                  CF.sub.3                                        N     232        CH.sub.3             H  Cl.sub.3 CCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     233        CH.sub.3             H  Cl.sub.3 CCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     234        CH.sub.3             H  CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     235        CH.sub.3             H  CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        CH     236        CH.sub.3             H  CH.sub.3 OCH.sub.2 CO                         H   CH.sub.3                                  CH.sub.3                                        CH     237        CH.sub.3             H  CH.sub.3 OCH.sub.2 CO                         H   Cl   OCH.sub.3                                        CH     238        CH.sub.3             H  CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        N     239        CH.sub.3             H  CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        N     240        CH.sub.3             H  CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  CF.sub.3                                        N     241        CH.sub.3             H  CH.sub.3 OCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     242        CH.sub.3             H  CH.sub.3 OCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     243        CH.sub.3             H  CH.sub.2 ═CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     244        CH.sub.3             H  CH.sub.2 ═CHCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     245        CH.sub.3             H  CH.sub.2 ═CHCO                         H   CH.sub.3                                  CH.sub.3                                        CH     246        CH.sub.3             H  CH.sub.2 ═CHCO                         H   Cl   OCH.sub.3                                        CH     247        CH.sub.3             H  CH.sub.2 ═CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     248        CH.sub.3             H  CH.sub.2 ═CHCO                         H   OCH.sub.3                                  CH.sub.3                                        N     249        CH.sub.3             H  CH.sub.2 ═CHCO                         H   OCH.sub.3                                  CF.sub.3                                        N     250        CH.sub.3             H  CH.sub.2 ═CHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     251        CH.sub.3             H  CH.sub.2 ═CHCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     252        CH.sub.3             H  CH.tbd.CCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     253        CH.sub.3             H  CH.tbd.CCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     254        CH.sub.3             H  CH.tbd.CCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     255        CH.sub.3             H  CH.tbd.CCO                         H   Cl   OCH.sub.3                                        CH     256        CH.sub.3             H  CH.tbd.CCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     257        CH.sub.3             H  CH.tbd.CCO                         H   OCH.sub.3                                  CH.sub.3                                        N     258        CH.sub.3             H  CH.tbd.CCO                         H   OCH.sub.3                                  CF.sub.3                                        N     259        CH.sub.3             H  CH.tbd.CCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     260        CH.sub.3             H  CH.tbd.CCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     261        CH.sub.3             H                2 #STR15##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     262        CH.sub.3             H                2 #STR16##                         H   OCH.sub.3                                  CH.sub.3                                        CH     263        CH.sub.3             H                2 #STR17##                         H   CH.sub.3                                  CH.sub.3                                        CH     264        CH.sub.3             H                2 #STR18##                         H   Cl   OCH.sub.3                                        CH     265        CH.sub.3             H                2 #STR19##                         H   OCH.sub.3                                  OCH.sub.3                                        N     266        CH.sub.3             H                2 #STR20##                         H   OCH.sub.3                                  CH.sub.3                                        N     267        CH.sub.3             H                2 #STR21##                         H   OCH.sub.3                                  CF.sub.3                                        N     268        CH.sub.3             H                2 #STR22##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     269        CH.sub.3             H                2 #STR23##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     270        CH.sub.3             H                3 #STR24##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     271        CH.sub.3             H                3 #STR25##                         H   OCH.sub.3                                  CH.sub.3                                        CH     272        CH.sub.3             H                3 #STR26##                         H   CH.sub.3                                  CH.sub.3                                        CH     273        CH.sub.3             H                3 #STR27##                         H   Cl   OCH.sub.3                                        CH     274        CH.sub.3             H                3 #STR28##                         H   OCH.sub.3                                  OCH.sub.3                                        N     275        CH.sub.3             H                3 #STR29##                         H   OCH.sub.3                                  CH.sub.3                                        N     276        CH.sub.3             H                3 #STR30##                         H   OCH.sub.3                                  CF.sub.3                                        N     277        CH.sub.3             H                3 #STR31##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     278        CH.sub.3             H                3 #STR32##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     279        CH.sub.3             H                4 #STR33##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     280        CH.sub.3             H                4 #STR34##                         H   OCH.sub.3                                  CH.sub.3                                        CH     281        CH.sub.3             H                4 #STR35##                         H   CH.sub.3                                  CH.sub.3                                        CH     282        CH.sub.3             H                4 #STR36##                         H   Cl   OCH.sub.3                                        CH     283        CH.sub.3             H                4 #STR37##                         H   OCH.sub.3                                  OCH.sub.3                                        N     283        CH.sub.3             H                4 #STR38##                         H   OCH.sub.3                                  OCH.sub.3                                        N     284        CH.sub.3             H                4 #STR39##                         H   OCH.sub.3                                  CH.sub.3                                        N     285        CH.sub.3             H                4 #STR40##                         H   OCH.sub.3                                  CF.sub.3                                        N     286        CH.sub.3             H                4 #STR41##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     287        CH.sub.3             H                4 #STR42##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     288        CH.sub.3             H                5 #STR43##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     289        CH.sub.3             H                5 #STR44##                         H   OCH.sub.3                                  CH.sub.3                                        CH     290        CH.sub.3             H                5 #STR45##                         H   CH.sub.3                                  CH.sub.3                                        CH     291        CH.sub.3             H                5 #STR46##                         H   Cl   OCH.sub.3                                        CH     292        CH.sub.3             H                5 #STR47##                         H   OCH.sub.3                                  OCH.sub.3                                        N     293        CH.sub.3             H                5 #STR48##                         H   OCH.sub.3                                  CH.sub.3                                        N     294        CH.sub.3             H                5 #STR49##                         H   OCH.sub.3                                  CF.sub.3                                        N     295        CH.sub.3             H                5 #STR50##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     296        CH.sub.3             H                5 #STR51##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     297        CH.sub.3             H  CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     298        CH.sub.3             H  CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     299        CH.sub.3             H  CF.sub.3 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     300        CH.sub.3             H  CF.sub.3 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     301        CH.sub.3             H  CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     302        CH.sub.3             H  CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     303        CH.sub.3             H  CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     304        CH.sub.3             H  CF.sub.3 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     305        CH.sub.3             H  CF.sub.3 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     306        CH.sub.3             H  FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     307        CH.sub.3             H  FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     308        CH.sub.3             H  FCH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     309        CH.sub.3             H  FCH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     310        CH.sub.3             H  FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     311        CH.sub.3             H  FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     312        CH.sub.3             H  FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     313        CH.sub.3             H  FCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     314        CH.sub.3             H  FCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     315        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     316        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     317        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     318        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     319        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     320        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     321        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     322        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     323        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     324        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     325        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     326        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     327        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     328        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     329        CH.sub.3             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     330        CH.sub.3             H  Cl.sub.2 CHSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     331        CH.sub.3             H  Cl.sub.2 CHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     332        CH.sub.3             H  Cl.sub.2 CHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     333        CH.sub.3             H  Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     334        CH.sub.3             H  Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     335        CH.sub.3             H  Cl.sub.3 CSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     336        CH.sub.3             H  Cl.sub.3 CSO.sub.2                         H   Cl   OCH.sub.3                                        CH     337        CH.sub.3             H  Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     338        CH.sub.3             H  Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     339        CH.sub.3             H  Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     340        CH.sub.3             H  Cl.sub.3 CSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     341        CH.sub.3             H  Cl.sub.3 CSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     342        CH.sub.3             H  nC.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     343        CH.sub.3             H  nC.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     344        CH.sub.3             H  nC.sub.4 H.sub.9 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     345        CH.sub.3             H  nC.sub.4 H.sub.9 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     346        CH.sub.3             H  nC.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     347        CH.sub.3             H  nC.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     348        CH.sub.3             H  nC.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     349        CH.sub.3             H  nC.sub.4 H.sub.9 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     350        CH.sub.3             H  nC.sub.4 H.sub.9 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     351        CH.sub.3             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     352        CH.sub.3             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     353        CH.sub.3             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     354        CH.sub.3             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     355        CH.sub.3             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     356        CH.sub.3             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     357        CH.sub.3             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     358        CH.sub.3             H  CF.sub.3 CH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     359        CH.sub.3             H  CF.sub.3 CH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     360        CH.sub.3             H  CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     361        CH.sub.3             H  CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     362        CH.sub.3             H  CH.sub.3 NHSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     363        CH.sub.3             H  CH.sub.3 NHSO.sub.2                         H   Cl   OCH.sub.3                                        CH     364        CH.sub.3             H  CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     365        CH.sub.3             H  CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     366        CH.sub.3             H  CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     367        CH.sub.3             H  CH.sub.3 NHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     368        CH.sub.3             H  CH.sub.3 NHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     369        CH.sub.3             H  Me.sub.2 NSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     370        CH.sub.3             H  Me.sub.2 NSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     371        CH.sub.3             H  Me.sub.2 NSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     372        CH.sub.3             H  Me.sub.2 NSO.sub.2                         H   Cl   OCH.sub.3                                        CH     373        CH.sub.3             H  Me.sub.2 NSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     374        CH.sub.3             H  Me.sub.2 NSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     375        CH.sub.3             H  Me.sub.2 NSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     376        CH.sub.3             H  Me.sub.2 NSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     377        CH.sub.3             H  Me.sub.2 NSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     378        CH.sub.3             H  Me.sub.3 C-- OCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     379        CH.sub.3             H  Me.sub.3 C-- OCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     380        CH.sub.3             H  Me.sub.3 C-- OCO                         H   CH.sub.3                                  CH.sub.3                                        CH     381        CH.sub.3             H  Me.sub.3 C-- OCO                         H   Cl   OCH.sub.3                                        CH     382        CH.sub.3             H  Me.sub.3 C-- OCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     383        CH.sub.3             H  Me.sub.3 C-- OCO                         H   OCH.sub.3                                  CH.sub.3                                        N     384        CH.sub.3             H  Me.sub.3 C-- OCO                         H   OCH.sub.3                                  CF.sub.3                                        N     385        CH.sub.3             H  Me.sub.3 C-- OCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     386        CH.sub.3             H  Me.sub.3 C-- OCO                         H   OCH.sub.3                                  CH.sub.3                                        N     387        CH.sub.3             H  PhCO     H   OCH.sub.3                                  OCH.sub.3                                        CH     388        CH.sub.3             H  PhCO     H   OCH.sub.3                                  CH.sub.3                                        CH     389        CH.sub.3             H  PhCO     H   CH.sub.3                                  CH.sub.3                                        CH     390        CH.sub.3             H  PhCO     H   Cl   OCH.sub.3                                        CH     391        CH.sub.3             H  PhCO     H   OCH.sub.3                                  OCH.sub.3                                        N     392        CH.sub.3             H  PhCO     H   OCH.sub.3                                  CH.sub.3                                        N     393        CH.sub.3             H  PhCO     H   OCH.sub.3                                  CF.sub.3                                        N     394        CH.sub.3             H  PhCO     CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     395        CH.sub.3             H  PhCO     CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     396        CH.sub.3             H  PhSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     397        CH.sub.3             H  PhSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     398        CH.sub.3             H  PhSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     399        CH.sub.3             H  PhSO.sub.2                         H   Cl   OCH.sub.3                                        CH     400        CH.sub.3             H  PhSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     401        CH.sub.3             H  PhSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     402        CH.sub.3             H  PhSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     403        CH.sub.3             H  PhSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     404        CH.sub.3             H  PhSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     405        CH.sub.3             H  MeNHCO   H   OCH.sub.3                                  OCH.sub.3                                        CH     406        CH.sub.3             H  MeNHCO   H   OCH.sub.3                                  CH.sub.3                                        CH     407        CH.sub.3             H  MeNHCO   H   CH.sub.3                                  CH.sub.3                                        CH     408        CH.sub.3             H  MeNHCO   H   Cl   OCH.sub.3                                        CH     409        CH.sub.3             H  MeNHCO   H   OCH.sub.3                                  OCH.sub.3                                        N     410        CH.sub.3             H  MeNHCO   H   OCH.sub.3                                  CH.sub.3                                        N     411        CH.sub.3             H  MeNHCO   H   OCH.sub.3                                  CF.sub.3                                        N - 412                                           CH.sub.3 H MeNHCO CH.sub.3 OCH.sub.3                                           9OCH.sub.3 CH     413        CH.sub.3             H  MeNHCO   CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     414        CH.sub.3             H  EtNHCO   H   OCH.sub.3                                  OCH.sub.3                                        CH     415        CH.sub.3             H  EtNHCO   H   OCH.sub.3                                  CH.sub.3                                        CH     416        CH.sub.3             H  EtNHCO   H   CH.sub.3                                  CH.sub.3                                        CH     417        CH.sub.3             H  EtNHCO   H   Cl   OCH.sub.3                                        CH     418        CH.sub.3             H  EtNHCO   H   OCH.sub.3                                  OCH.sub.3                                        N     419        CH.sub.3             H  EtNHCO   H   OCH.sub.3                                  CH.sub.3                                        N     420        CH.sub.3             H  EtNHCO   H   OCH.sub.3                                  CF.sub.3                                        N     421        CH.sub.3             H  EtNHCO   CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     422        CH.sub.3             H  EtNHCO   CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     423        CH.sub.3             H  MeNHCS   H   OCH.sub.3                                  OCH.sub.3                                        CH     424        CH.sub.3             H  MeNHCS   H   OCH.sub.3                                  CH.sub.3                                        CH     425        CH.sub.3             H  MeNHCS   H   CH.sub.3                                  CH.sub.3                                        CH     426        CH.sub.3             H  MeNHCS   H   Cl   OCH.sub.3                                        CH     427        CH.sub.3             H  MeNHCS   H   OCH.sub.3                                  OCH.sub.3                                        N     428        CH.sub.3             H  MeNHCS   H   OCH.sub.3                                  CH.sub.3                                        N     429        CH.sub.3             H  MeNHCS   H   OCH.sub.3                                  CF.sub.3                                        N     430        CH.sub.3             H  MeNHCS   CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     431        CH.sub.3             H  MeNHCS   CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     432        CH.sub.3             H  EtNHCS   H   OCH.sub.3                                  OCH.sub.3                                        CH     433        CH.sub.3             H  EtNHCS   H   OCH.sub.3                                  CH.sub.3                                        CH     434        CH.sub.3             H  EtNHCS   H   CH.sub.3                                  CH.sub.3                                        CH     435        CH.sub.3             H  EtNHCS   H   Cl   OCH.sub.3                                        CH     436        CH.sub.3             H  EtNHCS   H   OCH.sub.3                                  OCH.sub.3                                        N     437        CH.sub.3             H  EtNHCS   H   OCH.sub.3                                  CH.sub.3                                        N     438        CH.sub.3             H  EtNHCS   H   OCH.sub.3                                  CF.sub.3                                        N     439        CH.sub.3             H  EtNHCS   CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     440        CH.sub.3             H  EtNHCS   CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     441        CH.sub.3             6 #STR52##  H   OCH.sub.3                                  OCH.sub.3                                        CH     442        CH.sub.3             6 #STR53##  H   OCH.sub.3                                  CH.sub.3                                        CH     443        CH.sub.3             6 #STR54##  H   CH.sub.3                                  CH.sub.3                                        CH     444        CH.sub.3             6 #STR55##  H   Cl   OCH.sub.3                                        CH     445        CH.sub.3             6 #STR56##  H   OCH.sub.3                                  OCH.sub.3                                        N     446        CH.sub.3             6 #STR57##  H   OCH.sub.3                                  CH.sub.3                                        N     447        CH.sub.3             6 #STR58##  H   OCH.sub.3                                  CF.sub.3                                        N     448        CH.sub.3             6 #STR59##  CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     449        CH.sub.3             6 #STR60##  CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     450        CH.sub.3             7 #STR61##  H   OCH.sub.3                                  OCH.sub.3                                        CH     451        CH.sub.3             7 #STR62##  H   OCH.sub.3                                  CH.sub.3                                        CH     452        CH.sub.3             7 #STR63##  H   CH.sub.3                                  CH.sub.3                                        CH     453        CH.sub.3             7 #STR64##  H   Cl   OCH.sub.3                                        CH     454        CH.sub.3             7 #STR65##  H   OCH.sub.3                                  OCH.sub.3                                        N     455        CH.sub.3             7 #STR66##  H   OCH.sub.3                                  CH.sub.3                                        N     456        CH.sub.3             7 #STR67##  H   OCH.sub.3                                  CF.sub.3                                        N     457        CH.sub.3             7 #STR68##  CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     458        CH.sub.3             7 #STR69##  CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     459        CH.sub.3             8 #STR70##  H   OCH.sub.3                                  OCH.sub.3                                        CH     460        CH.sub.3             8 #STR71##  H   OCH.sub.3                                  CH.sub.3                                        CH     461        CH.sub.3             8 #STR72##  H   CH.sub.3                                  CH.sub.3                                        CH     462        CH.sub.3             8 #STR73##  H   Cl   OCH.sub.3                                        CH     463        CH.sub.3             8 #STR74##  H   OCH.sub.3                                  OCH.sub.3                                        N     464        CH.sub.3             8 #STR75##  H   OCH.sub.3                                  CH.sub.3                                        N     465        CH.sub.3             8 #STR76##  H   OCH.sub.3                                  CF.sub.3                                        N     466        CH.sub.3             8 #STR77##  CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     467        CH.sub.3             8 #STR78##  CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     468        CH.sub.3             9 #STR79##  H   OCH.sub.3                                  OCH.sub.3                                        CH     469        CH.sub.3             9 #STR80##  H   OCH.sub.3                                  CH.sub.3                                        CH     470        CH.sub.3             9 #STR81##  H   CH.sub.3                                  CH.sub.3                                        CH     471        CH.sub.3             9 #STR82##  H   Cl   OCH.sub.3                                        CH     472        CH.sub.3             9 #STR83##  H   OCH.sub.3                                  OCH.sub.3                                        N     473        CH.sub.3             9 #STR84##  H   OCH.sub.3                                  CH.sub.3                                        N     474        CH.sub.3             9 #STR85##  H   OCH.sub.3                                  CF.sub.3                                        N     475        CH.sub.3             9 #STR86##  CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     476        CH.sub.3             9 #STR87##  CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     477        CH.sub.3             0 #STR88##  H   OCH.sub.3                                  OCH.sub.3                                        CH     478        CH.sub.3             0 #STR89##  H   OCH.sub.3                                  CH.sub.3                                        CH     479        CH.sub.3             0 #STR90##  H   CH.sub.3                                  CH.sub.3                                        CH     480        CH.sub.3             0 #STR91##  H   Cl   OCH.sub.3                                        CH     481        CH.sub.3             0 #STR92##  H   OCH.sub.3                                  OCH.sub.3                                        N     482        CH.sub.3             0 #STR93##  H   OCH.sub.3                                  CH.sub.3                                        N     483        CH.sub.3             0 #STR94##  H   OCH.sub.3                                  CF.sub.3                                        N     484        CH.sub.3             0 #STR95##  CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     485        CH.sub.3             0 #STR96##  CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     486        CH.sub.3             H  COSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     487        CH.sub.3             H  COSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     488        CH.sub.3             H  COSCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     489        CH.sub.3             H  COSCH.sub.3                         H   Cl   OCH.sub.3                                        CH     490        CH.sub.3             H  COSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     491        CH.sub.3             H  COSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     492        CH.sub.3             H  COSCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     493        CH.sub.3             H  COSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     494        CH.sub.3             H  COSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     495        CH.sub.3             H  COSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     496        CH.sub.3             H  COSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     497        CH.sub.3             H  COSCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     498        CH.sub.3             H  COSCH.sub.3                         H   Cl   OCH.sub.3                                        CH     499        CH.sub.3             H  COSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     500        CH.sub.3             H  COSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     501        CH.sub.3             H  COSCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     502        CH.sub.3             H  CSOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     503        CH.sub.3             H  CSOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     504        CH.sub.3             H  CSSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     505        CH.sub.3             H  CSSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     506        CH.sub.3             H  CSSCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     507        CH.sub.3             H  CSSCH.sub.3                         H   Cl   OCH.sub.3                                        CH     508        CH.sub.3             H  CSSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     509        CH.sub.3             H  CSSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     510        CH.sub.3             H  CSSCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     511        CH.sub.3             H  CSSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     512        CH.sub.3             H  CSSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     513        CH.sub.3             H  COCOOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     514        CH.sub.3             H  COCOOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     515        CH.sub.3             H  COCOOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     516        CH.sub.3             H  COCOOCH.sub.3                         H   Cl   OCH.sub.3                                        CH     517        CH.sub.3             H  COCOOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     518        CH.sub.3             H  COCOOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     519        CH.sub.3             H  COCOOCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     520        CH.sub.3             H  COCOOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     521        CH.sub.3             H  COCOOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     522        CH.sub.3             H  i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     523        CH.sub.3             H  i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     524        CH.sub.3             H  i-C.sub.3 H.sub.7 OCO                         H   CH.sub.3                                  CH.sub.3                                        CH     525        CH.sub.3             H  i-C.sub.3 H.sub.7 OCO                         H   Cl   OCH.sub.3                                        CH     526        CH.sub.3             H  i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     527        CH.sub.3             H  i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  CH.sub.3                                        N     528        CH.sub.3             H  i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  CF.sub.3                                        N     529        CH.sub.3             H  i-C.sub.3 H.sub.7 OCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     530        CH.sub.3             H  i-C.sub.3 H.sub.7 OCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     531        CH.sub.3             CH.sub.3                CHO      H   OCH.sub.3                                  OCH.sub.3                                        CH 180-182     532        CH.sub.3             CH.sub.3                CHO      H   OCH.sub.3                                  CH.sub.3                                        CH     533        CH.sub.3             CH.sub.3                CHO      H   CH.sub.3                                  CH.sub.3                                        CH     534        CH.sub.3             CH.sub.3                CHO      H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     535        CH.sub.3             CH.sub.3                CHO      H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     536        CH.sub.3             CH.sub.3                CHO      H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     537        CH.sub.3             CH.sub.3                CHO      H   OCHF.sub.2                                  OCHF.sub.2                                        CH     538        CH.sub.3             CH.sub.3                CHO      H   CH.sub.3                                  OCHF.sub.2                                        CH     539        CH.sub.3             CH.sub.3                CHO      H   Cl   OCH.sub.3                                        CH     540        CH.sub.3             CH.sub.3                CHO      H   OCH.sub.3                                  OCH.sub.3                                        N     541        CH.sub.3             CH.sub.3                CHO      H   OCH.sub.3                                  CH.sub.3                                        N     542        CH.sub.3             CH.sub.3                CHO      H   CH.sub.3                                  CH.sub.3                                        N     543        CH.sub.3             CH.sub.3                CHO      H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     544        CH.sub.3             CH.sub.3                CHO      H   OCH.sub.3                                  CF.sub.3                                        N     545        CH.sub.3             CH.sub.3                CHO      H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     546        CH.sub.3             CH.sub.3                CHO      CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     547        CH.sub.3             CH.sub.3                CHO      CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     548        CH.sub.3             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 133-136     549        CH.sub.3             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     550        CH.sub.3             CH.sub.3                COCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     551        CH.sub.3             CH.sub.3                COCH.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     552        CH.sub.3             CH.sub.3                COCH.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     553        CH.sub.3             CH.sub.3                COCH.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     554        CH.sub.3             CH.sub.3                COCH.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     555        CH.sub.3             CH.sub.3                COCH.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     556        CH.sub.3             CH.sub.3                COCH.sub.3                         H   Cl   OCH.sub.3                                        CH     557        CH.sub.3             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     558        CH.sub.3             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     559        CH.sub.3             CH.sub.3                COCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     560        CH.sub.3             CH.sub.3                COCH.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     561        CH.sub.3             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     562        CH.sub.3             CH.sub.3                COCH.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     563        CH.sub.3             CH.sub.3                COCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     564        CH.sub.3             CH.sub.3                COCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     565        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH 182-185     566        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     567        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     568        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     569        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     570        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     571        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     572        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   CH.sub.3                                  OCHF.sub.2                                        CH     573        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     574        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     575        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     576        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        N     577        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     578        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     579        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     580        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     581        CH.sub.3             CH.sub.3                COC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     582        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH     583        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     584        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     585        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     586        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     587        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     588        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     589        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     590        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     591        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     592        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     593        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     594        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     595        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     596        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     597        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     598        CH.sub.3             CH.sub.3                CO-n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     599        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH 186-188     600        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     601        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     602        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     603        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     604        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     605        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     606        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     607        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     608        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     609        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     610        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     611        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     612        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     613        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     614        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     615        CH.sub.3             CH.sub.3                CO-i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     616        CH.sub.3             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 133-136     617        CH.sub.3             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     618        CH.sub.3             CH.sub.3                COCF.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     619        CH.sub.3             CH.sub.3                COCF.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     620        CH.sub.3             CH.sub.3                COCF.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     621        CH.sub.3             CH.sub.3                COCF.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     622        CH.sub.3             CH.sub.3                COCF.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     623        CH.sub.3             CH.sub.3                COCF.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     624        CH.sub.3             CH.sub.3                COCF.sub.3                         H   Cl   OCH.sub.3                                        CH     625        CH.sub.3             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     626        CH.sub.3             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     627        CH.sub.3             CH.sub.3                COCF.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     628        CH.sub.3             CH.sub.3                COCF.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     629        CH.sub.3             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     630        CH.sub.3             CH.sub.3                COCF.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     631        CH.sub.3             CH.sub.3                COCF.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     632        CH.sub.3             CH.sub.3                COCF.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     633        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 105-111     634        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     635        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     636        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     637        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     638        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     639        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     640        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     641        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   Cl   OCH.sub.3                                        CH     642        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     643        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     644        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     645        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     646        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     647        CH.sub.3             CH.sub.3                COOCH.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     648        CH.sub.3             CH.sub.3                COOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     649        CH.sub.3             CH.sub.3                COOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     650        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH 227-229     651        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     652        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     653        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     654        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     655        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     656        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     657        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   CH.sub.3                                  OCHF.sub.2                                        CH     658        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     659        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     660        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     661        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        N     662        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     663        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     664        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     665        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     666        CH.sub.3             CH.sub.3                COOC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     667        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 205-210     668        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     669        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     670        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     671        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     672        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     673        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     674        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     675        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   Cl   OCH.sub.3                                        CH     676        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     677        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     678        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     679        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     680        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     681        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     682        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     683        CH.sub.3             CH.sub.3                SO.sub.2 CH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     684        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH 206-208     685        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     686        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     687        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     688        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     689        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     690        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     691        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  OCHF.sub.2                                        CH     692        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     693        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     694        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     695        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        N     696        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     697        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     698        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     699        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     700        CH.sub.3             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     701        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH     702        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     703        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     704        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     705        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     706        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     707        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     708        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     709        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     710        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     711        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     712        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     713        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     714        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     715        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     716        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     717        CH.sub.3             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     718        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH     719        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     720        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     721        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     722        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     723        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     724        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     725        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     726        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     727        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     728        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     729        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     730        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     731        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     732        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     733        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     734        CH.sub.3             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     735        CH.sub.3             CH.sub.3                ClCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     736        CH.sub.3             CH.sub.3                ClCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        CH     737        CH.sub.3             CH.sub.3                ClCH.sub.2 CO                         H   CH.sub.3                                  CH.sub.3                                        CH     738        CH.sub.3             CH.sub.3                ClCH.sub.2 CO                         H   Cl   OCH.sub.3                                        CH     739        CH.sub.3             CH.sub.3                ClCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        N     740        CH.sub.3             CH.sub.3                ClCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        N     741        CH.sub.3             CH.sub.3                ClCH.sub.2 CO                         H   OCH.sub.3                                  CF.sub.3                                        N     742        CH.sub.3             CH.sub.3                ClCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     743        CH.sub.3             CH.sub.3                ClCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     744        CH.sub.3             CH.sub.3                Cl.sub.2 CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     745        CH.sub.3             CH.sub.3                Cl.sub.2 CHCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     746        CH.sub.3             CH.sub.3                Cl.sub.2 CHCO                         H   CH.sub.3                                  CH.sub.3                                        CH     747        CH.sub.3             CH.sub.3                Cl.sub.2 CHCO                         H   Cl   OCH.sub.3                                        CH     748        CH.sub.3             CH.sub.3                Cl.sub.2 CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     749        CH.sub.3             CH.sub.3                Cl.sub.2 CHCO                         H   OCH.sub.3                                  CH.sub.3                                        N     750        CH.sub.3             CH.sub.3                Cl.sub.2 CHCO                         H   OCH.sub.3                                  CF.sub.3                                        N     751        CH.sub.3             CH.sub.3                Cl.sub.2 CHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     752        CH.sub.3             CH.sub.3                Cl.sub.2 CHCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     753        CH.sub.3             CH.sub.3                Cl.sub.2 CCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH 144-146     754        CH.sub.3             CH.sub.3                Cl.sub.2 CCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     755        CH.sub.3             CH.sub.3                Cl.sub.2 CCO                         H   CH.sub.3                                  CH.sub.3                                        CH     756        CH.sub.3             CH.sub.3                Cl.sub.2 CCO                         H   Cl   OCH.sub.3                                        CH     757        CH.sub.3             CH.sub.3                Cl.sub.2 CCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     758        CH.sub.3             CH.sub.3                Cl.sub.2 CCO                         H   OCH.sub.3                                  CH.sub.3                                        N     759        CH.sub.3             CH.sub.3                Cl.sub.2 CCO                         H   OCH.sub.3                                  CF.sub.3                                        N     760        CH.sub.3             CH.sub.3                Cl.sub.2 CCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     761        CH.sub.3             CH.sub.3                Cl.sub.2 CCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     762        CH.sub.3             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     763        CH.sub.3             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        CH     764        CH.sub.3             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   CH.sub.3                                  CH.sub.3                                        CH     765        CH.sub.3             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   Cl   OCH.sub.3                                        CH     766        CH.sub.3             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        N     767        CH.sub.3             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        N     768        CH.sub.3             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  CF.sub.3                                        N     769        CH.sub.3             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     770        CH.sub.3             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     771        CH.sub.3             CH.sub.3                CH.sub.2 ═CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     772        CH.sub.3             CH.sub.3                CH.sub.2 ═CHCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     773        CH.sub.3             CH.sub.3                CH.sub.2 ═CHCO                         H   CH.sub.3                                  CH.sub.3                                        CH     774        CH.sub.3             CH.sub.3                CH.sub.2 ═CHCO                         H   Cl   OCH.sub.3                                        CH     775        CH.sub.3             CH.sub.3                CH.sub.2 ═CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     776        CH.sub.3             CH.sub.3                CH.sub.2 ═CHCO                         H   OCH.sub.3                                  CH.sub.3                                        N     777        CH.sub.3             CH.sub.3                CH.sub.2 ═CHCO                         H   OCH.sub.3                                  CF.sub.3                                        N     778        CH.sub.3             CH.sub.3                CH.sub.2 ═CHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     779        CH.sub.3             CH.sub.3                CH.sub.2 ═CHCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     780        CH.sub.3             CH.sub.3                CH.tbd.CCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     781        CH.sub.3             CH.sub.3                CH.tbd.CCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     782        CH.sub.3             CH.sub.3                CH.tbd.CCO                         H   CH.sub.3                                  CH.sub.3                                        CH     783        CH.sub.3             CH.sub.3                CH.tbd.CCO                         H   Cl   OCH.sub.3                                        CH     784        CH.sub.3             CH.sub.3                CH.tbd.CCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     785        CH.sub.3             CH.sub.3                CH.tbd.CCO                         H   OCH.sub.3                                  CH.sub.3                                        N     786        CH.sub.3             CH.sub.3                CH.tbd.CCO                         H   OCH.sub.3                                  CF.sub.3                                        N     787        CH.sub.3             CH.sub.3                CH.tbd.CCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     788        CH.sub.3             CH.sub.3                CH.tbd.CCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     789        CH.sub.3             CH.sub.3                2 #STR97##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     790        CH.sub.3             CH.sub.3                2 #STR98##                         H   OCH.sub.3                                  CH.sub.3                                        CH     791        CH.sub.3             CH.sub.3                2 #STR99##                         H   CH.sub.3                                  CH.sub.3                                        CH     792        CH.sub.3             CH.sub.3                2 #STR100##                         H   Cl   OCH.sub.3                                        CH     793        CH.sub.3             CH.sub.3                2 #STR101##                         H   OCH.sub.3                                  OCH.sub.3                                        N     794        CH.sub.3             CH.sub.3                2 #STR102##                         H   OCH.sub.3                                  CH.sub.3                                        N     795        CH.sub.3             CH.sub.3                2 #STR103##                         H   OCH.sub.3                                  CF.sub.3                                        N     796        CH.sub.3             CH.sub.3                2 #STR104##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     797        CH.sub.3             CH.sub.3                2 #STR105##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     798        CH.sub.3             CH.sub.3                3 #STR106##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     799        CH.sub.3             CH.sub.3                3 #STR107##                         H   OCH.sub.3                                  CH.sub.3                                        CH     800        CH.sub.3             CH.sub.3                3 #STR108##                         H   CH.sub.3                                  CH.sub.3                                        CH     801        CH.sub.3             CH.sub.3                3 #STR109##                         H   Cl   OCH.sub.3                                        CH     802        CH.sub.3             CH.sub.3                3 #STR110##                         H   OCH.sub.3                                  OCH.sub.3                                        N     803        CH.sub.3             CH.sub.3                3 #STR111##                         H   OCH.sub.3                                  CH.sub.3                                        N     804        CH.sub.3             CH.sub.3                3 #STR112##                         H   OCH.sub.3                                  CF.sub.3                                        N     805        CH.sub.3             CH.sub.3                3 #STR113##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     806        CH.sub.3             CH.sub.3                3 #STR114##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     807        CH.sub.3             CH.sub.3                4 #STR115##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     808        CH.sub.3             CH.sub.3                4 #STR116##                         H   OCH.sub.3                                  CH.sub.3                                        CH     809        CH.sub.3             CH.sub.3                4 #STR117##                         H   CH.sub.3                                  CH.sub.3                                        CH     810        CH.sub.3             CH.sub.3                4 #STR118##                         H   Cl   OCH.sub.3                                        CH     811        CH.sub.3             CH.sub.3                4 #STR119##                         H   OCH.sub.3                                  OCH.sub.3                                        N     812        CH.sub.3             CH.sub.3                4 #STR120##                         H   OCH.sub.3                                  CH.sub.3                                        N     813        CH.sub.3             CH.sub.3                4 #STR121##                         H   OCH.sub.3                                  CF.sub.3                                        N     814        CH.sub.3             CH.sub.3                4 #STR122##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     815        CH.sub.3             CH.sub.3                4 #STR123##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     816        CH.sub.3             CH.sub.3                5 #STR124##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     817        CH.sub.3             CH.sub.3                5 #STR125##                         H   OCH.sub.3                                  CH.sub.3                                        CH     818        CH.sub.3             CH.sub.3                5 #STR126##                         H   CH.sub.3                                  CH.sub.3                                        CH     819        CH.sub.3             CH.sub.3                5 #STR127##                         H   Cl   OCH.sub.3                                        CH     820        CH.sub.3             CH.sub.3                5 #STR128##                         H   OCH.sub.3                                  OCH.sub.3                                        N     821        CH.sub.3             CH.sub.3                5 #STR129##                         H   OCH.sub.3                                  CH.sub.3                                        N     822        CH.sub.3             CH.sub.3                5 #STR130##                         H   OCH.sub.3                                  CF.sub.3                                        N     823        CH.sub.3             CH.sub.3                5 #STR131##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     824        CH.sub.3             CH.sub.3                5 #STR132##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     825        CH.sub.3             CH.sub.3                CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     826        CH.sub.3             CH.sub.3                CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     827        CH.sub.3             CH.sub.3                CF.sub.3 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     828        CH.sub.3             CH.sub.3                CF.sub.3 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     829        CH.sub.3             CH.sub.3                CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     830        CH.sub.3             CH.sub.3                CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     831        CH.sub.3             CH.sub.3                CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     832        CH.sub.3             CH.sub.3                CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH - 833                                           CH.sub.3 CH.sub.3 CF.sub.3 SO.sub.2                                           CH.sub.3 OCH.sub.3 CH.sub.3 N     834        CH.sub.3             CH.sub.3                FCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     835        CH.sub.3             CH.sub.3                FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     836        CH.sub.3             CH.sub.3                FCH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     837        CH.sub.3             CH.sub.3                FCH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     838        CH.sub.3             CH.sub.3                FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     839        CH.sub.3             CH.sub.3                FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     840        CH.sub.3             CH.sub.3                FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     841        CH.sub.3             CH.sub.3                FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     842        CH.sub.3             CH.sub.3                FCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     843        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     844        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     845        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     846        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     847        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     848        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     849        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     850        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     851        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     852        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     853        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     854        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     855        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     856        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     857        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     858        CH.sub.3             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     859        CH.sub.3             CH.sub.3                Cl.sub.2 CHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     860        CH.sub.3             CH.sub.3                Cl.sub.2 CHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     861        CH.sub.3             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     862        CH.sub.3             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     863        CH.sub.3             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     864        CH.sub.3             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   Cl   OCH.sub.3                                        CH     865        CH.sub.3             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     866        CH.sub.3             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     867        CH.sub.3             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     868        CH.sub.3             CH.sub.3                Cl.sub.3 CSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     869        CH.sub.3             CH.sub.3                Cl.sub.3 CSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     870        CH.sub.3             CH.sub.3                n-C.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     871        CH.sub.3             CH.sub.3                n-C.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     872        CH.sub.3             CH.sub.3                n-C.sub.4 H.sub.9 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     873        CH.sub.3             CH.sub.3                n-C.sub.4 H.sub.9 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     874        CH.sub.3             CH.sub.3                n-C.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     875        CH.sub.3             CH.sub.3                n-C.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     876        CH.sub.3             CH.sub.3                n-C.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     877        CH.sub.3             CH.sub.3                n-C.sub.4 H.sub.9 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     878        CH.sub.3             CH.sub.3                n-C.sub.4 H.sub.9 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     879        CH.sub.3             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     880        CH.sub.3             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     881        CH.sub.3             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     882        CH.sub.3             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     883        CH.sub.3             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     884        CH.sub.3             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     885        CH.sub.3             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     886        CH.sub.3             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     887        CH.sub.3             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     888        CH.sub.3             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     889        CH.sub.3             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     890        CH.sub.3             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     891        CH.sub.3             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   Cl   OCH.sub.3                                        CH     892        CH.sub.3             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     893        CH.sub.3             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     894        CH.sub.3             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     895        CH.sub.3             CH.sub.3                CH.sub.3 NHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     896        CH.sub.3             CH.sub.3                CH.sub.3 NHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     897        CH.sub.3             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     898        CH.sub.3             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     899        CH.sub.3             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     900        CH.sub.3             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   Cl   OCH.sub.3                                        CH     901        CH.sub.3             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     902        CH.sub.3             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     903        CH.sub.3             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     904        CH.sub.3             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     905        CH.sub.3             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     906        CH.sub.3             CH.sub.3                (CH.sub.3).sub.3 COCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     907        CH.sub.3             CH.sub.3                (CH.sub.3).sub.3 COCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     908        CH.sub.3             CH.sub.3                (CH.sub.3).sub.3 COCO                         H   CH.sub.3                                  CH.sub.3                                        CH     909        CH.sub.3             CH.sub.3                (CH.sub.3).sub.3 COCO                         H   Cl   OCH.sub.3                                        CH     910        CH.sub.3             CH.sub.3                (CH.sub.3).sub.3 COCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     911        CH.sub.3             CH.sub.3                (CH.sub.3).sub.3 COCO                         H   OCH.sub.3                                  CH.sub.3                                        N     912        CH.sub.3             CH.sub.3                (CH.sub.3).sub.3 COCO                         H   OCH.sub.3                                  CF.sub.3                                        N     913        CH.sub.3             CH.sub.3                (CH.sub.3).sub.3 COCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     914        CH.sub.3             CH.sub.3                (CH.sub.3).sub.3 COCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     915        CH.sub.3             CH.sub.3                PhCO     H   OCH.sub.3                                  OCH.sub.3                                        CH     916        CH.sub.3             CH.sub.3                PhCO     H   OCH.sub.3                                  CH.sub.3                                        CH     917        CH.sub.3             CH.sub.3                PhCO     H   CH.sub.3                                  CH.sub.3                                        CH     918        CH.sub.3             CH.sub.3                PhCO     H   Cl   OCH.sub.3                                        CH     919        CH.sub.3             CH.sub.3                PhCO     H   OCH.sub.3                                  OCH.sub.3                                        N     920        CH.sub.3             CH.sub.3                PhCO     H   OCH.sub.3                                  CH.sub.3                                        N     921        CH.sub.3             CH.sub.3                PhCO     H   OCH.sub.3                                  CF.sub.3                                        N     922        CH.sub.3             CH.sub.3                PhCO     CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     923        CH.sub.3             CH.sub.3                PhCO     CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     924        CH.sub.3             CH.sub.3                PhSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     925        CH.sub.3             CH.sub.3                PhSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     926        CH.sub.3             CH.sub.3                PhSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     927        CH.sub.3             CH.sub.3                PhSO.sub.2                         H   Cl   OCH.sub.3                                        CH     928        CH.sub.3             CH.sub.3                PhSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     929        CH.sub.3             CH.sub.3                PhSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     930        CH.sub.3             CH.sub.3                PhSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     931        CH.sub.3             CH.sub.3                PhSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     932        CH.sub.3             CH.sub.3                PhSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     933        CH.sub.3             CH.sub.3                CH.sub.3 NHCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     934        CH.sub.3             CH.sub.3                CH.sub.3 NHCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     935        CH.sub.3             CH.sub.3                CH.sub.3 NHCO                         H   CH.sub.3                                  CH.sub.3                                        CH     936        CH.sub.3             CH.sub.3                CH.sub.3 NHCO                         H   Cl   OCH.sub.3                                        CH     937        CH.sub.3             CH.sub.3                CH.sub.3 NHCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     938        CH.sub.3             CH.sub.3                CH.sub.3 NHCO                         H   OCH.sub.3                                  CH.sub.3                                        N     939        CH.sub.3             CH.sub.3                CH.sub.3 NHCO                         H   OCH.sub.3                                  CF.sub.3                                        N     940        CH.sub.3             CH.sub.3                CH.sub.3 NHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     941        CH.sub.3             CH.sub.3                CH.sub.3 NHCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     942        CH.sub.3             CH.sub.3                EtNHCO   H   OCH.sub.3                                  OCH.sub.3                                        CH     943        CH.sub.3             CH.sub.3                EtNHCO   H   OCH.sub.3                                  CH.sub.3                                        CH     944        CH.sub.3             CH.sub.3                EtNHCO   H   CH.sub.3                                  CH.sub.3                                        CH     945        CH.sub.3             CH.sub.3                EtNHCO   H   Cl   OCH.sub.3                                        CH     946        CH.sub.3             CH.sub.3                EtNHCO   H   OCH.sub.3                                  OCH.sub.3                                        N     947        CH.sub.3             CH.sub.3                EtNHCO   H   OCH.sub.3                                  CH.sub.3                                        N     948        CH.sub.3             CH.sub.3                EtNHCO   H   OCH.sub.3                                  CF.sub.3                                        N     949        CH.sub.3             CH.sub.3                EtNHCO   CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     950        CH.sub.3             CH.sub.3                EtNHCO   CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     951        CH.sub.3             CH.sub.3                CH.sub.3 NHCS                         H   OCH.sub.3                                  OCH.sub.3                                        CH     952        CH.sub.3             CH.sub.3                CH.sub.3 NHCS                         H   OCH.sub.3                                  CH.sub.3                                        CH     953        CH.sub.3             CH.sub.3                CH.sub.3 NHCS                         H   CH.sub.3                                  CH.sub.3                                        CH     954        CH.sub.3             CH.sub.3                CH.sub.3 NHCS                         H   Cl   OCH.sub.3                                        CH     955        CH.sub.3             CH.sub.3                CH.sub.3 NHCS                         H   OCH.sub.3                                  OCH.sub.3                                        N     956        CH.sub.3             CH.sub.3                CH.sub.3 NHCS                         H   OCH.sub.3                                  CH.sub.3                                        N     957        CH.sub.3             CH.sub.3                CH.sub.3 NHCS                         H   OCH.sub.3                                  CF.sub.3                                        N     958        CH.sub.3             CH.sub.3                CH.sub.3 NHCS                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     959        CH.sub.3             CH.sub.3                CH.sub.3 NHCS                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     960        CH.sub.3             CH.sub.3                EtNHCS   H   OCH.sub.3                                  OCH.sub.3                                        CH     961        CH.sub.3             CH.sub.3                EtNHCS   H   OCH.sub.3                                  CH.sub.3                                        CH     962        CH.sub.3             CH.sub.3                EtNHCS   H   CH.sub.3                                  CH.sub.3                                        CH     963        CH.sub.3             CH.sub.3                EtNHCS   H   Cl   OCH.sub.3                                        CH     964        CH.sub.3             CH.sub.3                EtNHCS   H   OCH.sub.3                                  OCH.sub.3                                        N     965        CH.sub.3             CH.sub.3                EtNHCS   H   OCH.sub.3                                  CH.sub.3                                        N     966        CH.sub.3             CH.sub.3                EtNHCS   H   OCH.sub.3                                  CF.sub.3                                        N     967        CH.sub.3             CH.sub.3                EtNHCS   CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     968        CH.sub.3             CH.sub.3                EtNHCS   CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     969        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     970        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     971        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     972        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   Cl   OCH.sub.3                                        CH     973        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     974        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     975        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     976        CH.sub.3             CH.sub.3                COSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     977        CH.sub.3             CH.sub.3                COSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     978        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     979        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     980        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     981        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   Cl   OCH.sub.3                                        CH     982        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     983        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     984        CH.sub.3             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     985        CH.sub.3             CH.sub.3                CSOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     986        CH.sub.3             CH.sub.3                CSOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     987        CH.sub.3             CH.sub.3                CSSCH.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     988        CH.sub.3             CH.sub.3                CSSCH.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     989        CH.sub.3             CH.sub.3                CSSCH.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     990        CH.sub.3             CH.sub.3                CSSCH.sub.2                         H   Cl   OCH.sub.3                                        CH     991        CH.sub.3             CH.sub.3                CSSCH.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     992        CH.sub.3             CH.sub.3                CSSCH.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     993        CH.sub.3             CH.sub.3                CSSCH.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     994        CH.sub.3             CH.sub.3                CSSCH.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     995        CH.sub.3             CH.sub.3                CSSCH.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     996        CH.sub.3             CH.sub.3                COCOOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     997        CH.sub.3             CH.sub.3                COCOOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     998        CH.sub.3             CH.sub.3                COCOOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     999        CH.sub.3             CH.sub.3                COCOOCH.sub.3                         H   Cl   OCH.sub.3                                        CH     1000        CH.sub.3             CH.sub.3                COCOOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1001        CH.sub.3             CH.sub.3                COCOOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1002        CH.sub.3             CH.sub.3                COCOOCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1003        CH.sub.3             CH.sub.3                COCOOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1004        CH.sub.3             CH.sub.3                COCOOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1005        CH.sub.3             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1006        CH.sub.3             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1007        CH.sub.3             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   CH.sub.3                                  CH.sub.3                                        CH     1008        CH.sub.3             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   Cl   OCH.sub.3                                        CH     1009        CH.sub.3             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1010        CH.sub.3             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  CH.sub.3                                        N     1011        CH.sub.3             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  CF.sub.3                                        N     1012        CH.sub.3             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1013        CH.sub.3             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1014        CH.sub.3             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  OCH.sub.3                                        CH     1015        CH.sub.3             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  CH.sub.3                                        CH     1016        CH.sub.3             C.sub.2 H.sub.5                CHO      H   CH.sub.3                                  CH.sub.3                                        CH     1017        CH.sub.3             C.sub.2 H.sub.5                CHO      H   Cl   OCH.sub.3                                        CH     1018        CH.sub.3             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  OCH.sub.3                                        N     1019        CH.sub.3             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  CH.sub.3                                        N     1020        CH.sub.3             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  CF.sub.3                                        N     1021        CH.sub.3             C.sub.2 H.sub.5                CHO      CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1022        CH.sub.3             C.sub.2 H.sub.5                CHO      CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1023        CH.sub.3             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1024        CH.sub.3             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1025        CH.sub.3             C.sub.2 H.sub.5                COCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1026        CH.sub.3             C.sub.2 H.sub.5                COCH.sub.3                         H   Cl   OCH.sub.3                                        CH     1027        CH.sub.3             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1028        CH.sub.3             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1029        CH.sub.3             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1030        CH.sub.3             C.sub.2 H.sub.5                COCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1031        CH.sub.3             C.sub.2 H.sub.5                COCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1032        CH.sub.3             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1033        CH.sub.3             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1034        CH.sub.3             C.sub.2 H.sub.5                COOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1035        CH.sub.3             C.sub.2 H.sub.5                COOCH.sub.3                         H   Cl   OCH.sub.3                                        CH     1036        CH.sub.3             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1037        CH.sub.3             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1038        CH.sub.3             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1039        CH.sub.3             C.sub.2 H.sub.5                COOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1040        CH.sub.3             C.sub.2 H.sub.5                COOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1041        CH.sub.3             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1042        CH.sub.3             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     1043        CH.sub.3             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     1044        CH.sub.3             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     1045        CH.sub.3             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     1046        CH.sub.3             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     1047        CH.sub.3             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     1048        CH.sub.3             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1049        CH.sub.3             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1050        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1051        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1052        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1053        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   Cl   OCH.sub.3                                        CH     1054        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1055        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1056        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1057        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1058        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1059        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1060        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     1061        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     1062        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     1063        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     1064        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     1065        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     1066        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1067        CH.sub.3             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1068        C.sub.2 H.sub.5             H  CHO      H   OCH.sub.3                                  OCH.sub.3                                        CH 146-147     1069        C.sub.2 H.sub.5             H  CHO      H   OCH.sub.3                                  CH.sub.3                                        CH     1070        C.sub.2 H.sub.5             H  CHO      H   CH.sub.3                                  CH.sub.3                                        CH     1071        C.sub.2 H.sub.5             H  CHO      H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1072        C.sub.2 H.sub.5             H  CHO      H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1073        C.sub.2 H.sub.5             H  CHO      H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1074        C.sub.2 H.sub.5             H  CHO      H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1075        C.sub.2 H.sub.5             H  CHO      H   CH.sub.3                                  OCHF.sub.2                                        CH     1076        C.sub.2 H.sub.5             H  CHO      H   Cl   OCH.sub.3                                        CH     1077        C.sub.2 H.sub.5             H  CHO      H   OCH.sub.3                                  OCH.sub.3                                        N     1078        C.sub.2 H.sub.5             H  CHO      H   OCH.sub.3                                  CH.sub.3                                        N     1079        C.sub.2 H.sub.5             H  CHO      H   CH.sub.3                                  CH.sub.3                                        N     1080        C.sub.2 H.sub.5             H  CHO      H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1081        C.sub.2 H.sub.5             H  CHO      H   OCH.sub.3                                  CF.sub.3                                        N     1082        C.sub.2 H.sub.5             H  CHO      H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1083        C.sub.2 H.sub.5             H  CHO      CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1084        C.sub.2 H.sub.5             H  CHO      CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1085        C.sub.2 H.sub.5             H  COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 126-128     1086        C.sub.2 H.sub.5             H  COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1087        C.sub.2 H.sub.5             H  COCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1088        C.sub.2 H.sub.5             H  COCH.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1089        C.sub.2 H.sub.5             H  COCH.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1090        C.sub.2 H.sub.5             H  COCH.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1091        C.sub.2 H.sub.5             H  COCH.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1092        C.sub.2 H.sub.5             H  COCH.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1093        C.sub.2 H.sub.5             H  COCH.sub.3                         H   Cl   OCH.sub.3                                        CH     1094        C.sub.2 H.sub.5             H  COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1095        C.sub.2 H.sub.5             H  COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1096        C.sub.2 H.sub.5             H  COCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     1097        C.sub.2 H.sub.5             H  COCH.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1098        C.sub.2 H.sub.5             H  COCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1099        C.sub.2 H.sub.5             H  COCH.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1100        C.sub.2 H.sub.5             H  COCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1101        C.sub.2 H.sub.5             H  COCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1102        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1103        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     1104        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     1105        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1106        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1107        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1108        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1109        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1110        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     1111        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     1112        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     1113        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        N     1114        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1115        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     1116        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1117        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1118        C.sub.2 H.sub.5             H  COC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1119        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1120        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     1121        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     1122        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1123        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1124        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1125        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1126        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1127        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     1128        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     1129        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     1130        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     1131        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1132        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     1133        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1134        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1135        C.sub.2 H.sub.5             H  CO-n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1136        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1137        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     1138        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     1139        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1140        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1141        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1142        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1143        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1144        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     1145        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     1146        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     1147        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     1148        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1149        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     1150        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1151        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1152        C.sub.2 H.sub.5             H  CO-i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1153        C.sub.2 H.sub.5             H  COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1154        C.sub.2 H.sub.5             H  COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1155        C.sub.2 H.sub.5             H  COCF.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1156        C.sub.2 H.sub.5             H  COCF.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1157        C.sub.2 H.sub.5             H  COCF.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1158        C.sub.2 H.sub.5             H  COCF.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1159        C.sub.2 H.sub.5             H  COCF.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1160        C.sub.2 H.sub.5             H  COCF.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1161        C.sub.2 H.sub.5             H  COCF.sub.3                         H   Cl   OCH.sub.3                                        CH     1162        C.sub.2 H.sub.5             H  COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1163        C.sub.2 H.sub.5             H  COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1164        C.sub.2 H.sub.5             H  COCF.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     1165        C.sub.2 H.sub.5             H  COCF.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1166        C.sub.2 H.sub.5             H  COCF.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1167        C.sub.2 H.sub.5             H  COCF.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1168        C.sub.2 H.sub.5             H  COCF.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1169        C.sub.2 H.sub.5             H  COCF.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1170        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 132-136     1170        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1171        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1172        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1173        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1174        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1175        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1176        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1177        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   Cl   OCH.sub.3                                        CH     1178        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1179        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1180        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     1181        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1182        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1183        C.sub.2 H.sub.5             H  COOCH.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1184        C.sub.2 H.sub.5             H  COOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1185        C.sub.2 H.sub.5             H  COOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1186        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1186        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     a     1187        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     1188        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1189        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1190        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1191        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1192        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1193        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     1194        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     1195        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     1196        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        N     1197        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1198        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     1199        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1200        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1201        C.sub.2 H.sub.5             H  COOC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1202        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 130-132     1202        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     a     1203        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1204        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1205        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1206        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1207        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1208        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1209        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   Cl   OCH.sub.3                                        CH     1210        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1211        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1212        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     1213        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1214        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1215        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1216        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1217        C.sub.2 H.sub.5             H  SO.sub.2 CH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1218        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1218        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     a     1219        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     1220        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1221        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1222        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1223        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1224        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1225        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     1226        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     1227        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     1228        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        N     1229        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1230        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.2                                  CF.sub.3                                        N     1231        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1232        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1233        C.sub.2 H.sub.5             H  SO.sub.2 C.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1234        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1234        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     a     1235        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     1236        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1237        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1238        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1239        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1240        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1241        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     1242        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     1243        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     1244        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     1245        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1246        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     1247        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1248        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1249        C.sub.2 H.sub.5             H  SO.sub.2 -n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1250        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1250        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     a     1251        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     1252        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1253        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1254        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1255        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1256        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1257        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     1258        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     1259        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     1260        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     1261        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1262        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     1263        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1264        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1265        C.sub.2 H.sub.5             H  SO.sub.2 -i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1266        C.sub.2 H.sub.5             H  ClCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1267        C.sub.2 H.sub.5             H  ClCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1268        C.sub.2 H.sub.5             H  ClCH.sub.2 CO                         H   CH.sub.3                                  CH.sub.3                                        CH     1269        C.sub.2 H.sub.5             H  ClCH.sub.2 CO                         H   Cl   OCH.sub.3                                        CH     1270        C.sub.2 H.sub.5             H  ClCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1271        C.sub.2 H.sub.5             H  ClCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        N     1272        C.sub.2 H.sub.5             H  ClCH.sub.2 CO                         H   OCH.sub.3                                  CF.sub.3                                        N     1273        C.sub.2 H.sub.5             H  ClCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1274        C.sub.2 H.sub.5             H  ClCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1275        C.sub.2 H.sub.5             H  Cl.sub.2 CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1276        C.sub.2 H.sub.5             H  Cl.sub.2 CHCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1277        C.sub.2 H.sub.5             H  Cl.sub.2 CHCO                         H   CH.sub.3                                  CH.sub.3                                        CH     1278        C.sub.2 H.sub.5             H  Cl.sub.2 CHCO                         H   Cl   OCH.sub.3                                        CH     1279        C.sub.2 H.sub.5             H  Cl.sub.2 CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1280        C.sub.2 H.sub.5             H  Cl.sub.2 CHCO                         H   OCH.sub.3                                  CH.sub.3                                        N     1281        C.sub.2 H.sub.5             H  Cl.sub.2 CHCO                         H   OCH.sub.3                                  CF.sub.3                                        N     1282        C.sub.2 H.sub.5             H  Cl.sub.2 CHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1283        C.sub.2 H.sub.5             H  Cl.sub.2 CHCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1284        C.sub.2 H.sub.5             H  Cl.sub.3 CCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1285        C.sub.2 H.sub.5             H  Cl.sub.3 CCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1286        C.sub.2 H.sub.5             H  Cl.sub.3 CCO                         H   CH.sub.3                                  CH.sub.3                                        CH     1287        C.sub.2 H.sub.5             H  Cl.sub.3 CCO                         H   Cl   OCH.sub.3                                        CH     1288        C.sub.2 H.sub.5             H  Cl.sub.3 CCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1289        C.sub.2 H.sub.5             H  Cl.sub.3 CCO                         H   OCH.sub.3                                  CH.sub.3                                        N     1290        C.sub.2 H.sub.5             H  Cl.sub.3 CCO                         H   OCH.sub.3                                  CF.sub.3                                        N     1291        C.sub.2 H.sub.5             H  Cl.sub.3 CCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1292        C.sub.2 H.sub.5             H  Cl.sub.3 CCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1293        C.sub.2 H.sub.5             H  CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1294        C.sub.2 H.sub.5             H  CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1295        C.sub.2 H.sub.5             H  CH.sub.3 OCH.sub.2 CO                         H   CH.sub.3                                  CH.sub.3                                        CH     1296        C.sub.2 H.sub.5             H  CH.sub.3 OCH.sub.2 CO                         H   Cl   OCH.sub.3                                        CH     1297        C.sub.2 H.sub.5             H  CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1298        C.sub.2 H.sub.5             H  CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        N     1299        C.sub.2 H.sub.5             H  CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  CF.sub.3                                        N     1300        C.sub.2 H.sub.5             H  CH.sub.3 OCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1301        C.sub.2 H.sub.5             H  CH.sub.3 OCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1302        C.sub.2 H.sub.5             H  CH.sub.2 ═CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1303        C.sub.2 H.sub.5             H  CH.sub.2 ═CHCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1304        C.sub.2 H.sub.5             H  CH.sub.2 ═CHCO                         H   CH.sub.3                                  CH.sub.3                                        CH     1305        C.sub.2 H.sub.5             H  CH.sub.2 ═CHCO                         H   Cl   OCH.sub.3                                        CH     1306        C.sub.2 H.sub.5             H  CH.sub.2 ═CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1307        C.sub.2 H.sub.5             H  CH.sub.2 ═CHCO                         H   OCH.sub.3                                  CH.sub.3                                        N     1308        C.sub.2 H.sub.5             H  CH.sub.2 ═CHCO                         H   OCH.sub.3                                  CF.sub.3                                        N     1309        C.sub.2 H.sub.5             H  CH.sub.2 ═CHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1310        C.sub.2 H.sub.5             H  CH.sub.2 ═CHCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1311        C.sub.2 H.sub.5             H  CH.tbd.CCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1312        C.sub.2 H.sub.5             H  CH.tbd.CCO                         H   OC.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1313        C.sub.2 H.sub.5             H  CH.tbd.CCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1314        C.sub.2 H.sub.5             H  CH.tbd.CCO                         H   CH.sub.3                                  CH.sub.3                                        CH     1315        C.sub.2 H.sub.5             H  CH.tbd.CCO                         H   Cl   OCH.sub.3                                        CH     1316        C.sub.2 H.sub.5             H  CH.tbd.CCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1317        C.sub.2 H.sub.5             H  CH.tbd.CCO                         H   OCH.sub.3                                  CH.sub.3                                        N     1318        C.sub.2 H.sub.5             H  CH.tbd.CCO                         H   OCH.sub.3                                  CF.sub.3                                        N     1319        C.sub.2 H.sub.5             H  CH.tbd.CCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1320        C.sub.2 H.sub.5             H  CH.tbd.CCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1321        C.sub.2 H.sub.5             H                2 #STR133##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1322        C.sub.2 H.sub.5             H                2 #STR134##                         H   OCH.sub.3                                  CH.sub.3                                        CH     1323        C.sub.2 H.sub.5             H                2 #STR135##                         H   CH.sub.3                                  CH.sub.3                                        CH     1324        C.sub.2 H.sub.5             H                2 #STR136##                         H   Cl   OCH.sub.3                                        CH     1325        C.sub.2 H.sub.5             H                2 #STR137##                         H   OCH.sub.3                                  OCH.sub.3                                        N     1326        C.sub.2 H.sub.5             H                2 #STR138##                         H   OCH.sub.3                                  CH.sub.3                                        N     1327        C.sub.2 H.sub.5             H                2 #STR139##                         H   OCH.sub.3                                  CF.sub.3                                        N     1328        C.sub.2 H.sub.5             H                2 #STR140##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1329        C.sub.2 H.sub.5             H                2 #STR141##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1330        C.sub.2 H.sub.5             H                3 #STR142##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1331        C.sub.2 H.sub.5             H                3 #STR143##                         H   OCH.sub.3                                  CH.sub.3                                        CH     1332        C.sub.2 H.sub.5             H                3 #STR144##                         H   CH.sub.3                                  CH.sub.3                                        CH     1333        C.sub.2 H.sub.5             H                3 #STR145##                         H   Cl   OCH.sub.3                                        CH     1334        C.sub.2 H.sub.5             H                3 #STR146##                         H   OCH.sub.3                                  OCH.sub.3                                        N     1335        C.sub.2 H.sub.5             H                3 #STR147##                         H   OCH.sub.3                                  CH.sub.3                                        N     1336        C.sub.2 H.sub.5             H                3 #STR148##                         H   OCH.sub.3                                  CF.sub.3                                        N     1337        C.sub.2 H.sub.5             H                3 #STR149##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1338        C.sub.2 H.sub.5             H                3 #STR150##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1339        C.sub.2 H.sub.5             H                4 #STR151##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1340        C.sub.2 H.sub.5             H                4 #STR152##                         H   OCH.sub.3                                  CH.sub.3                                        CH     1341        C.sub.2 H.sub.5             H                4 #STR153##                         H   CH.sub.3                                  CH.sub.3                                        CH     1342        C.sub.2 H.sub.5             H                4 #STR154##                         H   Cl   OCH.sub.3                                        CH     1343        C.sub.2 H.sub.5             H                4 #STR155##                         H   OCH.sub.3                                  OCH.sub.3                                        N     1344        C.sub.2 H.sub.5             H                4 #STR156##                         H   OCH.sub.3                                  OCH.sub.3                                        N     1345        C.sub.2 H.sub.5             H                4 #STR157##                         H   OCH.sub.3                                  CF.sub.3                                        N     1346        C.sub.2 H.sub.5             H                4 #STR158##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1347        C.sub.2 H.sub.5             H                4 #STR159##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1348        C.sub.2 H.sub.5             H                4 #STR160##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1349        C.sub.2 H.sub.5             H                5 #STR161##                         H   OCH.sub.3                                  CH.sub.3                                        CH     1350        C.sub.2 H.sub.5             H                5 #STR162##                         H   CH.sub.3                                  CH.sub.3                                        CH     1351        C.sub.2 H.sub.5             H                5 #STR163##                         H   Cl   OCH.sub.3                                        CH     1352        C.sub.2 H.sub.5             H                5 #STR164##                         H   OCH.sub.3                                  OCH.sub.3                                        N     1353        C.sub.2 H.sub.5             H                5 #STR165##                         H   OCH.sub.3                                  CH.sub.3                                        N     1354        C.sub.2 H.sub.5             H                5 #STR166##                         H   OCH.sub.3                                  CF.sub.3                                        N     1355        C.sub.2 H.sub.5             H                5 #STR167##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1356        C.sub.2 H.sub.5             H                5 #STR168##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1357        C.sub.2 H.sub.5             H  CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1358        C.sub.2 H.sub.5             H  CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1359        C.sub.2 H.sub.5             H  CF.sub.3 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1360        C.sub.2 H.sub.5             H  CF.sub.3 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     1361        C.sub.2 H.sub.5             H  CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1362        C.sub.2 H.sub.5             H  CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1363        C.sub.2 H.sub.5             H  CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1364        C.sub.2 H.sub.5             H  CF.sub.3 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        CH     1365        C.sub.2 H.sub.5             H  CF.sub.3 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        N     1366        C.sub.2 H.sub.5             H  FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1367        C.sub.2 H.sub.5             H  FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1368        C.sub.2 H.sub.5             H  FCH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1369        C.sub.2 H.sub.5             H  FCH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     1370        C.sub.2 H.sub.5             H  FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1371        C.sub.2 H.sub.5             H  FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1372        C.sub.2 H.sub.5             H  FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1373        C.sub.2 H.sub.5             H  FCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1374        C.sub.2 H.sub.5             H  FCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        N     1375        C.sub.2 H.sub.5             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1376        C.sub.2 H.sub.5             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1377        C.sub.2 H.sub.5             H  ClCH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1378        C.sub.2 H.sub.5             H  ClCH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     1379        C.sub.2 H.sub.5             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1380        C.sub.2 H.sub.5             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1381        C.sub.2 H.sub.5             H  ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1382        C.sub.2 H.sub.5             H  ClCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1383        C.sub.2 H.sub.5             H  ClCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1384        C.sub.2 H.sub.5             H  Cl.sub.2 CHSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1385        C.sub.2 H.sub.5             H  Cl.sub.2 CHSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1386        C.sub.2 H.sub.5             H  Cl.sub.2 CHSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1387        C.sub.2 H.sub.5             H  Cl.sub.2 CHSO.sub.2                         H   Cl   OCH.sub.3                                        CH     1388        C.sub.2 H.sub.5             H  Cl.sub.2 CHSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1389        C.sub.2 H.sub.5             H  Cl.sub.2 CHSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1390        C.sub.2 H.sub.5             H  Cl.sub.2 CHSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1391        C.sub.2 H.sub.5             H  Cl.sub.2 CHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1392        C.sub.2 H.sub.5             H  Cl.sub.2 CHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1393        C.sub.2 H.sub.5             H  Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1394        C.sub.2 H.sub.5             H  Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1395        C.sub.2 H.sub.5             H  Cl.sub.3 CSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1396        C.sub.2 H.sub.5             H  Cl.sub.3 CSO.sub.2                         H   Cl   OCH.sub.3                                        CH     1397        C.sub.2 H.sub.5             H  Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1398        C.sub.2 H.sub.5             H  Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1399        C.sub.2 H.sub.5             H  Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1400        C.sub.2 H.sub.5             H  Cl.sub.3 CSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1401        C.sub.2 H.sub.5             H  Cl.sub.3 CSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1402        C.sub.2 H.sub.5             H  n-C.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1403        C.sub.2 H.sub.5             H  n-C.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1404        C.sub.2 H.sub.5             H  n-C.sub.4 H.sub.9 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1405        C.sub.2 H.sub.5             H  n-C.sub.4 H.sub.9 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     1406        C.sub.2 H.sub.5             H  n-C.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1407        C.sub.2 H.sub.5             H  n-C.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1408        C.sub.2 H.sub.5             H  n-C.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1409        C.sub.2 H.sub.5             H  n-C.sub.4 H.sub.9 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        CH     1410        C.sub.2 H.sub.5             H  n-C.sub.4 H.sub.9 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        N     1411        C.sub.2 H.sub.5             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1412        C.sub.2 H.sub.5             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1413        C.sub.2 H.sub.5             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1414        C.sub.2 H.sub.5             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     1415        C.sub.2 H.sub.5             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1416        C.sub.2 H.sub.5             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1417        C.sub.2 H.sub.5             H  CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1418        C.sub.2 H.sub.5             H  CF.sub.3 CH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1419        C.sub.2 H.sub.5             H  CF.sub.3 CH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        N     1420        C.sub.2 H.sub.5             H  CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1421        C.sub.2 H.sub.5             H  CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1422        C.sub.2 H.sub.5             H  CH.sub.3 NHSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1423        C.sub.2 H.sub.5             H  CH.sub.3 NHSO.sub.2                         H   Cl   OCH.sub.3                                        CH     1424        C.sub.2 H.sub.5             H  CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1425        C.sub.2 H.sub.5             H  CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1426        C.sub.2 H.sub.5             H  CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1427        C.sub.2 H.sub.5             H  CH.sub.3 NHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1428        C.sub.2 H.sub.5             H  CH.sub.3 NHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1429        C.sub.2 H.sub.5             H  (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1430        C.sub.2 H.sub.5             H  (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1431        C.sub.2 H.sub.5             H  (CH.sub.3).sub.2 NSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1432        C.sub.2 H.sub.5             H  (CH.sub.3).sub.2 NSO.sub.2                         H   Cl   OCH.sub.3                                        CH     1433        C.sub.2 H.sub.5             H  (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1434        C.sub.2 H.sub.5             H  (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1435        C.sub.2 H.sub.5             H  (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1436        C.sub.2 H.sub.5             H  (CH.sub.3).sub.2 NSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1437        C.sub.2 H.sub.5             H  (CH.sub.3).sub.2 NSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1438        C.sub.2 H.sub.5             H  (CH.sub.3).sub.3 C--                         H   OCH.sub.3                                  OCH.sub.3                                        CH                OCO     1439        C.sub.2 H.sub.5             H  (CH.sub.3).sub.3 C--                         H   OCH.sub.3                                  CH.sub.3                                        CH                OCO     1440        C.sub.2 H.sub.5             H  (CH.sub.3).sub.3 C--                         H   CH.sub.3                                  CH.sub.3                                        CH                OCO     1441        C.sub.2 H.sub.5             H  (CH.sub.3).sub.3 C--                         H   Cl   OCH.sub.3                                        CH                OCO     1442        C.sub.2 H.sub.5             H  (CH.sub.3).sub.3 C--                         H   OCH.sub.3                                  OCH.sub.3                                        N                OCO     1443        C.sub.2 H.sub.5             H  (CH.sub.3).sub.3 C--                         H   OCH.sub.3                                  CH.sub.3                                        N                OCO     1444        C.sub.2 H.sub.5             H  (CH.sub.3).sub.3 C--                         H   OCH.sub.3                                  CF.sub.3                                        N                OCO     1445        C.sub.2 H.sub.5             H  (CH.sub.3).sub.3 C--                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH                OCO     1446        C.sub.2 H.sub.5             H  (CH.sub.3).sub.3 C--                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N                OCO     1447        C.sub.2 H.sub.5             H  PhCO     H   OCH.sub.3                                  OCH.sub.3                                        CH     1448        C.sub.2 H.sub.5             H  PhCO     H   OCH.sub.3                                  CH.sub.3                                        CH     1449        C.sub.2 H.sub.5             H  PhCO     H   CH.sub.3                                  CH.sub.3                                        CH     1450        C.sub.2 H.sub.5             H  PhCO     H   Cl   OCH.sub.3                                        CH     1451        C.sub.2 H.sub.5             H  PhCO     H   OCH.sub.3                                  OCH.sub.3                                        N     1452        C.sub.2 H.sub.5             H  PhCO     H   OCH.sub.3                                  CH.sub.3                                        N     1453        C.sub.2 H.sub.5             H  PhCO     H   OCH.sub.3                                  CF.sub.3                                        N     1454        C.sub.2 H.sub.5             H  PhCO     CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1455        C.sub.2 H.sub.5             H  PhCO     CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1456        C.sub.2 H.sub.5             H  PhSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1457        C.sub.2 H.sub.5             H  PhSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1458        C.sub.2 H.sub.5             H  PhSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1459        C.sub.2 H.sub.5             H  PhSO.sub.2                         H   Cl   OCH.sub.3                                        CH     1460        C.sub.2 H.sub.5             H  PhSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1461        C.sub.2 H.sub.5             H  PhSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1462        C.sub.2 H.sub.5             H  PhSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1463        C.sub.2 H.sub.5             H  PhSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1464        C.sub.2 H.sub.5             H  PhSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        N     1465        C.sub.2 H.sub.5             H  CH.sub.3 NHCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1466        C.sub.2 H.sub.5             H  CH.sub.3 NHCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1467        C.sub.2 H.sub.5             H  CH.sub.3 NHCO                         H   CH.sub.3                                  CH.sub.3                                        CH     1468        C.sub.2 H.sub.5             H  CH.sub.3 NHCO                         H   Cl   OCH.sub.3                                        CH     1469        C.sub.2 H.sub.5             H  CH.sub.3 NHCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1470        C.sub.2 H.sub.5             H  CH.sub.3 NHCO                         H   OCH.sub.3                                  CH.sub.3                                        N     1471        C.sub.2 H.sub.5             H  CH.sub.3 NHCO                         H   OCH.sub.3                                  CF.sub.3                                        N     1472        C.sub.2 H.sub.5             H  CH.sub.3 NHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1473        C.sub.2 H.sub.5             H  CH.sub.3 NHCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1474        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1475        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1476        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCO                         H   CH.sub.3                                  CH.sub.3                                        CH     1477        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCO                         H   Cl   OCH.sub.3                                        CH     1478        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1479        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCO                         H   OCH.sub.3                                  CH.sub.3                                        N     1480        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCO                         H   OCH.sub.3                                  CF.sub.3                                        N     1481        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1482        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1483        C.sub.2 H.sub.5             H  CH.sub.3 NHCS                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1484        C.sub.2 H.sub.5             H  CH.sub.3 NHCS                         H   OCH.sub.3                                  CH.sub.3                                        CH     1485        C.sub.2 H.sub.5             H  CH.sub.3 NHCS                         H   CH.sub.3                                  CH.sub.3                                        CH     1486        C.sub.2 H.sub.5             H  CH.sub.3 NHCS                         H   Cl   OCH.sub.3                                        CH     1487        C.sub.2 H.sub.5             H  CH.sub.3 NHCS                         H   OCH.sub.3                                  OCH.sub.3                                        N     1488        C.sub.2 H.sub.5             H  CH.sub.3 NHCS                         H   OCH.sub.3                                  CH.sub.3                                        N     1489        C.sub.2 H.sub.5             H  CH.sub.3 NHCS                         H   OCH.sub.3                                  CF.sub.3                                        N     1490        C.sub.2 H.sub.5             H  CH.sub.3 NHCS                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1491        C.sub.2 H.sub.5             H  CH.sub.3 NHCS                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1492        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCS                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1493        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCS                         H   OCH.sub.3                                  CH.sub.3                                        CH     1494        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCS                         H   CH.sub.3                                  CH.sub.3                                        CH     1495        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCS                         H   Cl   OCH.sub.3                                        CH     1496        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCS                         H   OCH.sub.3                                  CH.sub.3                                        N     1497        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCS                         H   OCH.sub.3                                  CF.sub.3                                        N     1498        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCS                         H   OCH.sub.3                                  OCH.sub.3                                        N     1499        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCS                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        CH     1500        C.sub.2 H.sub.5             H  C.sub.2 H.sub.5 NHCS                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        N     1501        C.sub.2 H.sub.5             6 #STR169## H   OCH.sub.3                                  OCH.sub.3                                        CH     1502        C.sub.2 H.sub.5             6 #STR170## H   OCH.sub.3                                  CH.sub.3                                        CH     1503        C.sub.2 H.sub.5             6 #STR171## H   CH.sub.3                                  CH.sub.3                                        CH     1504        C.sub.2 H.sub.5             6 #STR172## H   Cl   OCH.sub.3                                        CH     1505        C.sub.2 H.sub.5             6 #STR173## H   OCH.sub.3                                  OCH.sub.3                                        N     1506        C.sub.2 H.sub.5             6 #STR174## H   OCH.sub.3                                  CH.sub.3                                        N     1507        C.sub.2 H.sub.5             6 #STR175## H   OCH.sub.3                                  CF.sub.3                                        N     1508        C.sub.2 H.sub.5             6 #STR176## CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1509        C.sub.2 H.sub.5             6 #STR177## H   OCH.sub.3                                  OCH.sub.3                                        CH     1510        C.sub.2 H.sub.5             7 #STR178## H   OCH.sub.3                                  OCH.sub.3                                        CH     1511        C.sub.2 H.sub.5             7 #STR179## H   OCH.sub.3                                  CH.sub.3                                        CH     1512        C.sub.2 H.sub.5             7 #STR180## H   CH.sub.3                                  CH.sub.3                                        CH     1513        C.sub.2 H.sub.5             7 #STR181## H   Cl   OCH.sub.3                                        CH     1514        C.sub.2 H.sub.5             7 #STR182## H   OCH.sub.3                                  OCH.sub.3                                        N     1515        C.sub.2 H.sub.5             7 #STR183## H   OCH.sub.3                                  CH.sub.3                                        N     1516        C.sub.2 H.sub.5             7 #STR184## H   OCH.sub.3                                  CF.sub.3                                        N     1517        C.sub.2 H.sub.5             7 #STR185## CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1518        C.sub.2 H.sub.5             7 #STR186## CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1519        C.sub.2 H.sub.5             8 #STR187## H   OCH.sub.3                                  OCH.sub.3                                        CH     1520        C.sub.2 H.sub.5             8 #STR188## H   OCH.sub.3                                  CH.sub.3                                        CH     1521        C.sub.2 H.sub.5             8 #STR189## H   CH.sub.3                                  CH.sub.3                                        CH     1522        C.sub.2 H.sub.5             8 #STR190## H   Cl   OCH.sub.3                                        CH     1523        C.sub.2 H.sub.5             8 #STR191## H   OCH.sub.3                                  OCH.sub.3                                        N     1524        C.sub.2 H.sub.5             8 #STR192## H   OCH.sub.3                                  CH.sub.3                                        N     1525        C.sub.2 H.sub.5             8 #STR193## H   OCH.sub.3                                  CF.sub.3                                        N     1526        C.sub.2 H.sub.5             8 #STR194## CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1527        C.sub.2 H.sub.5             8 #STR195## CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1528        C.sub.2 H.sub.5             9 #STR196## H   OCH.sub.3                                  OCH.sub.3                                        CH     1529        C.sub.2 H.sub.5             9 #STR197## H   OCH.sub.3                                  CH.sub.3                                        CH     1530        C.sub.2 H.sub.5             9 #STR198## H   CH.sub.3                                  CH.sub.3                                        CH     1531        C.sub.2 H.sub.5             9 #STR199## H   Cl   OCH.sub.3                                        CH     1532        C.sub.2 H.sub.5             9 #STR200## H   OCH.sub.3                                  OCH.sub.3                                        N     1533        C.sub.2 H.sub.5             9 #STR201## H   OCH.sub.3                                  CH.sub.3                                        N     1534        C.sub.2 H.sub.5             9 #STR202## H   OCH.sub.3                                  CF.sub.3                                        N     1535        C.sub.2 H.sub.5             9 #STR203## CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1536        C.sub.2 H.sub.5             9 #STR204## CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1537        C.sub.2 H.sub.5             0 #STR205## H   OCH.sub.3                                  OCH.sub.3                                        CH     1538        C.sub.2 H.sub.5             0 #STR206## H   OCH.sub.3                                  CH.sub.3                                        CH     1539        C.sub.2 H.sub.5             0 #STR207## H   CH.sub.3                                  CH.sub.3                                        CH     1540        C.sub.2 H.sub.5             0 #STR208## H   Cl   OCH.sub.3                                        CH     1541        C.sub.2 H.sub.5             0 #STR209## H   OCH.sub.3                                  CH.sub.3                                        N     1542        C.sub.2 H.sub.5             0 #STR210## H   OCH.sub.3                                  CF.sub.3                                        N     1543        C.sub.2 H.sub.5             0 #STR211## H   OCH.sub.3                                  OCH.sub.3                                        N     1544        C.sub.2 H.sub.5             0 #STR212## CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        CH     1545        C.sub.2 H.sub.5             0 #STR213## CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        N     1546        C.sub.2 H.sub.5             H  COSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1547        C.sub.2 H.sub.5             H  COSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1548        C.sub.2 H.sub.5             H  COSCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1549        C.sub.2 H.sub.5             H  COSCH.sub.3                         H   Cl   OCH.sub.3                                        CH     1550        C.sub.2 H.sub.5             H  COSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1551        C.sub.2 H.sub.5             H  COSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1552        C.sub.2 H.sub.5             H  COSCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1553        C.sub.2 H.sub.5             H  COSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1554        C.sub.2 H.sub.5             H  COSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1555        C.sub.2 H.sub.5             H  CSOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1556        C.sub.2 H.sub.5             H  CSOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1557        C.sub.2 H.sub.5             H  CSOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1558        C.sub.2 H.sub.5             H  CSOCH.sub.3                         H   Cl   OCH.sub.3                                        CH     1559        C.sub.2 H.sub.5             H  CSOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1560        C.sub.2 H.sub.5             H  CSOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1561        C.sub.2 H.sub.5             H  CSOCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1562        C.sub.2 H.sub.5             H  CSOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1563        C.sub.2 H.sub.5             H  CSOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1564        C.sub.2 H.sub.5             H  CSSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1565        C.sub.2 H.sub.5             H  CSSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1566        C.sub.2 H.sub.5             H  CSSCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1567        C.sub.2 H.sub.5             H  CSSCH.sub.3                         H   Cl   OCH.sub.3                                        CH     1568        C.sub.2 H.sub.5             H  CSSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1569        C.sub.2 H.sub.5             H  CSSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1570        C.sub.2 H.sub.5             H  CSSCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1571        C.sub.2 H.sub.5             H  CSSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1572        C.sub.2 H.sub.5             H  CSSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1573        C.sub.2 H.sub.5             H  COCOOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1574        C.sub.2 H.sub.5             H  COCOOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1575        C.sub.2 H.sub.5             H  COCOOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1576        C.sub.2 H.sub.5             H  COCOOCH.sub.3                         H   Cl   OCH.sub.3                                        CH     1577        C.sub.2 H.sub.5             H  COCOOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1578        C.sub.2 H.sub.5             H  COCOOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1579        C.sub.2 H.sub.5             H  COCOOCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1580        C.sub.2 H.sub.5             H  COCOOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1581        C.sub.2 H.sub.5             H  COCOOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1582        C.sub.2 H.sub.5             H  i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1583        C.sub.2 H.sub.5             H  i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1584        C.sub.2 H.sub.5             H  i-C.sub.3 H.sub.7 OCO                         H   CH.sub.3                                  CH.sub.3                                        CH     1585        C.sub.2 H.sub.5             H  i-C.sub.3 H.sub.7 OCO                         H   Cl   OCH.sub.3                                        CH     1586        C.sub.2 H.sub.5             H  i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1587        C.sub.2 H.sub.5             H  i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  CH.sub.3                                        N     1588        C.sub.2 H.sub.5             H  i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1589        C.sub.2 H.sub.5             H  i-C.sub.3 H.sub.7 OCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        CH     1590        C.sub.2 H.sub.5             H  i-C.sub.3 H.sub.7 OCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        N     1591        C.sub.2 H.sub.5             CH.sub.3                CHO      H   OCH.sub.3                                  OCH.sub.3                                        CH 212-213     1592        C.sub.2 H.sub.5             CH.sub.3                CHO      H   OCH.sub.3                                  CH.sub.3                                        CH     1593        C.sub.2 H.sub.5             CH.sub.3                CHO      H   CH.sub.3                                  CH.sub.3                                        CH     1594        C.sub.2 H.sub.5             CH.sub.3                CHO      H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1595        C.sub.2 H.sub.5             CH.sub.3                CHO      H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1596        C.sub.2 H.sub.5             CH.sub.3                CHO      H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1597        C.sub.2 H.sub.5             CH.sub.3                CHO      H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1598        C.sub.2 H.sub.5             CH.sub.3                CHO      H   CH.sub.3                                  OCHF.sub.2                                        CH     1599        C.sub.2 H.sub.5             CH.sub.3                CHO      H   Cl   OCH.sub.3                                        CH     1600        C.sub.2 H.sub.5             CH.sub.3                CHO      H   OCH.sub.3                                  OCH.sub.3                                        N     1601        C.sub.2 H.sub.5             CH.sub.3                CHO      H   OCH.sub.3                                  CH.sub.3                                        N     1602        C.sub.2 H.sub.5             CH.sub.3                CHO      H   CH.sub.3                                  CH.sub.3                                        N     1603        C.sub.2 H.sub.5             CH.sub.3                CHO      H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1604        C.sub.2 H.sub.5             CH.sub.3                CHO      H   OCH.sub.3                                  CF.sub.3                                        N     1605        C.sub.2 H.sub.5             CH.sub.3                CHO      H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1606        C.sub.2 H.sub.5             CH.sub.3                CHO      CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1607        C.sub.2 H.sub.5             CH.sub.3                CHO      CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1608        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 174-176     1609        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1610        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1611        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1612        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1613        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1614        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1615        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1616        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   Cl   OCH.sub.3                                        CH     1617        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1618        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1619        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     1620        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1621        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1622        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1623        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1624        C.sub.2 H.sub.5             CH.sub.3                COCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1625        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1626        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     1627        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     1628        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1629        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1630        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1631        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1632        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1633        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     1634        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     1635        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     1636        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        N     1637        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1638        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     1639        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1640        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1641        C.sub.2 H.sub.5             CH.sub.3                COC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1642        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1643        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     1644        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     1645        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1646        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1647        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1648        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1649        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1650        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     1651        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     1652        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     1653        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     1654        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1655        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     1656        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1657        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1658        C.sub.2 H.sub.5             CH.sub.3                CO-n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1659        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1660        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     1661        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     1662        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1663        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1664        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1665        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1666        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1667        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     1668        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     1669        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     1670        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     1671        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1672        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     1673        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1674        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1675        C.sub.2 H.sub.5             CH.sub.3                CO-i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1676        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 201-202     1677        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1678        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1679        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1680        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1681        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1682        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1683        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1684        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   Cl   OCH.sub.3                                        CH     1685        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1686        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1687        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     1688        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1689        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1690        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1691        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1692        C.sub.2 H.sub.5             CH.sub.3                COCF.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1693        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1694        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1695        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1696        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1697        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1698        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1699        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1700        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1701        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   Cl   OCH.sub.3                                        CH     1702        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1703        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1704        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     1705        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1706        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1707        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1708        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1709        C.sub.2 H.sub.5             CH.sub.3                COOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1710        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1711        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     1712        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     1713        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1714        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1715        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1716        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1717        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1718        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     1719        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     1720        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     1721        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        N     1722        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1723        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     1724        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1725        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1726        C.sub.2 H.sub.5             CH.sub.3                COOC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1727        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 195-196     1728        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     1729        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     1730        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1731        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1732        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1733        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1734        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1735        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   Cl   OCH.sub.3                                        CH     1736        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     1737        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     1738        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        N     1739        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1740        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     1741        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1742        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1743        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 CH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1744        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1745        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     1746        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     1747        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1748        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1749        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1750        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1751        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1752        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     1753        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     1754        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     1755        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        N     1756        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1757        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     1758        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1759        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1760        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1761        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1762        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     1763        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     1764        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1765        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1766        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1767        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1768        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1769        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     1770        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     1771        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     1772        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     1773        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1774        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     1775        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1776        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1777        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -n-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1778        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1779        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        CH     1780        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        CH     1781        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OC.sub.2 H.sub.5                                        CH     1782        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   C.sub.2 H.sub.5                                  OCH.sub.3                                        CH     1783        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  OC.sub.2 H.sub.5                                        CH     1784        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCHF.sub.2                                  OCHF.sub.2                                        CH     1785        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   CH.sub.3                                  OCHF.sub.2                                        CH     1786        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   Cl   OCH.sub.3                                        CH     1787        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  OCH.sub.3                                        N     1788        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CH.sub.3                                        N     1789        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   CH.sub.3                                  CH.sub.3                                        N     1790        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   N(CH.sub.3).sub.2                                  OCH.sub.2 CF.sub.3                                        N     1791        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OCH.sub.3                                  CF.sub.3                                        N     1792        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         H   OC.sub.2 H.sub.5                                  NHCH.sub.3                                        N     1793        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1794        C.sub.2 H.sub.5             CH.sub.3                SO.sub.2 -i-C.sub.3 H.sub.7                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1795        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1796        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1797        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 CO                         H   CH.sub.3                                  CH.sub.3                                        CH     1798        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 CO                         H   Cl   OCH.sub.3                                        CH     1799        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1800        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        N     1801        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 CO                         H   OCH.sub.3                                  CF.sub.3                                        N     1802        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1803        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1804        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1805        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1806        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHCO                         H   CH.sub.3                                  CH.sub.3                                        CH     1807        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHCO                         H   Cl   OCH.sub.3                                        CH     1808        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1809        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHCO                         H   OCH.sub.3                                  CH.sub.3                                        N     1810        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHCO                         H   OCH.sub.3                                  CF.sub.3                                        N     1811        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1812        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        N     1813        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1814        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1815        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CCO                         H   CH.sub.3                                  CH.sub.3                                        CH     1816        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CCO                         H   Cl   OCH.sub.3                                        CH     1817        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1818        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CCO                         H   OCH.sub.3                                  CH.sub.3                                        N     1819        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CCO                         H   OCH.sub.3                                  CF.sub.3                                        N     1820        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1821        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1822        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1823        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1824        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   CH.sub.3                                  CH.sub.3                                        CH     1825        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   Cl   OCH.sub.3                                        CH     1826        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1827        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  CH.sub.3                                        N     1828        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         H   OCH.sub.3                                  CF.sub.3                                        N     1829        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1830        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 OCH.sub.2 CO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1831        C.sub.2 H.sub.5             CH.sub.3                CH.sub.2 ═CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1832        C.sub.2 H.sub.5             CH.sub.3                CH.sub.2 ═CHCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1833        C.sub.2 H.sub.5             CH.sub.3                CH.sub.2 ═CHCO                         H   CH.sub.3                                  CH.sub.3                                        CH     1834        C.sub.2 H.sub.5             CH.sub.3                CH.sub.2 ═CHCO                         H   Cl   OCH.sub.3                                        CH     1835        C.sub.2 H.sub.5             CH.sub.3                CH.sub.2 ═CHCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1836        C.sub.2 H.sub.5             CH.sub.3                CH.sub.2 ═CHCO                         H   OCH.sub.3                                  CH.sub.3                                        N     1837        C.sub.2 H.sub.5             CH.sub.3                CH.sub.2 ═CHCO                         H   OCH.sub.3                                  CF.sub.3                                        N     1838        C.sub.2 H.sub.5             CH.sub.3                CH.sub.2 ═CHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1839        C.sub.2 H.sub.5             CH.sub.3                CH.sub.2 ═CHCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1840        C.sub.2 H.sub.5             CH.sub.3                CH.tbd.CCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1841        C.sub.2 H.sub.5             CH.sub.3                CH.tbd.CCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1842        C.sub.2 H.sub.5             CH.sub.3                CH.tbd.CCO                         H   CH.sub.3                                  CH.sub.3                                        CH     1843        C.sub.2 H.sub.5             CH.sub.3                CH.tbd.CCO                         H   Cl   OCH.sub.3                                        CH     1844        C.sub.2 H.sub.5             CH.sub.3                CH.tbd.CCO                         H   OCH.sub.3                                  CH.sub.3                                        N     1845        C.sub.2 H.sub.5             CH.sub.3                CH.tbd.CCO                         H   OCH.sub.3                                  CF.sub.3                                        N     1846        C.sub.2 H.sub.5             CH.sub.3                CH.tbd.CCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1847        C.sub.2 H.sub.5             CH.sub.3                CH.tbd.CCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1848        C.sub.2 H.sub.5             CH.sub.3                CH.tbd.CCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1849        C.sub.2 H.sub.5             CH.sub.3                2 #STR214##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1850        C.sub.2 H.sub.5             CH.sub.3                2 #STR215##                         H   OCH.sub.3                                  CH.sub.3                                        CH     1851        C.sub.2 H.sub.5             CH.sub.3                2 #STR216##                         H   CH.sub.3                                  CH.sub.3                                        CH     1852        C.sub.2 H.sub.5             CH.sub.3                2 #STR217##                         H   Cl   OCH.sub.3                                        CH     1853        C.sub.2 H.sub.5             CH.sub.3                2 #STR218##                         H   OCH.sub.3                                  OCH.sub.3                                        N     1854        C.sub.2 H.sub.5             CH.sub.3                2 #STR219##                         H   OCH.sub.3                                  CH.sub.3                                        N     1855        C.sub.2 H.sub.5             CH.sub.3                2 #STR220##                         H   OCH.sub.3                                  CF.sub.3                                        N     1856        C.sub.2 H.sub.5             CH.sub.3                2 #STR221##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1857        C.sub.2 H.sub.5             CH.sub.3                2 #STR222##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1858        C.sub.2 H.sub.5             CH.sub.3                3 #STR223##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1859        C.sub.2 H.sub.5             CH.sub.3                3 #STR224##                         H   OCH.sub.3                                  CH.sub.3                                        CH     1860        C.sub.2 H.sub.5             CH.sub.3                3 #STR225##                         H   CH.sub.3                                  CH.sub.3                                        CH     1861        C.sub.2 H.sub.5             CH.sub.3                3 #STR226##                         H   Cl   OCH.sub.3                                        CH     1862        C.sub.2 H.sub.5             CH.sub.3                3 #STR227##                         H   OCH.sub.3                                  OCH.sub.3                                        N     1863        C.sub.2 H.sub.5             CH.sub.3                3 #STR228##                         H   OCH.sub.3                                  CH.sub.3                                        N     1864        C.sub.2 H.sub.5             CH.sub.3                3 #STR229##                         H   OCH.sub.3                                  CF.sub.3                                        N     1865        C.sub.2 H.sub.5             CH.sub.3                3 #STR230##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1866        C.sub.2 H.sub.5             CH.sub.3                3 #STR231##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1867        C.sub.2 H.sub.5             CH.sub.3                4 #STR232##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1868        C.sub.2 H.sub.5             CH.sub.3                4 #STR233##                         H   OCH.sub.3                                  CH.sub.3                                        CH     1869        C.sub.2 H.sub.5             CH.sub.3                4 #STR234##                         H   CH.sub.3                                  CH.sub.3                                        CH     1870        C.sub.2 H.sub.5             CH.sub.3                4 #STR235##                         H   Cl   OCH.sub.3                                        CH     1871        C.sub.2 H.sub.5             CH.sub.3                4 #STR236##                         H   OCH.sub.3                                  OCH.sub.3                                        N     1872        C.sub.2 H.sub.5             CH.sub.3                4 #STR237##                         H   OCH.sub.3                                  CH.sub.3                                        N     1873        C.sub.2 H.sub.5             CH.sub.3                4 #STR238##                         H   OCH.sub.3                                  CF.sub.3                                        N     1874        C.sub.2 H.sub.5             CH.sub.3                4 #STR239##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1875        C.sub.2 H.sub.5             CH.sub.3                4 #STR240##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1876        C.sub.2 H.sub.5             CH.sub.3                5 #STR241##                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1877        C.sub.2 H.sub.5             CH.sub.3                5 #STR242##                         H   OCH.sub.3                                  CH.sub.3                                        CH     1878        C.sub.2 H.sub.5             CH.sub.3                5 #STR243##                         H   CH.sub.3                                  CH.sub.3                                        CH     1879        C.sub.2 H.sub.5             CH.sub.3                5 #STR244##                         H   Cl   OCH.sub.3                                        CH     1880        C.sub.2 H.sub.5             CH.sub.3                5 #STR245##                         H   OCH.sub.3                                  OCH.sub.3                                        N     1881        C.sub.2 H.sub.5             CH.sub.3                5 #STR246##                         H   OCH.sub.3                                  CH.sub.3                                        N     1882        C.sub.2 H.sub.5             CH.sub.3                5 #STR247##                         H   OCH.sub.3                                  CF.sub.3                                        N     1883        C.sub.2 H.sub.5             CH.sub.3                5 #STR248##                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1884        C.sub.2 H.sub.5             CH.sub.3                5 #STR249##                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1885        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1886        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1887        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1888        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     1889        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1890        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1891        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1892        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1893        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1894        C.sub.2 H.sub.5             CH.sub.3                FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1895        C.sub.2 H.sub.5             CH.sub.3                FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1896        C.sub.2 H.sub.5             CH.sub.3                FCH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1897        C.sub.2 H.sub.5             CH.sub.3                FCH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     1898        C.sub.2 H.sub.5             CH.sub.3                FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1899        C.sub.2 H.sub.5             CH.sub.3                FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1900        C.sub.2 H.sub.5             CH.sub.3                FCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1901        C.sub.2 H.sub.5             CH.sub.3                FCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1902        C.sub.2 H.sub.5             CH.sub.3                FCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1903        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1904        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1905        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1906        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     1907        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1908        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1909        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1910        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1911        C.sub.2 H.sub.5             CH.sub.3                ClCH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1912        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1913        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1914        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1915        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHSO.sub.2                         H   Cl   OCH.sub.3                                        CH     1916        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1917        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1918        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1919        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1920        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.2 CHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1921        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1922        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1923        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1924        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   Cl   OCH.sub.3                                        CH     1925        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1926        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1927        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1928        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1929        C.sub.2 H.sub.5             CH.sub.3                Cl.sub.3 CSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1930        C.sub.2 H.sub.5             CH.sub.3                nC.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1931        C.sub.2 H.sub.5             CH.sub.3                nC.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1932        C.sub.2 H.sub.5             CH.sub.3                nC.sub.4 H.sub.9 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1933        C.sub.2 H.sub.5             CH.sub.3                nC.sub.4 H.sub.9 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     1934        C.sub.2 H.sub.5             CH.sub.3                nC.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1935        C.sub.2 H.sub.5             CH.sub.3                nC.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1936        C.sub.2 H.sub.5             CH.sub.3                nC.sub.4 H.sub.9 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1937        C.sub.2 H.sub.5             CH.sub.3                nC.sub.4 H.sub.9 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1938        C.sub.2 H.sub.5             CH.sub.3                nC.sub.4 H.sub.9 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1939        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1940        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1941        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1942        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   Cl   OCH.sub.3                                        CH     1943        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1944        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1945        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1946        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1947        C.sub.2 H.sub.5             CH.sub.3                CF.sub.3 CH.sub.2 SO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1948        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1949        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1950        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1951        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   Cl   OCH.sub.3                                        CH     1952        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1953        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1954        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1955        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1956        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1957        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1958        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1959        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1960        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   Cl   OCH.sub.3                                        CH     1961        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1962        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1963        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1964        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1965        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.2 NSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1966        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.3 C--                         H   OCH.sub.3                                  OCH.sub.3                                        CH                OCO     1967        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.3 C--                         H   OCH.sub.3                                  CH.sub.3                                        CH                OCO     1968        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.3 C--                         H   CH.sub.3                                  CH.sub.3                                        CH                OCO     1969        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.3 C--                         H   Cl   OCH.sub.3                                        CH                OCO     1970        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.3 C--                         H   OCH.sub.3                                  OCH.sub.3                                        N                OCO     1971        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.3 C--                         H   OCH.sub.3                                  CH.sub.3                                        N                OCO     1972        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.3 C--                         H   OCH.sub.3                                  CF.sub.3                                        N                OCO     1973        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.3 C--                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH                OCO     1974        C.sub.2 H.sub.5             CH.sub.3                (CH.sub.3).sub.3 C--                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N                OCO     1975        C.sub.2 H.sub.5             CH.sub.3                PhCO     H   OCH.sub.3                                  OCH.sub.3                                        CH     1976        C.sub.2 H.sub.5             CH.sub.3                PhCO     H   OCH.sub.3                                  CH.sub.3                                        CH     1977        C.sub.2 H.sub.5             CH.sub.3                PhCO     H   CH.sub.3                                  CH.sub.3                                        CH     1978        C.sub.2 H.sub.5             CH.sub.3                PhCO     H   Cl   OCH.sub.3                                        CH     1979        C.sub.2 H.sub.5             CH.sub.3                PhCO     H   OCH.sub.3                                  OCH.sub.3                                        N     1980        C.sub.2 H.sub.5             CH.sub.3                PhCO     H   OCH.sub.3                                  CH.sub.3                                        N     1981        C.sub.2 H.sub.5             CH.sub.3                PhCO     H   OCH.sub.3                                  CF.sub.3                                        N     1982        C.sub.2 H.sub.5             CH.sub.3                PhCO     CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     1983        C.sub.2 H.sub.5             CH.sub.3                PhCO     CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     1984        C.sub.2 H.sub.5             CH.sub.3                PhSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1985        C.sub.2 H.sub.5             CH.sub.3                PhSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        CH     1986        C.sub.2 H.sub.5             CH.sub.3                PhSO.sub.2                         H   CH.sub.3                                  CH.sub.3                                        CH     1987        C.sub.2 H.sub.5             CH.sub.3                PhSO.sub.2                         H   Cl   OCH.sub.3                                        CH     1988        C.sub.2 H.sub.5             CH.sub.3                PhSO.sub.2                         H   OCH.sub.3                                  CH.sub.3                                        N     1989        C.sub.2 H.sub.5             CH.sub.3                PhSO.sub.2                         H   OCH.sub.3                                  CF.sub.3                                        N     1990        C.sub.2 H.sub.5             CH.sub.3                PhSO.sub.2                         H   OCH.sub.3                                  OCH.sub.3                                        N     1991        C.sub.2 H.sub.5             CH.sub.3                PhSO.sub.2                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        CH     1992        C.sub.2 H.sub.5             CH.sub.3                PhSO.sub.2                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        N     1993        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     1994        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     1995        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCO                         H   CH.sub.3                                  CH.sub.3                                        CH     1996        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCO                         H   Cl   OCH.sub.3                                        CH     1997        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     1998        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCO                         H   OCH.sub.3                                  CH.sub.3                                        N     1999        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCO                         H   OCH.sub.3                                  CF.sub.3                                        N     2000        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2001        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2002        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2003        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     2004        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCO                         H   CH.sub.3                                  CH.sub.3                                        CH     2005        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCO                         H   Cl   OCH.sub.3                                        CH     2006        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     2007        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCO                         H   OCH.sub.3                                  CH.sub.3                                        N     2008        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCO                         H   OCH.sub.3                                  CF.sub.3                                        N     2009        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2010        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2011        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCS                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2012        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCS                         H   OCH.sub.3                                  CH.sub.3                                        CH     2013        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCS                         H   CH.sub.3                                  CH.sub.3                                        CH     2014        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCS                         H   Cl   OCH.sub.3                                        CH     2015        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCS                         H   OCH.sub.3                                  OCH.sub.3                                        N     2016        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCS                         H   OCH.sub.3                                  CH.sub.3                                        N     2017        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCS                         H   OCH.sub.3                                  CF.sub.3                                        N     2018        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCS                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2019        C.sub.2 H.sub.5             CH.sub.3                CH.sub.3 NHCS                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2020        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCS                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2021        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCS                         H   OCH.sub.3                                  CH.sub.3                                        CH     2022        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCS                         H   CH.sub.3                                  CH.sub.3                                        CH     2023        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCS                         H   Cl   OCH.sub.3                                        CH     2024        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCS                         H   OCH.sub.3                                  OCH.sub.3                                        N     2025        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCS                         H   OCH.sub.3                                  CH.sub.3                                        N     2026        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCS                         H   OCH.sub.3                                  CF.sub.3                                        N     2027        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCS                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2028        C.sub.2 H.sub.5             CH.sub.3                C.sub.2 H.sub.5 NHCS                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2029        C.sub.2 H.sub.5             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2030        C.sub.2 H.sub.5             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     2031        C.sub.2 H.sub.5             CH.sub.3                COSCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     2032        C.sub.2 H.sub.5             CH.sub.3                COSCH.sub.3                         H   Cl   OCH.sub.3                                        CH     2033        C.sub.2 H.sub.5             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     2034        C.sub.2 H.sub.5             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2035        C.sub.2 H.sub.5             CH.sub.3                COSCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     2036        C.sub.2 H.sub.5             CH.sub.3                COSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CN     2037        C.sub.2 H.sub.5             CH.sub.3                COSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2038        C.sub.2 H.sub.5             CH.sub.3                CSOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2039        C.sub.2 H.sub.5             CH.sub.3                CSOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     2040        C.sub.2 H.sub.5             CH.sub.3                CSOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     2041        C.sub.2 H.sub.5             CH.sub.3                CSOCH.sub.3                         H   Cl   OCH.sub.3                                        CH     2042        C.sub.2 H.sub.5             CH.sub.3                CSOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     2043        C.sub.2 H.sub.5             CH.sub.3                CSOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2044        C.sub.2 H.sub.5             CH.sub.3                CSOCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     2045        C.sub.2 H.sub.5             CH.sub.3                CSOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2046        C.sub.2 H.sub.5             CH.sub.3                CSOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2047        C.sub.2 H.sub.5             CH.sub.3                CSSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2048        C.sub.2 H.sub.5             CH.sub.3                CSSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     2049        C.sub.2 H.sub.5             CH.sub.3                CSSCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     2050        C.sub.2 H.sub.5             CH.sub.3                CSSCH.sub.3                         H   Cl   OCH.sub.3                                        CH     2051        C.sub.2 H.sub.5             CH.sub.3                CSSCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     2052        C.sub.2 H.sub.5             CH.sub.3                CSSCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2053        C.sub.2 H.sub.5             CH.sub.3                CSSCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     2054        C.sub.2 H.sub.5             CH.sub.3                CSSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2055        C.sub.2 H.sub.5             CH.sub.3                CSSCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2056        C.sub.2 H.sub.5             CH.sub.3                COCOOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2057        C.sub.2 H.sub.5             CH.sub.3                COCOOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     2058        C.sub.2 H.sub.5             CH.sub.3                COCOOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     2059        C.sub.2 H.sub.5             CH.sub.3                COCOOCH.sub.3                         H   Cl   OCH.sub.3                                        CH     2060        C.sub.2 H.sub.5             CH.sub.3                COCOOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     2061        C.sub.2 H.sub.5             CH.sub.3                COCOOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2062        C.sub.2 H.sub.5             CH.sub.3                COCOOCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     2063        C.sub.2 H.sub.5             CH.sub.3                COCOOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2064        C.sub.2 H.sub.5             CH.sub.3                COCOOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2065        C.sub.2 H.sub.5             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2066        C.sub.2 H.sub.5             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  CH.sub.3                                        CH     2067        C.sub.2 H.sub.5             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   CH.sub.3                                  CH.sub.3                                        CH     2068        C.sub.2 H.sub.5             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   Cl   OCH.sub.3                                        CH     2069        C.sub.2 H.sub.5             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  OCH.sub.3                                        N     2070        C.sub.2 H.sub.5             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  CH.sub.3                                        N     2071        C.sub.2 H.sub.5             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         H   OCH.sub.3                                  CF.sub.3                                        N     2072        C.sub.2 H.sub.5             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2073        C.sub.2 H.sub.5             CH.sub.3                i-C.sub.3 H.sub.7 OCO                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2074        C.sub.2 H.sub.5             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  OCH.sub.3                                        CH 161-165     2075        C.sub.2 H.sub.5             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  CH.sub.3                                        CH     2076        C.sub.2 H.sub.5             C.sub.2 H.sub.5                CHO      H   CH.sub.3                                  CH.sub.3                                        CH     2077        C.sub.2 H.sub.5             C.sub.2 H.sub.5                CHO      H   Cl   OCH.sub.3                                        CH     2078        C.sub.2 H.sub.5             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  CH.sub.3                                        N     2079        C.sub.2 H.sub.5             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  CF.sub.3                                        N     2080        C.sub.2 H.sub.5             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  OCH.sub.3                                        N     2081        C.sub.2 H.sub.5             C.sub.2 H.sub.5                CHO      CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2082        C.sub.2 H.sub.5             C.sub.2 H.sub.5                CHO      CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2083        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 173-179     2084        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     2085        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     2086        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCH.sub.3                         H   Cl   OCH.sub.3                                        CH     2087        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2088        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     2089        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     2090        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        CH     2091        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        N     2092        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 158-160     2093        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     2094        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOCH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     2095        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOCH.sub.3                         H   Cl   OCH.sub.3                                        CH     2096        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2097        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     2098        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     2099        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2100        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOCH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2101        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2102        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     2103        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     2104        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     2105        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2106        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     2107        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     2108        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2109        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2110        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 98-101     2111        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     2112        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     2113        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   Cl   OCH.sub.3                                        CH     2114        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2115        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     2116        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     2117        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2118        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2119        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2120        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        CH     2121        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   CH.sub.3                                  CH.sub.3                                        CH     2122        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   Cl   OCH.sub.3                                        CH     2123        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2124        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CF.sub.3                                        N     2125        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        N     2126        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2127        C.sub.2 H.sub.5             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2128        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 143-146     2129        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        CH     2130        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCF.sub.3                         H   CH.sub.3                                  CH.sub.3                                        CH     2131        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCF.sub.3                         H   Cl   OCH.sub.3                                        CH     2132        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2133        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCF.sub.3                         H   OCH.sub.3                                  CF.sub.3                                        N     2134        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        N     2135        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCF.sub.3                         CH.sub.3                             OCH.sub.3                                  OCH.sub.3                                        CH     2136        C.sub.2 H.sub.5             C.sub.2 H.sub.5                COCF.sub.3                         CH.sub.3                             OCH.sub.3                                  CH.sub.3                                        N     2137        nC.sub.3 H.sub.7             H  CHO      H   OCH.sub.3                                  OCH.sub.3                                        CH 148-154     2138        nC.sub.3 H.sub.7             H  CHO      H   OCH.sub.3                                  CH.sub.3                                        N     2139        nC.sub.3 H.sub.7             H  COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 106-110     2140        nC.sub.3 H.sub.7             H  COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2141        nC.sub.3 H.sub.7             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2142        nC.sub.3 H.sub.7             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2143        nC.sub.3 H.sub.7             H  COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 194-197     2144        nC.sub.3 H.sub.7             H  COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2145        nC.sub.3 H.sub.7             H  COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 142-147     2146        nC.sub.3 H.sub.7             H  COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2147        nC.sub.3 H.sub.7             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2148        nC.sub.3 H.sub.7             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2149        nC.sub.3 H.sub.7             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 199-205     2150        nC.sub.3 H.sub.7             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2151        nC.sub.3 H.sub.7             H  SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH 128-133     2152        nC.sub.3 H.sub.7             H  SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2153        nC.sub.3 H.sub.7             CH.sub.3                CHO      H   OCH.sub.3                                  OCH.sub.3                                        CH 139-145     2154        nC.sub.3 H.sub.7             CH.sub.3                CHO      H   OCH.sub.3                                  CH.sub.3                                        N     2155        nC.sub.3 H.sub.7             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 138-141     2156        nC.sub.3 H.sub.7             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2157        nC.sub.3 H.sub.7             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2158        nC.sub.3 H.sub.7             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2159        nC.sub.3 H.sub.7             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 172-175     2160        nC.sub.3 H.sub.7             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2161        nC.sub.3 H.sub.7             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 182-185     2162        nC.sub.3 H.sub.7             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2163        nC.sub.3 H.sub.7             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2164        nC.sub.3 H.sub.7             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2165        nC.sub.3 H.sub.7             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 168-176     2166        nC.sub.3 H.sub.7             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2167        nC.sub.3 H.sub.7             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH 129-132     2168        nC.sub.3 H.sub.7             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2169        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  OCH.sub.3                                        CH 142-145     2170        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  CH.sub.3                                        N     2171        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2172        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2173        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2174        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2175        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2176        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2177        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 173-177     2178        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2179        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2180        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2181        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 173-179     2182        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2183        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2184        nC.sub.3 H.sub.7             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2185        N(CH.sub.3).sub.2             H  CHO      H   OCH.sub.3                                  OCH.sub.3                                        CH 143-144     2186        N(CH.sub.3).sub.2             H  CHO      H   OCH.sub.3                                  CH.sub.3                                        N     2187        N(CH.sub.3).sub.2             H  COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2188        N(CH.sub.3).sub.2             H  COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2189        N(CH.sub.3).sub.2             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2190        N(CH.sub.3).sub.2             H  COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2191        N(CH.sub.3).sub.2             H  COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2192        N(CH.sub.3).sub.2             H  COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2193        N(CH.sub.3).sub.2             H  COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2194        N(CH.sub.3).sub.2             H  COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2195        N(CH.sub.3).sub.2             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2196        N(CH.sub.3).sub.2             H  COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2197        N(CH.sub.3).sub.2             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2198        N(CH.sub.3).sub.2             H  SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2199        N(CH.sub.3).sub.2             H  SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2200        N(CH.sub.3).sub.2             H  SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2201        N(CH.sub.3).sub.2             CH.sub.3                CHO      H   OCH.sub.3                                  OCH.sub.3                                        CH 201-203     2202        N(CH.sub.3).sub.2             CH.sub.3                CHO      H   OCH.sub.3                                  CH.sub.3                                        N     2203        N(CH.sub.3).sub.2             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 176-179     2204        N(CH.sub.3).sub.2             CH.sub.3                COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2205        N(CH.sub.3).sub.2             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2206        N(CH.sub.3).sub.2             CH.sub.3                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2207        N(CH.sub.3).sub.2             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2208        N(CH.sub.3).sub.2             CH.sub.3                COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2209        N(CH.sub.3).sub.2             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 192-194     2210        N(CH.sub.3).sub.2             CH.sub.3                COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2211        N(CH.sub.3).sub.2             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2212        N(CH.sub.3).sub.2             CH.sub.3                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2213        N(CH.sub.3).sub.2             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 144-146     2214        N(CH.sub.3).sub.2             CH.sub.3                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2215        N(CH.sub.3).sub.2             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2216        N(CH.sub.3).sub.2             CH.sub.3                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2217        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  OCH.sub.3                                        CH 143-146     2218        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                CHO      H   OCH.sub.3                                  CH.sub.3                                        N     2219        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 116-118     2220        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                COCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2221        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2222        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                COC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2223        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                COCF.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2224        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                COCF.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2225        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 201-203     2226        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                COOCH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2227        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2228        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                COOC.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     2229        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  OCH.sub.3                                        CH 125-128     2230        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                SO.sub.2 CH.sub.3                         H   OCH.sub.3                                  CH.sub.3                                        N     2231        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  OCH.sub.3                                        CH     2232        N(CH.sub.3).sub.2             C.sub.2 H.sub.5                SO.sub.2 C.sub.2 H.sub.5                         H   OCH.sub.3                                  CH.sub.3                                        N     __________________________________________________________________________

                  TABLE 2     ______________________________________     Compounds of the formula (Ib)                                   (Ib)     1 #STR250##     No.  R.sup.1                 R.sup.4                        R.sup.5 X     Y     Z    mp.(° C.)     ______________________________________     2-1  CH.sub.3                 H      CHO     OCH.sub.3                                      OCH.sub.3                                            CH     2-2  CH.sub.3                 H      CHO     OCH.sub.3                                      CH.sub.3                                            N     2-3  CH.sub.3                 H      COOCH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     2-4  CH.sub.3                 H      COOCH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     2-5  CH.sub.3                 H      SO.sub.2 CH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     2-6  CH.sub.3                 H      SO.sub.2 CH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     2-7  CH.sub.3                 CH.sub.3                        CHO     OCH.sub.3                                      OCH.sub.3                                            CH     2-8  CH.sub.3                 CH.sub.3                        CHO     OCH.sub.3                                      CH.sub.3                                            N     2-9  CH.sub.3                 CH.sub.3                        COOCH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     2-10 CH.sub.3                 CH.sub.3                        COOCH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     2-11 CH.sub.3                 CH.sub.3                        SO.sub.2 CH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     2-12 CH.sub.3                 CH.sub.3                        SO.sub.2 CH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     2-13 C.sub.2 H.sub.5                 H      CHO     OCH.sub.3                                      OCH.sub.3                                            CH     2-14 C.sub.2 H.sub.5                 H      CHO     OCH.sub.3                                      CH.sub.3                                            N     2-15 C.sub.2 H.sub.5                 H      COOCH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     2-16 C.sub.2 H.sub.5                 H      COOCH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     2-17 C.sub.2 H.sub.5                 H      SO.sub.2 CH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     2-18 C.sub.2 H.sub.5                 H      SO.sub.2 CH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     2-19 C.sub.2 H.sub.5                 CH.sub.3                        CHO     OCH.sub.3                                      OCH.sub.3                                            CH     2-20 C.sub.2 H.sub.5                 CH.sub.3                        CHO     OCH.sub.3                                      CH.sub.3                                            N     2-21 C.sub.2 H.sub.5                 CH.sub.3                        COOCH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     2-22 C.sub.2 H.sub.5                 CH.sub.3                        COOCH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     2-23 C.sub.2 H.sub.5                 CH.sub.3                        SO.sub.2 CH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     2-24 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        SO.sub.2 CH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     2-25 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        CHO     OCH.sub.3                                      CH.sub.3                                            N     2-26 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        CHO     OCH.sub.3                                      CH.sub.3                                            N     2-27 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        COOCH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     2-28 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        COOCH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     2-29 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        SO.sub.2 CH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     2-30 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        SO.sub.2 CH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     ______________________________________

                  TABLE 3     ______________________________________     Compounds of the formula (Ic)                                   (Ic)     2 #STR251##     No.  R.sup.1                 R.sup.4                        R.sup.5 X     Y     Z    mp.(° C.)     ______________________________________     3-1  CH.sub.3                 H      CHO     OCH.sub.3                                      OCH.sub.3                                            CH     3-2  CH.sub.3                 H      CHO     OCH.sub.3                                      CH.sub.3                                            N     3-3  CH.sub.3                 H      COOCH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     3-4  CH.sub.3                 H      COOCH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     3-5  CH.sub.3                 H      SO.sub.2 CH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     3-6  CH.sub.3                 H      SO.sub.2 CH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     3-7  CH.sub.3                 CH.sub.3                        CHO     OCH.sub.3                                      OCH.sub.3                                            CH     3-8  CH.sub.3                 CH.sub.3                        CHO     OCH.sub.3                                      CH.sub.3                                            N     3-9  CH.sub.3                 CH.sub.3                        COOCH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     3-10 CH.sub.3                 CH.sub.3                        COOCH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     3-11 CH.sub.3                 CH.sub.3                        SO.sub.2 CH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     3-12 CH.sub.3                 CH.sub.3                        SO.sub.2 CH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     3-13 C.sub.2 H.sub.5                 H      CHO     OCH.sub.3                                      OCH.sub.3                                            CH   118-120     3-14 C.sub.2 H.sub.5                 H      CHO     OCH.sub.3                                      CH.sub.3                                            N     3-15 C.sub.2 H.sub.5                 H      COOCH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     3-16 C.sub.2 H.sub.5                 H      COOCH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     3-17 C.sub.2 H.sub.5                 H      SO.sub.2 CH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH     3-18 C.sub.2 H.sub.5                 H      SO.sub.2 CH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     3-19 C.sub.2 H.sub.5                 CH.sub.3                        CHO     OCH.sub.3                                      OCH.sub.3                                            CH   138-140     3-20 C.sub.2 H.sub.5                 CH.sub.3                        CHO     OCH.sub.3                                      CH.sub.3                                            N     3-21 C.sub.2 H.sub.5                 CH.sub.3                        COOCH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH   116-117     3-22 C.sub.2 H.sub.5                 CH.sub.3                        COOCH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     3-23 C.sub.2 H.sub.5                 CH.sub.3                        SO.sub.2 CH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH   179-180     3-24 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        SO.sub.2 CH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     3-25 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        CHO     OCH.sub.3                                      OCH.sub.3                                            CH   173-174     3-26 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        CHO     OCH.sub.3                                      CH.sub.3                                            N     3-27 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        COOCH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH   130-131     3-28 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        COOCH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     3-29 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        SO.sub.2 CH.sub.3                                OCH.sub.3                                      OCH.sub.3                                            CH   130-131     3-30 C.sub.2 H.sub.5                 C.sub.2 H.sub.5                        SO.sub.2 CH.sub.3                                OCH.sub.3                                      CH.sub.3                                            N     ______________________________________

                                      TABLE 4     __________________________________________________________________________     Na.sup.+  salts     Compounds of the formula (Id)                                 (Id)     3 #STR252##     No.        n  R.sup.1                R.sup.4                   R.sup.5                         X   Y   Z  mp.(° C.)     __________________________________________________________________________     4-1        2  CH.sub.3                H  CHO   OCH.sub.3                             OCH.sub.3                                 CH 204-209     4-2        2  CH.sub.3                H  COCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 190-193     4-3        2  CH.sub.3                H  COC.sub..sub.2 H.sub.5                         OCH.sub.3                             OCH.sub.3                                 CH 125-135     4-4        2  CH.sub.3                H  CO-i-C.sub.3 H.sub.7                         OCH.sub.3                             OCH.sub.3                                 CH 198-201     4-5        2  CH.sub.3                H  COCCl.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 256-260     4-6        2  CH.sub.3                H  COOC.sub.2 H.sub.5                         OCH.sub.3                             OCH.sub.3                                 CH 189-193     4-7        2  CH.sub.3                H  SO.sub.2 CH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 188-192     4-8        2  CH.sub.3                H  SO.sub.2 C.sub.2 H.sub.5                         OCH.sub.3                             OCH.sub.3                                 CH 194-198     4-9        2  CH.sub.3                H  CHO   OCH.sub.3                             OCH.sub.3                                 CH 178-182     4-10        2  CH.sub.3                CH.sub.3                   COCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 181-190     4-11        2  CH.sub.3                CH.sub.3                   COC.sub.2 H.sub.5                         OCH.sub.3                             OCH.sub.3                                 CH 187-195     4-12        2  CH.sub.3                CH.sub.3                   COCF.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 189-198     4-13        2  CH.sub.3                CH.sub.3                   COCCl.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 181-188     4-14        2  CH.sub.3                CH.sub.3                   CO-i-C.sub.3 H.sub.7                         OCH.sub.3                             OCH.sub.3                                 CH 175-180     4-15        2  CH.sub.3                CH.sub.3                   COOCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 142-150     4-16        2  CH.sub.3                CH.sub.3                   COOC.sub.2 H.sub.5                         OCH.sub.3                             OCH.sub.3                                 CH 138-145     4-17        2  CH.sub.3                CH.sub.3                   SO.sub.2 CH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 191-194     4-18        2  CH.sub.3                CH.sub.3                   SO.sub.2 C.sub.2 H.sub.5                         OCH.sub.3                             OCH.sub.3                                 CH 187-191     4-19        2  C.sub.2 H.sub.5                H  CHO   OCH.sub.3                             OCH.sub.3                                 CH 191-198     4-20        2  C.sub.2 H.sub.5                H  COCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 172-180     4-21        2  C.sub.2 H.sub.5                H  COOCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 184-189     4-22        2  C.sub.2 H.sub.5                H  SO.sub.2 CH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 172-180     4-23        2  C.sub.2 H.sub.5                CH.sub.3                   CHO   OCH.sub.3                             OCH.sub.3                                 CH 182-185     4-24        2  C.sub.2 H.sub.5                CH.sub.3                   COCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 184-187     4-25        2  C.sub.2 H.sub.5                CH.sub.3                   SO.sub.2 CH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 228-229     4-26        2  C.sub.2 H.sub.5                C.sub.2 H.sub.5                   CHO   OCH.sub.3                             OCH.sub.3                                 CH 184-189     4-27        2  C.sub.2 H.sub.5                C.sub.2 H.sub.5                   COCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 173-179     4-28        2  C.sub.2 H.sub.5                C.sub.2 H.sub.5                   COCF.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 182-186     4-29        2  C.sub.2 H.sub.5                C.sub.2 H.sub.5                   COOCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 155-162     4-30        2  C.sub.2 H.sub.5                C.sub.2 H.sub.5                   SO.sub.2 CH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 225-227     4-31        2  nC.sub.3 H.sub.7                H  CHO   OCH.sub.3                             OCH.sub.3                                 CH 177-183     4-32        2  nC.sub.3 H.sub.7                H  COCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 178-182     4-33        2  nC.sub.3 H.sub.7                H  COCF.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 240-246     4-34        2  nC.sub.3 H.sub.7                H  COOCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 192-200     4-35        2  nC.sub.3 H.sub.7                H  SO.sub.2 Cl.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 247-250     4-36        2  nC.sub.3 H.sub.7                H  SO.sub.2 C.sub.2 H.sub.5                         OCH.sub.3                             OCH.sub.3                                 CH 183-187     4-37        2  nC.sub.3 H.sub.7                CH.sub.3                   CHO   OCH.sub.3                             OCH.sub.3                                 CH 194-202     4-38        2  nC.sub.3 H.sub.7                CH.sub.3                   COCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 175-178     4-39        2  nC.sub.3 H.sub.7                CH.sub.3                   COCF.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 155-161     4-40        2  nC.sub.3 H.sub.7                CH.sub.3                   COOCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 213-216     4-41        2  nC.sub.3 H.sub.7                CH.sub.3                   SO.sub.2 CH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 213-216     4-42        2  nC.sub.3 H.sub.7                CH.sub.3                   SO.sub.2 C.sub.2 H.sub.5                         OCH.sub.3                             OCH.sub.3                                 CH 168-174     4-43        2  nC.sub.3 H.sub.7                C.sub.2 H.sub.5                   CHO   OCH.sub.3                             OCH.sub.3                                 CH 170-176     4-44        2  nC.sub.3 H.sub.7                C.sub.2 H.sub.5                   COOCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 150-155     4-45        2  nC.sub.3 H.sub.7                C.sub.2 H.sub.5                   SO.sub.2 CH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 167-173     4-46        2  N(CH.sub.3).sub.2                H  CHO   OCH.sub.3                             OCH.sub.3                                 CH 188-192     4-47        2  N(CH.sub.3).sub.2                H  SO.sub.2 CH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 192-197     4-48        2  N(CH.sub.3).sub.2                CH.sub.3                   CHO   OCH.sub.3                             OCH.sub.3                                 CH 180-184     4-49        2  N(CH.sub.3).sub.2                CH.sub.3                   COCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 140-145     4-50        2  N(CH.sub.3).sub.2                CH.sub.3                   COOCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 116     4-51        2  N(CH.sub.3).sub.2                CH.sub.3                   SO.sub.2 CH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 172-180     4-52        2  N(CH.sub.3).sub.2                C.sub.2 H.sub.5                   CHO   OCH.sub.3                             OCH.sub.3                                 CH 167-171     4-53        2  N(CH.sub.3).sub.2                C.sub.2 H.sub.5                   COCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 128-133     4-54        2  N(CH.sub.3).sub.2                C.sub.2 H.sub.5                   COOCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 163-168     4-55        2  N(CH.sub.3).sub.2                C.sub.2 H.sub.5                   SO.sub.2 CH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 178-182     4-56        1  C.sub.2 H.sub.5                H  CHO   OCH.sub.3                             OCH.sub.3                                 CH 197-199     4-57        1  C.sub.2 H.sub.5                CH.sub.3                   CHO   OCH.sub.3                             OCH.sub.3                                 CH 112-115     4-58        1  C.sub.2 H.sub.5                CH.sub.3                   COOCH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 160-164     4-59        1  C.sub.2 H.sub.5                CH.sub.3                   SO.sub.2 CH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 180-183     4-60        1  C.sub.2 H.sub.5                C.sub.2 H.sub.5                   CHO   OCH.sub.3                             OCH.sub.3                                 CH 166-172     4-61        1  C.sub.2 H.sub.5                C.sub.2 H.sub.5                   SO.sub.2 CH.sub.3                         OCH.sub.3                             OCH.sub.3                                 CH 221-222     __________________________________________________________________________

B. Formulation examples

a) A dust is obtained by mixing 10 parts by weight of a compound of the formula (I) and 90 parts by weight of talc as inert substance and comminuting the mixture in a hammer mill.

b) A wettable power which is readily dispersible in water is obtained by mixing 25 parts by weight of a compound of the formula (I), 64 parts by weight of kaolin-containing quartz as inert substance, 10 parts by weight of potassium lignosulfonate and 1 part by weight of sodium oleoylmethyltaurate as wetting agent and dispersant, and grinding the mixture in a pinned-disk mill.

c) A dispersion concentrate which is readily dispersible in water is obtained by mixing 20 parts by weight of a compound of the formula (I) with 6 parts by weight of akylphenyl polyglycol ether (®Triton X207), 3 parts by weight of isotridecanol polyglycol ether (8 EO) and 71 parts by weight of paraffinic mineral oil (boiling range for example approx. 255 to above 277° C.), and grinding the mixture in a ball mill to a fineness of below 5 microns.

d) An emulsifiable concentrate is obtained from 15 parts by weight of a compound of the formula (I), 75 parts by weight of cyclohexanone as solvent and 10 parts by weight of oxethylated nonylphenol as emulsifier.

e) Granules which are dispersible in water are obtained by mixing

75 parts by weight of a compound of the formula (I),

10 " of calcium lignosulfonate,

5 " of sodium lauryl sulfate,

3 " of polyvinyl alcohol and

7 " of kaolin,

grinding the mixture on a pinned-disk mill and granulating the powder in a fluidized bed by spraying on water as granulation liquid.

f) Water-dispersible granules are also obtained by homogenizing, on a colloid

25 parts by weight of a compound of the formula (I),

5 " of sodium 2,2'-dinaphthylmethane,6,6'-disulfonate,

2 " of sodium oleoylmethyltaurate,

1 part by weight of polyvinyl alcohol,

17 parts by weight of calcium carbonate and

50 " of water,

precomminuting the mixture, subsequently grinding it on a bead mill and atomizing and drying the resulting suspension in a spray tower by means of a single-substance nozzle.

C. Biological examples

1. Pre-emergence effect on weeds

Seeds or rhizome pieces of monocotyledonous and dicotyledonous weed plants are placed in sandy loam soil in plastic pots and covered with soil. The compounds of the formula (I) or salts thereof according to the invention which have been formulated in the form of wettable powders or emulsion concentrates are then applied to the surface of the soil cover in the form of aqueous suspensions or emulsions at an application rate of 600 to 800 l of water/ha (converted), in various dosages.

After the treatment, the pots are placed in a greenhouse and kept under good growth conditions for the weeds. After the test plants have emerged after a period of 3 to 4 weeks, the damage to the plants or the negative effect on the emergence i5 scored visually by comparison with untreated controls. As shown by the test results, the compounds according to the invention have a good herbicidal pre-emergence activity against a broad spectrum of grass weeds and broad-leaved weeds. For example, the compounds of Examples Nos. 1, 18, 35, 69, 86, 103, 120, 138, 155, 225, 531, 548, 565, 599, 616, 633, 650, 667, 684, 753, 1068, 1085, 1170, 1202, 1591, 1608, 1676, 1727, 2074, 2068, 2092, 2110, 2128, 2137, 2139,2144, 2145, 2149, 2151, 2153, 2155, 2159, 2161, 2165, 2167, 2169, 2177, 2181, 2185, 2201, 2203, 2209, 2213, 2217, 2219, 2225, 2229, 3-13, 3-19, 3-21, 3-23, 3-25, 3-27, 3-29 (see Section A) and their sodium salts show a very good herbicidal activity in the test against harmful plants such as Sinapis alba, Stellaria media, Chrysanthemum segetum, and Lolium multiflorum when applied pre-emergence at a rate of application of 0.3 kg to 0.005 kg of active ingredient per hectare.

2. Post-emergence effect on weeds

Seeds or rhizome pieces of monocotyledonous and diotyledonous weeds are placed in sandy loam soil in plastic pots, covered with soil and grown in a greenhouse under good growth conditions. Three weeks after sowing, the test plants are treated in the three-leaf stage. The compounds of the formula (I) or salts thereof according to the invention which have been formulated as wettable powders or as emulsion concentrates are sprayed in various dosages onto the green parts of the plants at an application rate of 600 to 800 l of water/ha (converted). After the test plants have remained in the greenhouse for about 3 to 4 weeks under ideal growth conditions, the effect of the preparations is scored visually by comparison with untreated controls. The agents according to the invention also have a good herbicidal post-emergence activity against a broad range of economically important grass weeds and broad-leaved weeds. For example, Examples Nos. 1, 18, 35, 69, 86, 103, 120, 138, 155, 225, 531, 548, 565, 599, 616, 633, 650, 667, 684, 753, 1068, 1085, 1170, 1202, 1591, 1608, 1676, 1727, 2074, 2068, 2092, 2110, 2128, 2137, 2139, 2144, 2145, 2149, 2151, 2153, 2155, 2159, 2161, 2165, 2167, 2169, 2177, 2181, 2185, 2201, 2203, 2209, 2213, 2217, 2219, 2225, 2229, 3-13, 3-19, 3-21, 3-23, 3-25, 3-27, 3-29 (see Section A) and their sodium salts show a very good herbicidal activity in the test against harmful plants such as Sinapis alba, Stellaria media, Chrysanthemum segetum, and Lolium murlifflorum when applied post-emergence at an application rate of 0.3 kg to 0.005 kg of active ingredient per hectare.

3. Tolerance by crop plants

In further greenhouse experiments, seeds of a substantial number of crop plants and weeds were placed in sandy loam substrate and covered with soil.

Some of the pots were treated immediately as described in Section 1, and the remaining pots were placed in a greenhouse until the plants had developed two to three true leaves and then sprayed with various dosages of the substances of the formula (I) or salts thereof according to the invention as described in Section 2.

Visual scoring four to five weeks after application and after the plants had remained in the greenhouse revealed that the compounds according to the invention did not inflict any damage to dicotyledonous crops such as soy beans, cotton, oil seed rape, sugar beet and potatoes when used pre- and post-emergence, even when high dosages of active substance were used. Moreover, some substances also left Gramineae crops such as barley, wheat, rye, Sorghum species, maize or rice unharmed. The compounds of the formula (I) or their salts therefore have a high selectivity when used for controlling undesirable vegetation in agricultural crops. 

We claim:
 1. A compound of the formula (I) or a salt thereof ##STR253## where R¹ is NR⁸ R⁹ or an unsubstituted or substituted hydrocarbon radical,n is 0, 1 or 2, excluding n=0 or 1 if R¹ =NR⁸ R⁹, R² and R³ are each independently of the other H or (1-4)alkyl, R⁴ is H, OH, formyl, or a radical of the formula R, R--O--, R--CO-- or R--SO₂ --, R being an unsubstituted or substituted hydrocarbon radical, R⁵ is an acyl radical or NR⁴ R⁵ together are an unsubstituted or substituted heterocyclic radical, W is an oxygen or sulfur atom, R⁶ is H, (1-4)alkyl, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkyl!-carbonyl, or (1-4)alkoxy!carbonyl, each of the last radicals being unsubstituted or substituted by one or more halogen atoms, or halogen, NO₂, CN or mono- or disubstituted amino, R⁷ is H or (1-4)alkyl, R⁸ and R⁹ are each independently of the other H, (1-4)alkyl, (1-4)alkoxy, (1-4)alkyl!carbonyl or (1-4)alkylsulfonyl, A is a radical of the formula ##STR254## one of the radicals X and Y being hydrogen, (1-3)alkyl or (1-3)alkoxy, the last two radicals being unsubstituted or mono- or polysubstituted by halogen or monosubstituted by (1-3)alkoxy, and the other of the radicals X and Y being hydrogen, halogen, (1-3)alkyl, (1-3)alkoxy or (1-3)alkyithio, the last three alkyl-containing radicals being unsubstituted or mono- or polysubstituted by halogen or mono- or disubstituted by (1-3)alkoxy or (1-3)alkylthio, or a radical of the formula NR^(a) R^(b), where R^(a) and R^(b), independently of each other, are H, (1-3)alkyl or (1-3)alkenyl, or (3-6)cycloalkyl, (2-4)alkenyl, (2-4)alkynyl, (3-4)-alkenyloxy or (3-4)alkynyloxy, Z is CH or N, X¹ is CH₃, OCH₃, OC₂ H₅ or OCHF₂, Y¹ is --O-- or --CH₂ --, X² is CH₃, C₂ H₅ or CH₂ CF₃, Y² is OCH₃, OC₂ H₅, SCH₃, SCH₂ CH₃, CH₃ or C₂ H₅, X³ is CH₃ or OCH₃, Y³ is H or CH₃, X⁴ is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃ or Cl, Y⁴ is CH₃, OCH₃, OC₂ H₅ or Cl and Y⁵ is CH₃, C₂ H₅, OCH₃ or Cl.
 2. A compound or a salt thereof as claimed in claim 1, whereinR¹ is NR⁸ R⁹, (1-6)alkyl, (2-6)alkenyl, (2-6)alkynyl, (3-6)cycloalkyl, (3-6)cycloalkenyl or phenyl, each of the last 6 radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, CN, (1-4)alkoxy, (1-4)haloalkoxy, (1-4)alkoxy(1-4)alkoxy, (1-4)alkylthio, (1-4)alkylsulfinyl, (1-4)-alkylsulfony, formyl, (1-4)alkyl!-carbonyl, (1-4)alkoxy!carbonyl, (1-4)alkyl!carbonyloxy and in the case of cyclic radicals also (1-4)alkyl, (1-4)haloalkyl and (1-4)alkoxy-(1-4)alkyl, n is 0, 1 or 2, excluding n=0 or 1 if R¹ =NR⁸ R⁹, R² and R³ are each independently of the other H or (1-4)alkyl, R⁴ is H, OH, formyl, (1-6)alkyl, (2-6)alkenyl, (2-6)alkynyl, (1-6)alkoxy, (2-5)alkenyloxy, (2-5)alkynyloxy, (1-6)alkyl!-carbonyl, (1-6)alkylsulfonyl, (2-6)alkenyl!carbonyl, (2-6)alkenylsulfonyl, (2-6)alkynyl!carbonyl, (2-6)-alkynyl-sulfonyl, (3-6)cycloalkyl, (3-6)cycloalkenyl, (3-6)cycloalkyl!-carbonyl, (3-6)cycloalkylsulfonyl, (3-6)cycloalkenyl!carbonyl or (3-6)cycloalkenylsulfonyl, each of the last 18 radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkylsulfinyl, (1-4)alkylsulfonyl, (1-4)alkoxy!carbonyl, (1-4)alkyl!carbonyl, (1-4)alkyl!carbonyloxy and CN and in the case of cyclic radicals also (1-4)alkyl and (1-4)haloalkyl, or phenylcarbonyl or phenylsulfonyl, the phenyl ring in the last two radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, CN, NO₂, (1-4)alkyl, (1-4)haloalkyl, (1-4)alkoxy and (1-4)haloalkoxy, and R⁵ is CHO, (1-6)alkyl!carbonyl, (2-6)alkenyl!carbonyl, (2-6)alkynyl!carbonyl, (1-6)alkylsulfonyl, (2-6)alkenylsulfonyl, (2-6)alkynylsulfonyl, !(3-6)cycloalkyl!carbonyl, (3-6)cycloalkenylsulfonyl, each of the last 10 radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (1-4)alkyl!-carbonyl, (1-4)alkoxy!carbonyl, (1-4)alkyl!carbonyloxy and CN and in the case of cyclic radicals also (1-4)alkyl and (1-4)haloalkyl, or phenylcarbonyl or phenylsulfonyl, each of the last two radicals being unsubstituted in the phenyl ring or substituted by one or more radicals from the group consisting of halogen, CN, NO₂, (1-4)alkyl, (1-4)haloalkyl, (1-4)alkoxy and (1-4)haloalkoxy, or mono- or di- (1-4)alkyl!aminosulfonyl which is unsubstituted in the alkyl moiety or substituted by one or more radicals from the group consisting of halogen, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkylsulfinyl, (1-4)alkyl!-carbonyl, (1-4)alkyl!carbonyloxy, (1-4)alkoxy!carbonyl and CN or a group of the formula COCOR' where R'=H, OH, (1-4)alkoxy or (1-4)alkyl, or a group of the formula 1290 ##STR255## R⁴ and R⁵ together are a chain of the formula (--CH₂)_(m1) B¹ -- or --B¹ --(CH₂)_(m2) B² where individual groups CH₂ may be replaced by oxygen atoms and where the chain is unsubstituted or substituted by one or more (1-3)alkyl radicals or halogen and m1=3, 4 or 5 or m2=2, 3 or 4, and W is O or S, B¹ and B² are each independently of the other SO₂ or CO, T is O or S, R⁶ is H, (1-4)alkyl, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkyl!-carbonyl or (1-4)alkoxy!carbonyl, each of the last 5 radicals being unsubstituted or substituted in the alkyl moiety by one or more halogen atoms, or halogen, NO₂, CN or mono- or di- (1-4)alkyl!amino, R⁷ is H or (1-4)alkyl, R⁸ is (1-4)alkyl, (1-4)alkoxy, (3-6)cycloalkyl or (3-6)cycloalkenyl, R⁹ is H or (1-4)alkyl, R¹⁰ is (1-4)alkyl, (3-4)alkenyl or (3-4)alkynyl, each of the last three radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkyl!carbonyl and (1-4)alkoxy!carbonyl, R¹¹ and R¹² are each independently of the other H, (1-4)alkyl, (3-4)alkenyl or (3-4)alkynyl, each of the last three radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkyl!carbonyl and (1-4)alkoxy!carbonyl,the radicals R¹³ together with the nitrogen atom are a 5- to 6-membered heterocyclic ring which may contain further hetero atoms from the group consisting of N, O and S in the possible oxidation states and is unsubstituted or substituted by (1-4)alkyl or the oxo group or is benzo-fused.
 3. A compound or a salt thereof as claimed in claim 1, whereinR¹ is NR⁸ R⁹, (1-4)alkyl, (3-6)cycloalkyl or phenyl, each of the last 3 radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, CN, (1-4)alkoxy, (1-4)haloalkoxy, (1-4)alkylthio, (1-4)-alkylsulfonyl, formyl, (1-4)alkoxy!carbonyl, (1-4)alkyl!carbonyloxy and in the case of cyclic radicals also (1-4)alkyl, (1-4)haloalkyl and (1-4)alkoxy-(1-4)alkyl, or (2-4)alkenyl or (2-4)alkynyl, n is 0, 1 or 2, excluding n=0 or 1 if R¹ =NR⁸ R⁹, R² and R³ are each independently of the other H or (1-4)alkyl, R⁴ is H, OH, formyl, (1-4)alkyl, (2-4)alkenyl, (2-4)alkynyl, (1-4)alkoxy, (1-4)alkyl!carbonyl, (1-4)alkylsulfony, each of the last 6 radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen and (1-4)alkoxy, or phenylcarbonyl or phenysulfonyl, the phanyl ring of the last two radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (1-4)alkyl, (1-4)haloalkyl, (1-4)alkoxy and (1-4)haloalkoxy, and R⁵ is CHO, (1-4)alkyl!carbonyl, (2-4)alkenyl!carbonyl, (2-4)alkynyl!carbonyl, (1-4)alkylsulfonyl, (2-4)alkenylsulfonyl, (2-4)alkynylsulfonyl, (3-6)cycloalkyl!carbonyl, each of the last 7 radicals being unsubstituted or substituted by one or more radicals from the group consisting of halogen, (1-4)alkoxy, (1-4)alkylthio, (1-4)alkoxy!carbonyl, (1-4)alkyl!-carbonyloxy and CN and in the case of cyclic radicals also (1-4)alkyl and (1-4)haloalkyl, or phenylcarbonyl or phenylsulfonyl, each of the last two radicals being unsubstituted in the phenyl ring or substituted by one or more radicals from the group consisting of halogen, CN, NO₂, (1-4)alkyl, (1-4)haloalkyl, (1-4)alkoxy and (1-4)haloalkoxy, or mono- or di- (1-4)alkyl!aminosulfonyl which is unsubstituted in the alkyl moiety or substituted by one or more halogen atoms, or a group of the formula COCOR' where R'=H, OH, (1-4)alkoxy or (1-4)alkyl, or a group of the formula ##STR256## or R⁴ and R⁵ together are a chain of the formula (--CH₂)_(m1) B¹ -- or --B¹ --(CH₂)_(m2) B² --, where individual groups CH₂ may be replaced by oxygen atoms and where the chain is unsubstituted or substituted by one or more (1-3)alkyl radicals or halogen and m1=3, 4 or 5 or m2=2, 3 or 4, and W is O or S, B¹ and B² are each independently of the other SO₂ or CO, are each independently of the other SO₂ or CO, T is O or S, R⁶ is H, (1-4)alkyl, (1-4)alkoxy or halogen, R⁷ is H or CH₃, R⁸ is (1-4)alkyl, R⁹ is H or (1-4)alkyl, R¹⁰ is (1-4)alkyl, (1-4)haloalkyl, (3-4)alkenyl or (3-4)alkynyl, R¹¹ and R¹² are each independently of the other H or (1-4)alkyl, the radicals R¹³ together are an alkylene chain having 4 or 5 carbon atoms, A is a radical of the formula ##STR257## one of the radicals X and Y being (1-3)alkyl, halo(1-3)alkyl, (1-3)alkoxy or halo(1-3)alkoxy and the other of the radicals X and Y being (1-3)alkyl, halo(1-3)alkyl, (1-3)alkoxy, halo(1-3)alkoxy, halogen, mono- or di- (1-3)alkyl!amino and Z is CH or N.
 4. A compound or a salt thereof as claimed in claim 1, whereinR¹ is mono- or di- (1-4)alkyl!amino or (1-4)alkyl, n is 2, R² and R³ are each hydrogen, R⁴ is H or (1-4)alkyl, R⁵ is CHO, (1-4)alkyl!carbonyl, (1-4)haloalkyl!carbonyl, (1-4)alkylsulfonyl, (1-4)haloalkylsulfonyl, (1-4)alkoxy!-carbonyl, mono- or di- (1-4)alkyl!aminocarbonyl, mono- or di- (1-4)alkyl!aminosulfonyl or R⁴ and R⁵ together are a chain of the formula (--CH₂)_(m1) B¹ -- or --B¹ --(CH₂)_(m2) B² -- where B¹ and B² independently of each other are SO₂ or CO, W and T are each O, R⁶ is H and R⁷ is H or CH₃.
 5. A process for preparing compounds of the formula (I) or salts thereof as defined in claim 1, which comprisesa) reacting a compound of the formula (II) ##STR258## with a heterocyclic carbamate of the formula (III),

    R*--O--CO--NR.sup.7 --A                                    (III)

where R* is unsubstituted or substituted phenyl or (1-4)alkyl, or b) reacting an arylsulfonylcarbamate of the formula (IV) ##STR259## where Ar is an aryl radical, with an amino heterocycle of the formula (V)

    H--NR.sup.7 --A                                            (V)

or c) reacting a sulfonyl isocyanate of the formula (VI) ##STR260## with an amino heterocycle of the formula H--NR⁷ --A (V), or d) reacting in a one-pot reaction first an amino heterocycle of the formula H--NR⁷ --A (V) in the presence of a base with phosgene and then the intermediate formed with a phenylsulfonamide of the formula (II), or e) reacting a sulfonyl chloride of the formula (VII) ##STR261## with a cyanate M--OCN where M=a cation and with an amino heterocycle of the formula H--R⁷ --A (V) in the presence of a base, or f) reacting a sulfonamide of the formula (II) mentioned with a (thio)isocyanate of the formula (V')

    W=C=N--A                                                   (V')

in the presence of a base, where the radicals or symbols R¹ to R⁷, A, W and n in the formulae (II)-(VII) and (V') are as defined in formula (I) and where the compounds initially obtained in variants a) and c)-e) are compounds of the formula (I) where W=O.
 6. A herbicidal or plant growth regulating composition, which comprises one or more compounds of the formula (I) or a salt thereof as claimed in claim 1 and formulation auxiliaries customary in crop protection.
 7. A method for controlling harmful plants or for regulating the growth of plants, which comprises applying an active amount of one or more compounds of the formula (I) or a salt thereof as claimed in claim 1 to the plants, plant seeds or to the area cultivated. 